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Published in Frontiers in immunology (20.06.2018)
Published in Frontiers in immunology (20.06.2018)
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Chemical Proteomics and Phenotypic Profiling Identifies the Aryl Hydrocarbon Receptor as a Molecular Target of the Utrophin Modulator Ezutromid
Wilkinson, Isabel V. L., Perkins, Kelly J., Dugdale, Hannah, Moir, Lee, Vuorinen, Aini, Chatzopoulou, Maria, Squire, Sarah E., Monecke, Sebastian, Lomow, Alexander, Geese, Marcus, Charles, Philip D., Burch, Peter, Tinsley, Jonathan M., Wynne, Graham M., Davies, Stephen G., Wilson, Francis X., Rastinejad, Fraydoon, Mohammed, Shabaz, Davies, Kay E., Russell, Angela J.
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The BET inhibitor CPI203 promotes ex vivo expansion of cord blood long-term repopulating HSCs and megakaryocytes
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Identification and Preliminary Structure-Activity Relationship Studies of 1,5-Dihydrobenzo[ e ][1,4]oxazepin-2(3 H )-ones That Induce Differentiation of Acute Myeloid Leukemia Cells In Vitro
Josa-Culleré, Laia, Cogswell, Thomas J, Georgiou, Irene, Jay-Smith, Morgan, Jackson, Thomas R, Bataille, Carole J R, Davies, Stephen G, Vyas, Paresh, Milne, Thomas A, Wynne, Graham M, Russell, Angela J
Published in Molecules (Basel, Switzerland) (02.11.2021)
Published in Molecules (Basel, Switzerland) (02.11.2021)
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From diagnosis to therapy in Duchenne muscular dystrophy
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Published in Biochemical Society transactions (30.06.2020)
Published in Biochemical Society transactions (30.06.2020)
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Second-generation compound for the modulation of utrophin in the therapy of DMD
Guiraud, Simon, Squire, Sarah E, Edwards, Benjamin, Chen, Huijia, Burns, David T, Shah, Nandini, Babbs, Arran, Davies, Stephen G, Wynne, Graham M, Russell, Angela J, Elsey, David, Wilson, Francis X, Tinsley, Jon M, Davies, Kay E
Published in Human molecular genetics (01.08.2015)
Published in Human molecular genetics (01.08.2015)
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2,4-Diaminothieno[3,2-d]pyrimidines, a new class of anthelmintic with activity against adult and egg stages of whipworm
Partridge, Frederick A, Forman, Ruth, Willis, Nicky J, Bataille, Carole J R, Murphy, Emma A, Brown, Anwen E, Heyer-Chauhan, Narinder, Marinič, Bruno, Sowood, Daniel J C, Wynne, Graham M, Else, Kathryn J, Russell, Angela J, Sattelle, David B
Published in PLoS neglected tropical diseases (11.07.2018)
Published in PLoS neglected tropical diseases (11.07.2018)
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Dihydrobenz[e][1,4]oxazepin-2(3H)-ones, a new anthelmintic chemotype immobilising whipworm and reducing infectivity in vivo
Partridge, Frederick A, Murphy, Emma A, Willis, Nicky J, Bataille, Carole J R, Forman, Ruth, Heyer-Chauhan, Narinder, Marinič, Bruno, Sowood, Daniel J C, Wynne, Graham M, Else, Kathryn J, Russell, Angela J, Sattelle, David B
Published in PLoS neglected tropical diseases (01.02.2017)
Published in PLoS neglected tropical diseases (01.02.2017)
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Anthelmintic drug discovery: target identification, screening methods and the role of open science
Partridge, Frederick A, Forman, Ruth, Bataille, Carole J R, Wynne, Graham M, Nick, Marina, Russell, Angela J, Else, Kathryn J, Sattelle, David B
Published in Beilstein journal of organic chemistry (02.06.2020)
Published in Beilstein journal of organic chemistry (02.06.2020)
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A Phenotypic Screen Identifies a Compound Series That Induces Differentiation of Acute Myeloid Leukemia Cells In Vitro and Shows Antitumor Effects In Vivo
Josa-Culleré, Laia, Madden, Katrina S, Cogswell, Thomas J, Jackson, Thomas R, Carter, Tom S, Zhang, Douzi, Trevitt, Graham, Davies, Stephen G, Vyas, Paresh, Wynne, Graham M, Milne, Thomas A, Russell, Angela J
Published in Journal of medicinal chemistry (11.11.2021)
Published in Journal of medicinal chemistry (11.11.2021)
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Structure-activity relationships of 2-pyrimidinecarbohydrazides as utrophin modulators for the potential treatment of Duchenne muscular dystrophy
Chatzopoulou, Maria, Conole, Daniel, Emer, Enrico, Rowley, Jessica A., Willis, Nicky J., Squire, Sarah E., Gill, Becky, Brough, Steve, Wilson, Francis X., Wynne, Graham M., Davies, Stephen G., Davies, Kay E., Russell, Angela J.
Published in Bioorganic & medicinal chemistry (01.09.2022)
Published in Bioorganic & medicinal chemistry (01.09.2022)
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An automated high-throughput system for phenotypic screening of chemical libraries on C. elegans and parasitic nematodes
Partridge, Frederick A., Brown, Anwen E., Buckingham, Steven D., Willis, Nicky J., Wynne, Graham M., Forman, Ruth, Else, Kathryn J., Morrison, Alison A., Matthews, Jacqueline B., Russell, Angela J., Lomas, David A., Sattelle, David B.
Published in International journal for parasitology -- drugs and drug resistance (01.04.2018)
Published in International journal for parasitology -- drugs and drug resistance (01.04.2018)
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A Biased Agonist at Immunometabolic Receptor GPR84 Causes Distinct Functional Effects in Macrophages
Lucy, Daniel, Purvis, Gareth S. D, Zeboudj, Lynda, Chatzopoulou, Maria, Recio, Carlota, Bataille, Carole J. R, Wynne, Graham M, Greaves, David R, Russell, Angela J
Published in ACS chemical biology (20.09.2019)
Published in ACS chemical biology (20.09.2019)
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Synthesis of SMT022357 enantiomers and in vivo evaluation in a Duchenne muscular dystrophy mouse model
Babbs, Arran, Berg, Adam, Chatzopoulou, Maria, Davies, Kay E., Davies, Stephen G., Edwards, Benjamin, Elsey, David J., Emer, Enrico, Figuccia, Aude L.A., Fletcher, Ai M., Guiraud, Simon, Harriman, Shawn, Moir, Lee, Robinson, Neil, Rowley, Jessica A., Russell, Angela J., Squire, Sarah E., Thomson, James E., Tinsley, Jonathon M., Wilson, Francis X., Wynne, Graham M.
Published in Tetrahedron (10.01.2020)
Published in Tetrahedron (10.01.2020)
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Phenotypic screening identifies a trisubstituted imidazo[1,2-a]pyridine series that induces differentiation in multiple AML cell lines
Josa-Culleré, Laia, Galan, Sébastien R.G., Cogswell, Thomas J., Jackson, Thomas R., Jay-Smith, Morgan, Mola, Laura, Greaves, Christopher R., Carter, Tom S., Madden, Katrina S., Trott, Sophie, Zhang, Douzi, Bataille, Carole J.R., Davies, Stephen G., Vyas, Paresh, Milne, Thomas A., Naylor, Alan, Wynne, Graham M., Russell, Angela J.
Published in European journal of medicinal chemistry (05.10.2023)
Published in European journal of medicinal chemistry (05.10.2023)
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2‑Arylbenzo[d]oxazole Phosphinate Esters as Second-Generation Modulators of Utrophin for the Treatment of Duchenne Muscular Dystrophy
Babbs, Arran, Berg, Adam, Chatzopoulou, Maria, Davies, Kay E, Davies, Stephen G, Edwards, Benjamin, Elsey, David J, Emer, Enrico, Guiraud, Simon, Harriman, Shawn, Lecci, Cristina, Moir, Lee, Peters, David, Robinson, Neil, Rowley, Jessica A, Russell, Angela J, Squire, Sarah E, Tinsley, Jonathon M, Wilson, Francis X, Wynne, Graham M
Published in Journal of medicinal chemistry (23.07.2020)
Published in Journal of medicinal chemistry (23.07.2020)
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Thiazolidine derivatives as potent and selective inhibitors of the PIM kinase family
Bataille, Carole J.R., Brennan, Méabh B., Byrne, Simon, Davies, Stephen G., Durbin, Matthew, Fedorov, Oleg, Huber, Kilian V.M., Jones, Alan M., Knapp, Stefan, Liu, Gu, Nadali, Anna, Quevedo, Camilo E., Russell, Angela J., Walker, Roderick G., Westwood, Robert, Wynne, Graham M.
Published in Bioorganic & medicinal chemistry (01.05.2017)
Published in Bioorganic & medicinal chemistry (01.05.2017)
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Efficacy of a series of alpha-pyrone derivatives against Leishmania (L.) infantum and Trypanosoma cruzi
Tempone, Andre Gustavo, Ferreira, Daiane Dias, Lima, Marta Lopes, Costa Silva, Thais Alves, Borborema, Samanta E.T., Reimão, Juliana Quero, Galuppo, Mariana K., Guerra, Juliana Mariotti, Russell, Angelie J., Wynne, Graham M., Lai, Roy Y.L., Cadelis, Melissa M., Copp, Brent R.
Published in European journal of medicinal chemistry (20.10.2017)
Published in European journal of medicinal chemistry (20.10.2017)
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Pilot Study to Quantify Palladium Impurities in Lead-like Compounds Following Commonly Used Purification Techniques
Chatzopoulou, Maria, Madden, Katrina S, Bromhead, Liam J, Greaves, Christopher, Cogswell, Thomas J, Da Silva Pinto, Solange, Galan, Sébastien R G, Georgiou, Irene, Kennedy, Matthew S, Kennett, Alice, Apps, Geraint, Russell, Angela J, Wynne, Graham M
Published in ACS medicinal chemistry letters (10.02.2022)
Published in ACS medicinal chemistry letters (10.02.2022)
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Discovery and mechanism of action studies of 4,6-diphenylpyrimidine-2-carbohydrazides as utrophin modulators for the treatment of Duchenne muscular dystrophy
Vuorinen, Aini, Wilkinson, Isabel V.L., Chatzopoulou, Maria, Edwards, Ben, Squire, Sarah E., Fairclough, Rebecca J., Bazan, Noelia Araujo, Milner, Josh A., Conole, Daniel, Donald, James R., Shah, Nandini, Willis, Nicky J., Martínez, R. Fernando, Wilson, Francis X., Wynne, Graham M., Davies, Stephen G., Davies, Kay E., Russell, Angela J.
Published in European journal of medicinal chemistry (05.08.2021)
Published in European journal of medicinal chemistry (05.08.2021)
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