Synthesis of a Novel Disubstituted Indole
Wright, Stephen W. W., Gribble, Gordon W. W.
Published in Organic preparations and procedures international (03.09.2023)
Published in Organic preparations and procedures international (03.09.2023)
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Journal Article
Discovery of a Series of Pyrimidine Carboxamides as Inhibitors of Vanin‑1
Casimiro-Garcia, Agustin, Allais, Christophe, Brennan, Agnes, Choi, Chulho, Dower, Gabriela, Farley, Kathleen A, Fleming, Margaret, Flick, Andrew, Frisbie, Richard K, Hall, Justin, Hepworth, David, Jones, Hannah, Knafels, John D, Kortum, Steve, Lovering, Frank E, Mathias, John P, Mohan, Sashi, Morgan, Paul M, Parng, Chuenlei, Parris, Kevin, Pullen, Nick, Schlerman, Franklin, Stansfield, John, Strohbach, Joseph W, Vajdos, Felix F, Vincent, Fabien, Wang, Hong, Wang, Xiaolun, Webster, Robert, Wright, Stephen W
Published in Journal of medicinal chemistry (13.01.2022)
Published in Journal of medicinal chemistry (13.01.2022)
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Journal Article
Aminocarbonylation of Aryl Tosylates to Carboxamides
Chung, Seungwon, Sach, Neal, Choi, Chulho, Yang, Xiaojing, Drozda, Susan E, Singer, Robert A, Wright, Stephen W
Published in Organic letters (05.06.2015)
Published in Organic letters (05.06.2015)
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Journal Article
Distinct signals and immune cells drive liver pathology and glomerulonephritis in ABIN1[D485N] mice
Nanda, Sambit Kumar, Petrova, Tsvetana, Marchesi, Francesco, Gierlinski, Marek, Razsolkov, Momchil, Lee, Katherine L, Wright, Stephen W, Rao, Vikram R, Cohen, Philip, Arthur, J Simon C
Published in Life science alliance (01.12.2019)
Published in Life science alliance (01.12.2019)
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Journal Article
Small Change, Big Impact: Reversal of Diastereoselection in Cuprate Conjugate Additions to α,β-Unsaturated Lactams and Identification of a Competing Mechanism
Wright, Stephen W., Choi, Chulho, Kawamata, Yu, Baran, Phil S.
Published in Journal of organic chemistry (07.04.2023)
Published in Journal of organic chemistry (07.04.2023)
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Journal Article
Discovery of Tyrosine Kinase 2 (TYK2) Inhibitor (PF-06826647) for the Treatment of Autoimmune Diseases
Gerstenberger, Brian S, Ambler, Catherine, Arnold, Eric P, Banker, Mary-Ellen, Brown, Matthew F, Clark, James D, Dermenci, Alpay, Dowty, Martin E, Fensome, Andrew, Fish, Susan, Hayward, Matthew M, Hegen, Martin, Hollingshead, Brett D, Knafels, John D, Lin, David W, Lin, Tsung H, Owen, Dafydd R, Saiah, Eddine, Sharma, Raman, Vajdos, Felix F, Xing, Li, Yang, Xiaojing, Yang, Xin, Wright, Stephen W
Published in Journal of medicinal chemistry (25.11.2020)
Published in Journal of medicinal chemistry (25.11.2020)
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Discovery of Clinical Candidate 1‑{[(2S,3S,4S)‑3-Ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide (PF-06650833), a Potent, Selective Inhibitor of Interleukin‑1 Receptor Associated Kinase 4 (IRAK4), by Fragment-Based Drug Design
Lee, Katherine L, Ambler, Catherine M, Anderson, David R, Boscoe, Brian P, Bree, Andrea G, Brodfuehrer, Joanne I, Chang, Jeanne S, Choi, Chulho, Chung, Seungwon, Curran, Kevin J, Day, Jacqueline E, Dehnhardt, Christoph M, Dower, Ken, Drozda, Susan E, Frisbie, Richard K, Gavrin, Lori K, Goldberg, Joel A, Han, Seungil, Hegen, Martin, Hepworth, David, Hope, Heidi R, Kamtekar, Satwik, Kilty, Iain C, Lee, Arthur, Lin, Lih-Ling, Lovering, Frank E, Lowe, Michael D, Mathias, John P, Morgan, Heidi M, Murphy, Elizabeth A, Papaioannou, Nikolaos, Patny, Akshay, Pierce, Betsy S, Rao, Vikram R, Saiah, Eddine, Samardjiev, Ivan J, Samas, Brian M, Shen, Marina W. H, Shin, Julia H, Soutter, Holly H, Strohbach, Joseph W, Symanowicz, Peter T, Thomason, Jennifer R, Trzupek, John D, Vargas, Richard, Vincent, Fabien, Yan, Jiangli, Zapf, Christoph W, Wright, Stephen W
Published in Journal of medicinal chemistry (13.07.2017)
Published in Journal of medicinal chemistry (13.07.2017)
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Journal Article
cis-2,5-Dicyanopyrrolidine Inhibitors of Dipeptidyl Peptidase IV: Synthesis and in Vitro, in Vivo, and X-ray Crystallographic Characterization
Wright, Stephen W, Ammirati, Mark J, Andrews, Kim M, Brodeur, Anne M, Danley, Dennis E, Doran, Shawn D, Lillquist, Jay S, McClure, Lester D, McPherson, R. Kirk, Orena, Stephen J, Parker, Janice C, Polivkova, Jana, Qiu, Xiayang, Soeller, Walter C, Soglia, Carolyn B, Treadway, Judith L, VanVolkenburg, Maria A, Wang, Hong, Wilder, Donald C, Olson, Thanh V
Published in Journal of medicinal chemistry (01.06.2006)
Published in Journal of medicinal chemistry (01.06.2006)
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Journal Article
Improvements to Enable the Large Scale Synthesis of 1‑{[(2S,3S,4S)-3-Ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide (PF-06650833)
Wright, Stephen W, Li, Bryan, Peng, Zhihui, Wei, Lulin, McInturff, Emma, Place, David, Damon, David B, Singer, Robert A
Published in Organic process research & development (21.12.2018)
Published in Organic process research & development (21.12.2018)
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Identification of Morpholino‑2H‑pyrido[3,2‑b][1,4]oxazin-3(4H)‑ones as Nonsteroidal Mineralocorticoid Antagonists
Piotrowski, David W, Futatsugi, Kentaro, Casimiro-Garcia, Agustin, Wei, Liuqing, Sammons, Matthew F, Herr, Michael, Jiao, Wenhua, Lavergne, Sophie Y, Coffey, Steven B, Wright, Stephen W, Song, Kun, Loria, Paula M, Banker, Mary Ellen, Petersen, Donna N, Bauman, Jonathan
Published in Journal of medicinal chemistry (08.02.2018)
Published in Journal of medicinal chemistry (08.02.2018)
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Journal Article
Synthesis of Chiral Azabicycles from Pyroglutaminols
Choi, Chulho, Nuhant, Philippe, Mousseau, James J, Yang, Xiaojing, Gerstenberger, Brian S, Williams, Jessica M, Wright, Stephen W
Published in Organic letters (04.11.2016)
Published in Organic letters (04.11.2016)
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Journal Article
Binding site elucidation and structure guided design of macrocyclic IL-17A antagonists
Liu, Shenping, Dakin, Leslie A, Xing, Li, Withka, Jane M, Sahasrabudhe, Parag V, Li, Wei, Banker, Mary Ellen, Balbo, Paul, Shanker, Suman, Chrunyk, Boris A, Guo, Zuojun, Chen, Jinshan M, Young, Jennifer A, Bai, Guoyun, Starr, Jeremy T, Wright, Stephen W, Bussenius, Joerg, Tan, Sheng, Gopalsamy, Ariamala, Lefker, Bruce A, Vincent, Fabien, Jones, Lyn H, Xu, Hua, Hoth, Lise R, Geoghegan, Kieran F, Qiu, Xiayang, Bunnage, Mark E, Thorarensen, Atli
Published in Scientific reports (16.08.2016)
Published in Scientific reports (16.08.2016)
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