MM/GBSA Binding Energy Prediction on the PDBbind Data Set: Successes, Failures, and Directions for Further Improvement
Greenidge, Paulette A, Kramer, Christian, Mozziconacci, Jean-Christophe, Wolf, Romain M
Published in Journal of chemical information and modeling (28.01.2013)
Published in Journal of chemical information and modeling (28.01.2013)
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Journal Article
Development and testing of a general amber force field
Wang, Junmei, Wolf, Romain M., Caldwell, James W., Kollman, Peter A., Case, David A.
Published in Journal of computational chemistry (15.07.2004)
Published in Journal of computational chemistry (15.07.2004)
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Journal Article
Discovery of Amino Alcohols as Highly Potent, Selective, and Orally Efficacious Inhibitors of Leukotriene A4 Hydrolase
Thoma, Gebhard, Markert, Christian, Lueoend, Rainer, Miltz, Wolfgang, Spanka, Carsten, Bollbuck, Birgit, Wolf, Romain M., Srinivas, Honnappa, Penno, Carlos A., Kiffe, Michael, Gajewska, Monika, Bednarczyk, Dallas, Wieczorek, Grazyna, Evans, Amanda, Beerli, Christian, Röhn, Till A.
Published in Journal of medicinal chemistry (14.12.2023)
Published in Journal of medicinal chemistry (14.12.2023)
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Journal Article
Discovery of CDZ173 (Leniolisib), Representing a Structurally Novel Class of PI3K Delta-Selective Inhibitors
Hoegenauer, Klemens, Soldermann, Nicolas, Zécri, Frédéric, Strang, Ross S, Graveleau, Nadege, Wolf, Romain M, Cooke, Nigel G, Smith, Alexander B, Hollingworth, Gregory J, Blanz, Joachim, Gutmann, Sascha, Rummel, Gabriele, Littlewood-Evans, Amanda, Burkhart, Christoph
Published in ACS medicinal chemistry letters (14.09.2017)
Published in ACS medicinal chemistry letters (14.09.2017)
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Journal Article
Optimizing a Weakly Binding Fragment into a Potent RORγt Inverse Agonist with Efficacy in an in Vivo Inflammation Model
Carcache, David A, Vulpetti, Anna, Kallen, Joerg, Mattes, Henri, Orain, David, Stringer, Rowan, Vangrevelinghe, Eric, Wolf, Romain M, Kaupmann, Klemens, Ottl, Johannes, Dawson, Janet, Cooke, Nigel G, Hoegenauer, Klemens, Billich, Andreas, Wagner, Juergen, Guntermann, Christine, Hintermann, Samuel
Published in Journal of medicinal chemistry (09.08.2018)
Published in Journal of medicinal chemistry (09.08.2018)
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Journal Article
Feasibility and physiological relevance of designing highly potent aminopeptidase-sparing leukotriene A4 hydrolase inhibitors
Numao, Shin, Hasler, Franziska, Laguerre, Claire, Srinivas, Honnappa, Wack, Nathalie, Jäger, Petra, Schmid, Andres, Osmont, Arnaud, Röthlisberger, Patrik, Houguenade, Jeremy, Bergsdorf, Christian, Dawson, Janet, Carte, Nathalie, Hofmann, Andreas, Markert, Christian, Hardaker, Liz, Billich, Andreas, Wolf, Romain M, Penno, Carlos A, Bollbuck, Birgit, Miltz, Wolfgang, Röhn, Till A
Published in Scientific reports (19.10.2017)
Published in Scientific reports (19.10.2017)
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Journal Article
Discovery of novel pyrrolidineoxy-substituted heteroaromatics as potent and selective PI3K delta inhibitors with improved physicochemical properties
Hoegenauer, Klemens, Soldermann, Nicolas, Hebach, Christina, Hollingworth, Gregory J., Lewis, Ian, von Matt, Anette, Smith, Alexander B., Wolf, Romain M., Wilcken, Rainer, Haasen, Dorothea, Burkhart, Christoph, Zécri, Frédéric
Published in Bioorganic & medicinal chemistry letters (01.12.2016)
Published in Bioorganic & medicinal chemistry letters (01.12.2016)
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Journal Article
Discovery and Pharmacological Characterization of Novel Quinazoline-Based PI3K Delta-Selective Inhibitors
Hoegenauer, Klemens, Soldermann, Nicolas, Stauffer, Frédéric, Furet, Pascal, Graveleau, Nadege, Smith, Alexander B, Hebach, Christina, Hollingworth, Gregory J, Lewis, Ian, Gutmann, Sascha, Rummel, Gabriele, Knapp, Mark, Wolf, Romain M, Blanz, Joachim, Feifel, Roland, Burkhart, Christoph, Zécri, Frédéric
Published in ACS medicinal chemistry letters (11.08.2016)
Published in ACS medicinal chemistry letters (11.08.2016)
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Journal Article
Proton-sensing G-protein-coupled receptors
Seuwen, Klaus, Ludwig, Marie-Gabrielle, Vanek, Miroslava, Guerini, Danilo, Gasser, Jürg A, Jones, Carol E, Junker, Uwe, Hofstetter, Hans, Wolf, Romain M
Published in Nature (04.09.2003)
Published in Nature (04.09.2003)
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Journal Article
Molecular Characterization of Oxysterol Binding to the Epstein-Barr Virus-induced Gene 2 (GPR183)
Benned-Jensen, Tau, Norn, Christoffer, Laurent, Stephane, Madsen, Christian M., Larsen, Hjalte M., Arfelt, Kristine N., Wolf, Romain M., Frimurer, Thomas, Sailer, Andreas W., Rosenkilde, Mette M.
Published in The Journal of biological chemistry (12.10.2012)
Published in The Journal of biological chemistry (12.10.2012)
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Journal Article
Homology Modeling of the Transmembrane Domain of the Human Calcium Sensing Receptor and Localization of an Allosteric Binding Site
Miedlich, Susanne U., Gama, Lucio, Seuwen, Klaus, Wolf, Romain M., Breitwieser, Gerda E.
Published in The Journal of biological chemistry (20.02.2004)
Published in The Journal of biological chemistry (20.02.2004)
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Journal Article
Receptors for protons or lipid messengers or both?
Seuwen, Klaus, Ludwig, Marie-Gabrielle, Wolf, Romain M
Published in Journal of receptors and signal transduction (2006)
Published in Journal of receptors and signal transduction (2006)
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Journal Article
1-Alkyl-4-phenyl-6-alkoxy-1H-quinazolin-2-ones: A Novel Series of Potent Calcium-Sensing Receptor Antagonists
Widler, Leo, Altmann, Eva, Beerli, René, Breitenstein, Werner, Bouhelal, Rochdi, Buhl, Thomas, Gamse, Rainer, Gerspacher, Marc, Halleux, Christine, John, Markus R, Lehmann, Hansjoerg, Kalb, Oskar, Kneissel, Michaela, Missbach, Martin, Müller, Irene R, Reidemeister, Sibylle, Renaud, Johanne, Taillardat, Agnes, Tommasi, Ruben, Weiler, Sven, Wolf, Romain M, Seuwen, Klaus
Published in Journal of medicinal chemistry (11.03.2010)
Published in Journal of medicinal chemistry (11.03.2010)
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Journal Article
Dual Recognition of Double-Stranded DNA by 2′-Aminoethoxy-Modified Oligonucleotides
Cuenoud, Bernard, Casset, Florence, Hüsken, Dieter, Natt, François, Wolf, Romain M., Altmann, Karl-Heinz, Martin, Pierre, Moser, Heinz E.
Published in Angewandte Chemie (International ed.) (18.05.1998)
Published in Angewandte Chemie (International ed.) (18.05.1998)
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Journal Article
Comparison of pure epoxy vs. epoxy-anhydride photopolymerization
Kavalli, Tuba, Wolf, Romain, Ozen, Serife, Lalevée, Jacques
Published in European polymer journal (05.03.2022)
Published in European polymer journal (05.03.2022)
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Journal Article
Ultrafast Epoxy‐Anhydride Photopolyaddition Reaction
Kavalli, Tuba, Wolf, Romain, Lalevée, Jacques
Published in Macromolecular chemistry and physics (01.10.2020)
Published in Macromolecular chemistry and physics (01.10.2020)
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