Optimization of biaryl Selective HDAC1&2 Inhibitors (SHI-1:2)
Witter, David J., Harrington, Paul, Wilson, Kevin J., Chenard, Melissa, Fleming, Judith C., Haines, Brian, Kral, Astrid M., Secrist, J. Paul, Miller, Thomas A.
Published in Bioorganic & medicinal chemistry (15.01.2008)
Published in Bioorganic & medicinal chemistry (15.01.2008)
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Journal Article
Histone Deacetylase Inhibitors
Miller, Thomas A, Witter, David J, Belvedere, Sandro
Published in Journal of medicinal chemistry (20.11.2003)
Published in Journal of medicinal chemistry (20.11.2003)
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Journal Article
Exploring the pharmacokinetic properties of phosphorus-containing selective HDAC 1 and 2 inhibitors (SHI-1:2)
HEIDEBRECHT, Richard W, CHENARD, Melissa, KRAL, Astrid M, MIDDLETON, Richard E, MUSHTI, Chandrasekhar, OZEROVA, Nicole, SZEWCZAK, Alexander A, HONGMEI WANG, WILSON, Kevin, WITTER, David J, SECRIST, J. Paul, MILLER, Thomas A, CLOSE, Joshua, DAHLBERG, William K, FLEMING, Judith, GRIMM, Jonathan B, HAMILL, Julie E, HARSCH, Andreas, HAINES, Brian B, HUGHES, Bethany
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
Published in Bioorganic & medicinal chemistry letters (01.04.2009)
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Journal Article
Evaluation of JAK3 Biology in Autoimmune Disease Using a Highly Selective, Irreversible JAK3 Inhibitor
Elwood, Fiona, Witter, David J, Piesvaux, Jennifer, Kraybill, Brian, Bays, Nathan, Alpert, Carla, Goldenblatt, Peter, Qu, Yujie, Ivanovska, Irena, Lee, Hyun-Hee, Chiu, Chi-Sung, Tang, Hao, Scott, Mark E, Deshmukh, Sujal V, Zielstorff, Mark, Byford, Alan, Chakravarthy, Kalyan, Dorosh, Lauren, Rivkin, Alexey, Klappenbach, Joel, Pan, Bo-Sheng, Kariv, Ilona, Dinsmore, Christopher, Slipetz, Deborah, Dandliker, Peter J
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2017)
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Journal Article
Exploration of the internal cavity of histone deacetylase (HDAC) with selective HDAC1/HDAC2 inhibitors (SHI-1:2)
Methot, Joey L., Chakravarty, Prasun K., Chenard, Melissa, Close, Joshua, Cruz, Jonathan C., Dahlberg, William K., Fleming, Judith, Hamblett, Christopher L., Hamill, Julie E., Harrington, Paul, Harsch, Andreas, Heidebrecht, Richard, Hughes, Bethany, Jung, Joon, Kenific, Candia M., Kral, Astrid M., Meinke, Peter T., Middleton, Richard E., Ozerova, Nicole, Sloman, David L., Stanton, Matthew G., Szewczak, Alexander A., Tyagarajan, Sriram, Witter, David J., Paul Secrist, J., Miller, Thomas A.
Published in Bioorganic & medicinal chemistry (01.02.2008)
Published in Bioorganic & medicinal chemistry (01.02.2008)
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Journal Article
Lovastatin Nonaketide Synthase Catalyzes an Intramolecular Diels−Alder Reaction of a Substrate Analogue
Auclair, Karine, Sutherland, Andrew, Kennedy, Jonathan, Witter, David J, Van den Heever, Johan P, Hutchinson, C. Richard, Vederas, John C
Published in Journal of the American Chemical Society (22.11.2000)
Published in Journal of the American Chemical Society (22.11.2000)
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Journal Article
Delayed and Prolonged Histone Hyperacetylation with a Selective HDAC1/HDAC2 Inhibitor
Methot, Joey L, Hoffman, Dawn Mampreian, Witter, David J, Stanton, Matthew G, Harrington, Paul, Hamblett, Christopher, Siliphaivanh, Phieng, Wilson, Kevin, Hubbs, Jed, Heidebrecht, Richard, Kral, Astrid M, Ozerova, Nicole, Fleming, Judith C, Wang, Hongmei, Szewczak, Alexander A, Middleton, Richard E, Hughes, Bethany, Cruz, Jonathan C, Haines, Brian B, Chenard, Melissa, Kenific, Candia M, Harsch, Andreas, Secrist, J. Paul, Miller, Thomas A
Published in ACS medicinal chemistry letters (10.04.2014)
Published in ACS medicinal chemistry letters (10.04.2014)
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Journal Article
Benzo[b]thiophene-based histone deacetylase inhibitors
Witter, David J., Belvedere, Sandro, Chen, Liqiang, Secrist, J. Paul, Mosley, Ralph T., Miller, Thomas A.
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
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Journal Article
Design of novel histone deacetylase inhibitors
Siliphaivanh, Phieng, Harrington, Paul, Witter, David J., Otte, Karin, Tempest, Paul, Kattar, Sam, Kral, Astrid M., Fleming, Judith C., Deshmukh, Sujal V., Harsch, Andreas, Secrist, Paul J., Miller, Thomas A.
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
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Journal Article
PRMT5 억제제
KAWAMURA SHUHEI, WITTER DAVID J, MACHACEK MICHELLE, ALTMAN MICHAEL D, GIBEAU CRAIG R, SLOMAN DAVID L
Year of Publication 17.08.2022
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Year of Publication 17.08.2022
Patent
Phenylglycine and phenylalanine derivatives as potent and selective HDAC1 inhibitors (SHI-1)
WILSON, Kevin J, WITTER, David J, CHENARD, Melissa, SZEWCZAK, Alexander A, MIDDLETON, Richard E, HUGHES, Bethany L, DAHLBERG, William K, SECRIST, J. Paul, MILLER, Thomas A, GRIMM, Jonathan B, SILIPHAIVANH, Phieng, OTTE, Karin M, KRAL, Astrid M, FLEMING, Judith C, HARSCH, Andreas, HAMILL, Julie E, CRUZ, Jonathan C
Published in Bioorganic & medicinal chemistry letters (01.03.2008)
Published in Bioorganic & medicinal chemistry letters (01.03.2008)
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Journal Article
PRMT5 억제제
REUTERSHAN MICHAEL H, WITTER DAVID J, MACHACEK MICHELLE, HUANG CHUNHUI, ALTMAN MICHAEL D, GIBEAU CRAIG R, SLOMAN DAVID L
Year of Publication 06.09.2022
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Year of Publication 06.09.2022
Patent
Phenylglycine and phenylalanine derivatives as potent and selective HDAC1 inhibitors (SHI-1)
Wilson, Kevin J, Witter, David J, Grimm, Jonathan B, Siliphaivanh, Phieng, Otte, Karin M, Kral, Astrid M, Fleming, Judith C, Harsch, Andreas, Hamill, Julie E, Cruz, Jonathan C, Chenard, Melissa, Szewczak, Alexander A, Middleton, Richard E, Hughes, Bethany L, Dahlberg, William K, Secrist, J Paul, Miller, Thomas A
Published in Bioorganic & medicinal chemistry (15.03.2008)
Published in Bioorganic & medicinal chemistry (15.03.2008)
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Journal Article
NOVEL COMPOUNDS THAT ARE ERK INHIBITORS
WITTER DAVID J, O'BOYLE BRENDAN, BOYCE CHRISTOPHER, KURUKULASURIYA RAVI, SLOMAN DAVID, TONG LING, SHINKRE BIDHAN A, THATAI JAYANTH THIRUVELLORE, SILIPHAIVANH PHIENG, FALCONE DANIELLE, MANSOOR UMAR FARUK, ZHOU WEI, KARUNAKARAN GANESH BABU, FEVRIER SALEM, LIPFORD KATHRYN, METHOT JOEY L, CHEN LEI, MALETIC MILANA M, HUANG XIANHAI, KOZLOWSKI JOSEPH, DANIELS MATTHEW H, LIM, JONG WON, WILSON KEVIN J, BAKSHI RAMAN KUMAR
Year of Publication 03.06.2015
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Year of Publication 03.06.2015
Patent