Xanthine mimetics as potent dipeptidyl peptidase IV inhibitors
Kurukulasuriya, Ravi, Rohde, Jeffrey J., Szczepankiewicz, Bruce G., Basha, Fatima, Lai, Chunqui, Jae, Hwan-Soo, Winn, Martin, Stewart, Kent D., Longenecker, Kenton L., Lubben, Thomas W., Ballaron, Stephen J., Sham, Hing L., von Geldern, Thomas W.
Published in Bioorganic & medicinal chemistry letters (15.12.2006)
Published in Bioorganic & medicinal chemistry letters (15.12.2006)
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Pyrrolidine-3-carboxylic Acids as Endothelin Antagonists. 4. Side Chain Conformational Restriction Leads to ETB Selectivity
von Geldern, Thomas W, Tasker, Andrew S, Sorensen, Bryan K, Winn, Martin, Szczepankiewicz, Bruce G, Dixon, Douglas B, Chiou, William J, Wang, Liming, Wessale, Jerry L, Adler, Andy, Marsh, Kennan C, Nguyen, Bach, Opgenorth, Terry J
Published in Journal of medicinal chemistry (09.09.1999)
Published in Journal of medicinal chemistry (09.09.1999)
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Discovery of Novel p-Arylthio Cinnamides as Antagonists of Leukocyte Function-Associated Antigen-1/Intercellular Adhesion Molecule-1 Interaction. 4. Structure−Activity Relationship of Substituents on the Benzene Ring of the Cinnamide
Winn, Martin, Reilly, Edward B, Liu, Gang, Huth, Jeffrey R, Jae, Hwan-Soo, Freeman, Jennifer, Pei, Zhonghua, Xin, Zhili, Lynch, John, Kester, Jeff, von Geldern, Thomas W, Leitza, Sandra, DeVries, Peter, Dickinson, Robert, Mussatto, Donna, Okasinski, Gregory F
Published in Journal of medicinal chemistry (06.12.2001)
Published in Journal of medicinal chemistry (06.12.2001)
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Phaser crystallographic software
McCoy, Airlie J., Grosse-Kunstleve, Ralf W., Adams, Paul D., Winn, Martyn D., Storoni, Laurent C., Read, Randy J.
Published in Journal of applied crystallography (01.08.2007)
Published in Journal of applied crystallography (01.08.2007)
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Potent and Selective Non-Benzodioxole-Containing Endothelin-A Receptor Antagonists
Tasker, Andrew S, Sorensen, Bryan K, Jae, Hwan-Soo, Winn, Martin, von Geldern, Thomas W, Dixon, Douglas B, Chiou, William J, Dayton, Brian D, Calzadila, Samuel, Hernandez, Lisa, Marsh, Kennan C, WuWong, J. Ruth, Opgenorth, Terry J
Published in Journal of medicinal chemistry (31.01.1997)
Published in Journal of medicinal chemistry (31.01.1997)
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Adamantane sulfone and sulfonamide 11-β-HSD1 Inhibitors
Sorensen, Bryan, Winn, Martin, Rohde, Jeff, Shuai, Qi, Wang, Jiahong, Fung, Steven, Monzon, Katina, Chiou, William, Stolarik, DeAnne, Imade, Hovis, Pan, Liping, Deng, Xiaoqing, Chovan, Linda, Longenecker, Kenton, Judge, Russell, Qin, Wenying, Brune, Michael, Camp, Heidi, Frevert, Ernst U., Jacobson, Peer, Link, J.T.
Published in Bioorganic & medicinal chemistry letters (15.01.2007)
Published in Bioorganic & medicinal chemistry letters (15.01.2007)
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Pyrrolidine-3-carboxylic acids as endothelin antagonists. 4. Side chain conformational restriction leads to ET(B) selectivity
von Geldern, T W, Tasker, A S, Sorensen, B K, Winn, M, Szczepankiewicz, B G, Dixon, D B, Chiou, W J, Wang, L, Wessale, J L, Adler, A, Marsh, K C, Nguyen, B, Opgenorth, T J
Published in Journal of medicinal chemistry (09.09.1999)
Published in Journal of medicinal chemistry (09.09.1999)
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Pharmacological characterization of A-127722: an orally active and highly potent ETA-selective receptor antagonist
Opgenorth, T J, Adler, A L, Calzadilla, S V, Chiou, W J, Dayton, B D, Dixon, D B, Gehrke, L J, Hernandez, L, Magnuson, S R, Marsh, K C, Novosad, E I, Von Geldern, T W, Wessale, J L, Winn, M, Wu-Wong, J R
Published in The Journal of pharmacology and experimental therapeutics (01.02.1996)
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Published in The Journal of pharmacology and experimental therapeutics (01.02.1996)
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ADAMANTYL DERIVATIVES AS INHIBITORS OF THE 11-BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 ENZYME
YEH VINCE S, YONG HONG, PATEL JYOTI R, LINK JAMES T, SHUAI QI, SORENSEN BRYAN K, WINN MARTIN, DINGES JURGEN, ROHDE JEFFREY J
Year of Publication 18.03.2013
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Year of Publication 18.03.2013
Patent
Pharmacology of endothelin receptor antagonists ABT-627, ABT-546, A-182086 and A-192621: ex vivo and in vivo studies
Wessale, Jerry L, Adler, Andrew L, Novosad, Eugene I, Calzadilla, Samuel V, Dayton, Brian D, Marsh, Kennan C, Winn, Martin, Jae, Hwan-Soo, von Geldern, Thomas W, Opgenorth, Terry J, Wu-Wong, J Ruth
Published in Clinical science (1979) (01.08.2002)
Published in Clinical science (1979) (01.08.2002)
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Transaction counterpart identification
Crudele, Marcel, Howard, Tyler, Robertson, John Michael, Crockett, Nathan, Martin, Winn, Robinson, Jason, Toloff, Andrew
Year of Publication 24.10.2023
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Year of Publication 24.10.2023
Patent
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Chelko, Jeff, Gorantla, Nikhil, Crudele, Marcel, Robertson, John Michael, Gholston, Thaddeus, Lam, Kien, Martin, Winn, Toloff, Andrew
Year of Publication 13.08.2024
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Year of Publication 13.08.2024
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Synthesis and biological evaluation of novel, selective, nonsteroidal glucocorticoid receptor antagonists
AKRITOPOULOU-ZANZE, Irini, PATEL, Jyoti R, HARTANDI, Kresna, BRENNEMAN, Jehrod, WINN, Martin, PRATT, John K, GRYNFARB, Marlene, GOOS-NISSON, Annika, VON GELDERN, Thomas W, KYM, Philip R
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
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TRANSACTION COUNTERPART IDENTIFICATION
Crudele, Marcel, Howard, Tyler, Robertson, John Michael, Crockett, Nathan, Martin, Winn, Robinson, Jason, Toloff, Andrew
Year of Publication 15.12.2022
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Year of Publication 15.12.2022
Patent
Pyrrolidine-3-carboxylic Acids as Endothelin Antagonists. 5. Highly Selective, Potent, and Orally Active ETA Antagonists
Jae, Hwan-Soo, Winn, Martin, von Geldern, Thomas W, Sorensen, Bryan K, Chiou, William J, Nguyen, Bach, Marsh, Kennan C, Opgenorth, Terry J
Published in Journal of medicinal chemistry (08.11.2001)
Published in Journal of medicinal chemistry (08.11.2001)
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Pharmacology of endothelin receptor antagonists ABT-627, ABT-546, A-182086 and A-192621: in vitro studies
Wu-Wong, J Ruth, Dixon, Douglas B, Chiou, William J, Sorensen, Brian K, Liu, Gang, Jae, H-S, Tasker, Andrew, von Geldern, Thomas W, Winn, Martin, Opgenorth, Terry J
Published in Clinical science (1979) (01.08.2002)
Published in Clinical science (1979) (01.08.2002)
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WORK INCOME VISUALIZATION AND OPTIMIZATION PLATFORM
Chelko, Jeff, Crudele, Marcel, Howard, Tyler, Hentschel, Jasmine, Shukla, Kabir, Miguel, Amanda, Martin, Winn, Nabors, Antonea
Year of Publication 10.02.2022
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Year of Publication 10.02.2022
Patent
2,4-Diarylpyrrolidine-3-carboxylic AcidsPotent ETA Selective Endothelin Receptor Antagonists. 1. Discovery of A-127722
Winn, Martin, von Geldern, Thomas W, Opgenorth, Terry J, Jae, Hwan-Soo, Tasker, Andrew S, Boyd, Steven A, Kester, Jeffrey A, Mantei, Robert A, Bal, Radhika, Sorensen, Bryan K, Wu-Wong, Jinshyun R, Chiou, William J, Dixon, Douglas B, Novosad, Eugene I, Hernandez, Lisa, Marsh, Kennan C
Published in Journal of medicinal chemistry (01.03.1996)
Published in Journal of medicinal chemistry (01.03.1996)
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