APR-246 overcomes resistance to cisplatin and doxorubicin in ovarian cancer cells
Mohell, N, Alfredsson, J, Fransson, Å, Uustalu, M, Byström, S, Gullbo, J, Hallberg, A, Bykov, V J N, Björklund, U, Wiman, K G
Published in Cell death & disease (18.06.2015)
Published in Cell death & disease (18.06.2015)
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APR-246/PRIMA-1MET inhibits thioredoxin reductase 1 and converts the enzyme to a dedicated NADPH oxidase
Peng, X, Zhang, M-Q-Z, Conserva, F, Hosny, G, Selivanova, G, Bykov, V J N, Arnér, E S J, Wiman, K G
Published in Cell death & disease (24.10.2013)
Published in Cell death & disease (24.10.2013)
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Journal Article
Mutant p53 reactivation by PRIMA-1MET induces multiple signaling pathways converging on apoptosis
Lambert, J M R, Moshfegh, A, Hainaut, P, Wiman, K G, Bykov, V J N
Published in Oncogene (04.03.2010)
Published in Oncogene (04.03.2010)
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PRIMA-1MET induces mitochondrial apoptosis through activation of caspase-2
Shen, J, Vakifahmetoglu, H, Stridh, H, Zhivotovsky, B, Wiman, K G
Published in Oncogene (30.10.2008)
Published in Oncogene (30.10.2008)
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The p53 target Wig-1: a regulator of mRNA stability and stem cell fate?
Vilborg, A, Bersani, C, Wilhelm, M T, Wiman, K G
Published in Cell death and differentiation (01.09.2011)
Published in Cell death and differentiation (01.09.2011)
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PRIMA-1Met induces mitochondrial apoptosis through activation of caspase-2
Shen, J, Vakifahmetoglu, H, Stridh, H, Zhivotovsky, B, Wiman, K G
Published in Oncogene (15.12.2016)
Published in Oncogene (15.12.2016)
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Journal Article
PRIMA-1 APR-246 targets mutant forms of p53 family members p63 and p73
Rökaeus, N, Shen, J, Eckhardt, I, Bykov, V J N, Wiman, K G, Wilhelm, M T
Published in Oncogene (09.12.2010)
Published in Oncogene (09.12.2010)
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Mutated and non‐mutated TP53 as targets in the treatment of leukaemia
Nahi, H., Selivanova, G., Lehmann, S., Möllgård, L., Bengtzen, S., Concha, H., Svensson, A., Wiman, K. G., Merup, M., Paul, C.
Published in British journal of haematology (01.05.2008)
Published in British journal of haematology (01.05.2008)
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Journal Article
Mutant p53 protein, master regulator of human malignancies: a report on the fifth Mutant p53 Workshop
Blandino, G, Deppert, W, Hainaut, P, Levine, A, Lozano, G, Olivier, M, Rotter, V, Wiman, K, Oren, M
Published in Cell death and differentiation (01.01.2012)
Published in Cell death and differentiation (01.01.2012)
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Conference Proceeding
Small molecules that reactivate mutant p53
Bykov, V.J.N., Selivanova, G., Wiman, K.G.
Published in European journal of cancer (1990) (01.09.2003)
Published in European journal of cancer (1990) (01.09.2003)
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