Green Drug Discovery: Novel Fragment Space from the Biomass-Derived Molecule Dihydrolevoglucosenone (Cyrene TM )
Dekker, Tom, Harteveld, Jaap W, Wágner, Gábor, de Vries, Max C M, Custers, Hans, van de Stolpe, Andrea C, de Esch, Iwan J P, Wijtmans, Maikel
Published in Molecules (Basel, Switzerland) (13.02.2023)
Published in Molecules (Basel, Switzerland) (13.02.2023)
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Journal Article
Self-cleavage of the Pseudomonas aeruginosa Cell-surface Signaling Anti-sigma Factor FoxR Occurs through an N-O Acyl Rearrangement
Bastiaansen, Karlijn C., van Ulsen, Peter, Wijtmans, Maikel, Bitter, Wilbert, Llamas, María A.
Published in The Journal of biological chemistry (08.05.2015)
Published in The Journal of biological chemistry (08.05.2015)
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Journal Article
A toolbox of molecular photoswitches to modulate the CXCR3 chemokine receptor with light
Gómez-Santacana, Xavier, de Munnik, Sabrina M, Mocking, Tamara A M, Hauwert, Niels J, Sun, Shanliang, Vijayachandran, Prashanna, de Esch, Iwan J P, Vischer, Henry F, Wijtmans, Maikel, Leurs, Rob
Published in Beilstein journal of organic chemistry (23.10.2019)
Published in Beilstein journal of organic chemistry (23.10.2019)
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Journal Article
Development of a Selective ESI-MS Derivatization Reagent: Synthesis and Optimization for the Analysis of Aldehydes in Biological Mixtures
Eggink, Mark, Wijtmans, Maikel, Ekkebus, Reggy, Lingeman, Henk, Esch, Iwan J. P. de, Kool, Jeroen, Niessen, Wilfried M. A, Irth, Hubertus
Published in Analytical chemistry (Washington) (01.12.2008)
Published in Analytical chemistry (Washington) (01.12.2008)
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Journal Article
Combined CXCR3/CXCR4 measurements are of high prognostic value in chronic lymphocytic leukemia due to negative co-operativity of the receptors
Ganghammer, Sylvia, Gutjahr, Julia, Hutterer, Evelyn, Krenn, Peter W, Pucher, Susanne, Zelle-Rieser, Claudia, Jöhrer, Karin, Wijtmans, Maikel, Leurs, Rob, Smit, Martine J, Gattei, Valter, Greil, Richard, Hartmann, Tanja N
Published in Haematologica (Roma) (01.03.2016)
Published in Haematologica (Roma) (01.03.2016)
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Journal Article
Bromo-Cyclobutenaminones as New Covalent UDP-N-Acetylglucosamine Enolpyruvyl Transferase (MurA) Inhibitors
Hamilton, David J., Ábrányi-Balogh, Péter, Keeley, Aaron, Petri, László, Hrast, Martina, Imre, Tímea, Wijtmans, Maikel, Gobec, Stanislav, Esch, Iwan J. P. de, Keserű, György Miklós
Published in Pharmaceuticals (Basel, Switzerland) (03.11.2020)
Published in Pharmaceuticals (Basel, Switzerland) (03.11.2020)
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Journal Article
Synthesis, modeling and functional activity of substituted styrene-amides as small-molecule CXCR7 agonists
Wijtmans, Maikel, Maussang, David, Sirci, Francesco, Scholten, Danny J., Canals, Meritxell, Mujić-Delić, Azra, Chong, Milagros, Chatalic, Kristell L.S., Custers, Hans, Janssen, Elwin, de Graaf, Chris, Smit, Martine J., de Esch, Iwan J.P., Leurs, Rob
Published in European journal of medicinal chemistry (01.05.2012)
Published in European journal of medicinal chemistry (01.05.2012)
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Journal Article
Optical control of the β2-adrenergic receptor with opto-prop-2: A cis-active azobenzene analog of propranolol
Bosma, Reggie, Dijon, Nicola C., Zheng, Yang, Schihada, Hannes, Hauwert, Niels J., Shi, Shuang, Arimont, Marta, Riemens, Rick, Custers, Hans, van de Stolpe, Andrea, Vischer, Henry F., Wijtmans, Maikel, Holliday, Nicholas D., Kuster, Diederik W.D., Leurs, Rob
Published in iScience (16.09.2022)
Published in iScience (16.09.2022)
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Journal Article
Exploring the Effect of Cyclization of Histamine H1 Receptor Antagonists on Ligand Binding Kinetics
Wang, Zhiyong, Bosma, Reggie, Kuhne, Sebastiaan, van den Bor, Jelle, Garabitian, Wrej, Vischer, Henry F, Wijtmans, Maikel, Leurs, Rob, de Esch, Iwan J.P
Published in ACS omega (18.05.2021)
Published in ACS omega (18.05.2021)
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Journal Article
Development of an on-line weak-cation exchange liquid chromatography–tandem mass spectrometric method for screening aldehyde products in biological matrices
Eggink, Mark, Charret, Ségolène, Wijtmans, Maikel, Lingeman, Henk, Kool, Jeroen, Niessen, Wilfried M.A., Irth, Hubertus
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.12.2009)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.12.2009)
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Journal Article
Synthesis and Reactivity of Some 6-Substituted-2,4-dimethyl-3-pyridinols, a Novel Class of Chain-Breaking Antioxidants
Wijtmans, Maikel, Pratt, Derek A, Brinkhorst, Johan, Serwa, Remigiusz, Valgimigli, Luca, Pedulli, Gian Franco, Porter, Ned A
Published in Journal of organic chemistry (24.12.2004)
Published in Journal of organic chemistry (24.12.2004)
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Journal Article
Identification and analysis of products formed from phospholipids in the free radical oxidation of human low density lipoproteins
Milne, Ginger L., Seal, Jennifer R., Havrilla, Christine M., Wijtmans, Maikel, Porter, Ned A.
Published in Journal of lipid research (01.02.2005)
Published in Journal of lipid research (01.02.2005)
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Journal Article
Optical control of Class A G protein-coupled receptors with photoswitchable ligands
Wijtmans, Maikel, Josimovic, Ivana, Vischer, Henry F., Leurs, Rob
Published in Current opinion in pharmacology (01.04.2022)
Published in Current opinion in pharmacology (01.04.2022)
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Journal Article
Modulators of CXCR4 and CXCR7/ACKR3 Function
Adlere, Ilze, Caspar, Birgit, Arimont, Marta, Dekkers, Sebastian, Visser, Kirsten, Stuijt, Jeffrey, de Graaf, Chris, Stocks, Michael, Kellam, Barrie, Briddon, Stephen, Wijtmans, Maikel, de Esch, Iwan, Hill, Stephen, Leurs, Rob
Published in Molecular pharmacology (01.12.2019)
Published in Molecular pharmacology (01.12.2019)
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Journal Article
High‐Pressure‐Mediated Fragment Library Synthesis of 1,2‐Disubsituted Cyclobutane Derivatives
Janssen, Mathilde A. C. H., Rappard, Rico, Dekker, Tom, Heiming, Mitchel, Beens, Marjolijn, Pieters, Dyon, Kuijpers, Brian H. M., Benningshof, Jorg C. J., Wijtmans, Maikel, de Esch, Iwan J. P., Blanco‐Ania, Daniel, Rutjes, Floris P. J. T.
Published in European journal of organic chemistry (29.10.2024)
Published in European journal of organic chemistry (29.10.2024)
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