The first selective agonist for the neuropeptide YY5 receptor increases food intake in rats
Cabrele, C, Langer, M, Bader, R, Wieland, H A, Doods, H N, Zerbe, O, Beck-Sickinger, A G
Published in The Journal of biological chemistry (17.11.2000)
Published in The Journal of biological chemistry (17.11.2000)
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Journal Article
A single histidine in GABAA receptors is essential for benzodiazepine agonist binding
Wieland, H A, Lüddens, H, Seeburg, P H
Published in The Journal of biological chemistry (25.01.1992)
Published in The Journal of biological chemistry (25.01.1992)
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Journal Article
Pharmacological characterization of the selective nonpeptide neuropeptide Y Y1 receptor antagonist BIBP 3226
Doods, H N, Wienen, W, Entzeroth, M, Rudolf, K, Eberlein, W, Engel, W, Wieland, H A
Published in The Journal of pharmacology and experimental therapeutics (01.10.1995)
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Published in The Journal of pharmacology and experimental therapeutics (01.10.1995)
Journal Article
The role of NPY in metabolic homeostasis: implications for obesity therapy
Wieland, H A, Hamilton, B S, Krist, B, Doods, H N
Published in Expert opinion on investigational drugs (01.06.2000)
Published in Expert opinion on investigational drugs (01.06.2000)
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Journal Article
Subtype selectivity and antagonistic profile of the nonpeptide Y1 receptor antagonist BIBP 3226
Wieland, H A, Willim, K D, Entzeroth, M, Wienen, W, Rudolf, K, Eberlein, W, Engel, W, Doods, H N
Published in The Journal of pharmacology and experimental therapeutics (01.10.1995)
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Published in The Journal of pharmacology and experimental therapeutics (01.10.1995)
Journal Article
BIBP 3226, the first selective neuropeptide Y1 receptor antagonist: A review of its pharmacological properties
Doods, Henri N., Wieland, Heike A., Engel, Wolfhard, Eberlein, Wolfgang, Willim, Klaus-Dieter, Entzeroth, Michael, Wienen, Wolfgang, Rudolf, Klaus
Published in Regulatory peptides (27.08.1996)
Published in Regulatory peptides (27.08.1996)
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Journal Article
Current potentiation by diazepam but not GABA sensitivity is determined by a single histidine residue
Kleingoor, C, Wieland, H A, Korpi, E R, Seeburg, P H, Kettenmann, H
Published in Neuroreport (01.02.1993)
Published in Neuroreport (01.02.1993)
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Journal Article
Weighing the options in the pharmacotherapy of obesity
Wieland, H A, Hamilton, B S
Published in International journal of clinical pharmacology and therapeutics (01.09.2001)
Published in International journal of clinical pharmacology and therapeutics (01.09.2001)
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Journal Article
The first highly potent and selective non-peptide neuropeptide Y Y1 receptor antagonist : BIBP3226
RUDOLF, K, EBERLEIN, W, ENGEL, W, WIELAND, H. A, WILLIM, K. D, ENTZEROTH, M, WIENEN, W, BECK-SICKINGER, A. G, DOODS, H. N
Published in European journal of pharmacology (27.12.1994)
Published in European journal of pharmacology (27.12.1994)
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Journal Article
Further characterization of neuropeptide Y receptor subtypes using centrally truncated analogs of neuropeptide Y: evidence for subtype-differentiating effects on affinity and intrinsic efficacy
MICHEL, M. C, GAIDA, W, BECK-SICKINGER, A. G, WIELAND, H. A, DOODS, H, DÜRR, H, KUNG, G, SCHNORRENBERG, G
Published in Molecular pharmacology (01.10.1992)
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Published in Molecular pharmacology (01.10.1992)
Journal Article
High-affinity analogues of neuropeptide Y containing conformationally restricted non-proteinogenic amino acids
Beck-Sickinger, A G, Hoffmann, E, Paulini, K, Reissig, H U, Willim, K D, Wieland, H A, Jung, G
Published in Biochemical Society transactions (01.02.1994)
Published in Biochemical Society transactions (01.02.1994)
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Journal Article
Labeling of neuropeptide Y receptors in SK-N-MC cells using the novel, nonpeptide Y1 receptor-selective antagonist [3H]BIBP3226
ENTZEROTH, M, BRAUNGER, H, EBERLEIN, W, ENGEL, W, RUDOLF, K, WIENEN, W, WIELAND, H. A, WILLIM, K.-D, DOODS, H. N
Published in European journal of pharmacology (24.05.1995)
Published in European journal of pharmacology (24.05.1995)
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Journal Article
Molecular determinants in GABAA/BZ receptor subtypes
Wieland, H A, Lüddens, H, Seeburg, P H
Published in Advances in biochemical psychopharmacology (1992)
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Published in Advances in biochemical psychopharmacology (1992)
Journal Article
Osteoarthritis - an untreatable disease?
Wieland, Heike A, Michaelis, Martin, Kirschbaum, Bernhard J, Rudolphi, Karl A
Published in Nature reviews. Drug discovery (01.04.2005)
Published in Nature reviews. Drug discovery (01.04.2005)
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Journal Article
Comparison of antibodies directed against receptor segments of NPY-receptors
Eckard, C P, Beck-Sickinger, A G, Wieland, H A
Published in Journal of receptors and signal transduction (01.01.1999)
Published in Journal of receptors and signal transduction (01.01.1999)
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Journal Article
Biodynamer Nano-Complexes and -Emulsions for Peptide and Protein Drug Delivery
Liu, Yun, Hamm, Timo, Eichinger, Thomas Ralf, Kamm, Walter, Wieland, Heike Andrea, Loretz, Brigitta, Hirsch, Anna K H, Lee, Sangeun, Lehr, Claus-Michael
Published in International journal of nanomedicine (01.01.2024)
Published in International journal of nanomedicine (01.01.2024)
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