Synthesis and SAR studies of benzimidazolone derivatives as histamine H3-receptor antagonists
Zeng, Qingbei, Rosenblum, Stuart B., Yang, Zhaoxia, Jiang, Yueheng, McCormick, Kevin D., Aslanian, Robert G., Duguma, Luli, Kozlowski, Joseph A., Shih, Neng-Yang, Hey, John A., West, Robert E., Korfmacher, Walter A., Berlin, Michael, Boyce, Christopher W.
Published in Bioorganic & medicinal chemistry letters (01.11.2013)
Published in Bioorganic & medicinal chemistry letters (01.11.2013)
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Synthesis and structure–activity relationship (SAR) study of 4-azabenzoxazole analogues as H3 antagonists
Shao, Ning, Aslanian, Robert, West, Robert E., Williams, Shirley M., Wu, Ren-Long, Hwa, Joyce, Sondey, Christopher, Lachowicz, Jean, Palani, Anandan
Published in Bioorganic & medicinal chemistry letters (01.03.2012)
Published in Bioorganic & medicinal chemistry letters (01.03.2012)
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Fused bicycles as arylketone bioisosteres leading to potent, orally active thiadiazole H3 antagonists
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Published in Bioorganic & medicinal chemistry letters (01.05.2012)
Published in Bioorganic & medicinal chemistry letters (01.05.2012)
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Biochemical characterization of desloratadine, a potent antagonist of the human histamine H1 receptor
ANTHES, John C, GILCHREST, Helen, EGAN, Robert W, RICHARD, Christian, ECKEL, Stephen, HESK, Dave, WEST, Robert E, WILLIAMS, Shirley M, GREENFEDER, Scott, BILLAH, Motasim, KREUTNER, William
Published in European journal of pharmacology (01.08.2002)
Published in European journal of pharmacology (01.08.2002)
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Synthesis and structure-activity relationships of 2-(1,4'-bipiperidin-1'-yl) thiazolopyridine as H3 receptor antagonists
RAO, Ashwin U, PALANI, Anandan, LACHOWICZ, Jean, XIAO CHEN, YING HUANG, ASLANIAN, Robert G, WEST, Robert E, WILLIAMS, Shirley M, WU, Ren-Long, HWA, Joyce, SONDEY, Christopher
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
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Reduction of hERG inhibitory activity in the 4-piperidinyl urea series of H3 antagonists
Berlin, Michael, Lee, Yoon Joo, Boyce, Christopher W., Wang, Yi, Aslanian, Robert, McCormick, Kevin D., Sorota, Steve, Williams, Shirley M., West, Robert E., Korfmacher, Walter
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
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Pharmacological characterization of the novel histamine H3-receptor antagonist N-(3,5-dichlorophenyl)-N'-[[4-(1H-imidazol-4-ylmethyl)phenyl]-methyl]-urea (SCH 79687)
McLeod, Robbie L, Rizzo, Charlie A, West, Jr, Robert E, Aslanian, Robert, McCormick, Kevin, Bryant, Matthew, Hsieh, Yunsheng, Korfmacher, Walter, Mingo, Garfield G, Varty, LoriAnn, Williams, Shirley M, Shih, Neng-Yang, Egan, Robert W, Hey, John A
Published in The Journal of pharmacology and experimental therapeutics (01.06.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2003)
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Discovery of a Potent Thiadiazole Class of Histamine H3 Receptor Antagonist for the Treatment of Diabetes
Rao, Ashwin U, Shao, Ning, Aslanian, Robert G, Chan, Tin-Yau, Degrado, Sylvia J, Wang, Li, McKittrick, Brian, Senior, Mary, West, Robert E, Williams, Shirley M, Wu, Ren-Long, Hwa, Joyce, Patel, Bhuneshwari, Zheng, Shuqin, Sondey, Christopher, Palani, Anandan
Published in ACS medicinal chemistry letters (08.03.2012)
Published in ACS medicinal chemistry letters (08.03.2012)
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Reduction of CYP450 inhibition in the 4-[(1H-imidazol-4-yl)methyl]piperidine series of histamine H3 receptor antagonists
BERLIN, Michael, TING, Pauline C, DUGUMA, Luli, SOLOMON, Daniel M, WEI ZHOU, SHER, Rosy, FAVREAU, Leonard, BRYANT, Matthew, KORFMACHER, Walter A, NARDO, Cymbelene, WEST, Robert E, ANTHES, John C, VACCARO, Wayne D, WILLIAMS, Shirley M, WU, Ren-Long, SHE, H. Susan, RIVELLI, Maria A, CORBOZ, Michel R, HEY, John A, ASLANIAN, Robert, MCCORMICK, Kevin D, LEE, Joe F, ALBANESE, Margaret M, MUTAHI, Mwangi W, PIWINSKI, John J, SHIH, Neng-Yang
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
Published in Bioorganic & medicinal chemistry letters (15.02.2006)
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Novel histamine H3 receptor antagonists based on the 4-[(1H-imidazol-4-yl)methyl]piperidine scaffold
VACCARO, Wayne D, SHER, Rosy, WILLIAMS, Shirley M, WU, Ren-Long, SHE, H. Susan, RIVELLI, Maria A, MUTTER, Jennifer C, CORBOZ, Michel R, HEY, John A, FAVREAU, Leonard, BERLIN, Michael, SHIH, Neng-Yang, ASLANIAN, Robert, SCHWERDT, John H, MCCORMICK, Kevin D, PIWINSKI, John J, WEST, Robert E, ANTHES, John C
Published in Bioorganic & medicinal chemistry letters (15.01.2006)
Published in Bioorganic & medicinal chemistry letters (15.01.2006)
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Cloning and Characterization of a Novel Human Histamine Receptor
Morse, K L, Behan, J, Laz, T M, West, Jr, R E, Greenfeder, S A, Anthes, J C, Umland, S, Wan, Y, Hipkin, R W, Gonsiorek, W, Shin, N, Gustafson, E L, Qiao, X, Wang, S, Hedrick, J A, Greene, J, Bayne, M, Monsma, Jr, F J
Published in The Journal of pharmacology and experimental therapeutics (01.03.2001)
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Published in The Journal of pharmacology and experimental therapeutics (01.03.2001)
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Discovery of a series of potent arylthiadiazole H₃ antagonists
Xiao, Dong, Palani, Anandan, Sofolarides, Michael, Huang, Ying, Aslanian, Robert, Vaccaro, Henry, Hong, Liwu, McKittrick, Brian, West, Robert E., Jr, Williams, Shirley M, Wu, Ren-Long, Hwa, Joyce, Sondey, Christopher, Lachowicz, Jean
Published in Bioorganic & medicinal chemistry letters (2011)
Published in Bioorganic & medicinal chemistry letters (2011)
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Structural determinants for histamine H1 affinity, hERG affinity and QTc prolongation in a series of terfenadine analogs
ASLANIAN, Robert, PIWINSKI, John J, HEY, John A, XIAOHONG ZHU, PRIESTLEY, Tony, SOROTA, Steve, DU, Xiao-Yi, ZHANG, Xue-Song, MCLEOD, Robbie L, WEST, Robert E, WILLIAMS, Shirley M
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
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The synthesis and structure-activity relationship of 4-benzimidazolyl-piperidinylcarbonyl-piperidine analogs as histamine H3 antagonists
TING, Pauline C, LEE, Joe F, ANTHES, John C, RIVELLI, Maria A, CORBOZ, Michel R, HEY, John A, ALBANESE, Margaret M, JIE WU, ASLANIAN, Robert, FAVREAU, Leonard, NARDO, Cymbelene, KORFMACHER, Walter A, WEST, Robert E, WILLIAMS, Shirley M
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
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Thermal Analysis of Microfluidic cooling in Processing-in-3D-Stacked Memory
Han, Jun-Han, Torres-Castro, Karina, West, Robert E., Swami, Nathan, Stan, Mircea
Published in 2021 22nd International Conference on Thermal, Mechanical and Multi-Physics Simulation and Experiments in Microelectronics and Microsystems (EuroSimE) (19.04.2021)
Published in 2021 22nd International Conference on Thermal, Mechanical and Multi-Physics Simulation and Experiments in Microelectronics and Microsystems (EuroSimE) (19.04.2021)
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Conference Proceeding
Power and Thermal Modeling of In-3D-Memory Computing
Han, Jun-Han, West, Robert E., Torres-Castro, Karina, Swami, Nathan, Khan, Samira, Stan, Mircea
Published in 2021 International Symposium on Devices, Circuits and Systems (ISDCS) (03.03.2021)
Published in 2021 International Symposium on Devices, Circuits and Systems (ISDCS) (03.03.2021)
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Dual antagonists of platelet-activating factor and histamine. Identification of structural requirements for dual activity of N-acyl-4-(5,6-dihydro-11H-benzo[5,6]cyclohepta[1,2-b]pyridin-11-ylidene)piperidines
Piwinski, John J, Wong, Jesse K, Green, Michael J, Ganguly, Ashit K, Billah, M. Motasim, West, Robert E, Kreutner, William
Published in Journal of medicinal chemistry (01.01.1991)
Published in Journal of medicinal chemistry (01.01.1991)
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