Discovery and Optimization of a Novel Class of Orally Active Nonpeptidic Endothelin-A Receptor Antagonists
Riechers, Hartmut, Albrecht, Hans-Peter, Amberg, Willi, Baumann, Ernst, Bernard, Harald, Böhm, Hans-Joachim, Klinge, Dagmar, Kling, Andreas, Müller, Stefan, Raschack, Manfred, Unger, Liliane, Walker, Nigel, Wernet, Wolfgang
Published in Journal of medicinal chemistry (24.05.1996)
Published in Journal of medicinal chemistry (24.05.1996)
Get full text
Journal Article
Potent and selective oxindole-based vasopressin 1b receptor antagonists with improved pharmacokinetic properties
Oost, Thorsten, Backfisch, Gisela, Bhowmik, Swati, van Gaalen, Marcel M., Geneste, Hervé, Hornberger, Wilfried, Lubisch, Wilfried, Netz, Astrid, Unger, Liliane, Wernet, Wolfgang
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Get full text
Journal Article
Discovery and SAR of 2-(1-propylpiperidin-4-yl)-1H-benzimidazole-4-carboxamide: A potent inhibitor of poly(ADP-ribose) polymerase (PARP) for the treatment of cancer
Penning, Thomas D, Zhu, Gui-Dong, Gandhi, Viraj B, Gong, Jianchun, Thomas, Sheela, Lubisch, Wilfried, Grandel, Roland, Wernet, Wolfgang, Park, Chang H, Fry, Elizabeth H, Liu, Xuesong, Shi, Yan, Klinghofer, Vered, Johnson, Eric F, Donawho, Cherrie K, Frost, David J, Bontcheva-Diaz, Velitchka, Bouska, Jennifer J, Olson, Amanda M, Marsh, Kennan C, Luo, Yan, Rosenberg, Saul H, Giranda, Vincent L
Published in Bioorganic & medicinal chemistry (15.07.2008)
Published in Bioorganic & medicinal chemistry (15.07.2008)
Get full text
Journal Article
Synthesis and SAR of highly potent and selective dopamine D 3-receptor antagonists: Quinolin(di)one and benzazepin(di)one derivatives
Geneste, Hervé, Backfisch, Gisela, Braje, Wilfried, Delzer, Jürgen, Haupt, Andreas, Hutchins, Charles W., King, Linda L., Lubisch, Wilfried, Steiner, Gerd, Teschendorf, Hans-Jürgen, Unger, Liliane, Wernet, Wolfgang
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Published in Bioorganic & medicinal chemistry letters (01.02.2006)
Get full text
Journal Article
A Polypyrrole/Three-Enzyme Electrode for Creatinine Detection
Yamato, Hitoshi, Ohwa, Masaki, Wernet, Wolfgang
Published in Analytical chemistry (Washington) (01.09.1995)
Published in Analytical chemistry (Washington) (01.09.1995)
Get full text
Journal Article
Synthesis and SAR of highly potent and selective dopamine D sub(3)-receptor antagonists: Variations on the 1H-pyrimidin-2-one theme
Geneste, Herve, Amberg, Wilhelm, Backfisch, Gisela, Beyerbach, Armin, Braje, Wilfried M, Delzer, Juergen, Haupt, Andreas, Hutchins, Charles W, King, Linda L, Sauer, Daryl R, Unger, Liliane, Wernet, Wolfgang
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Published in Bioorganic & medicinal chemistry letters (01.04.2006)
Get full text
Journal Article
Discovery and SAR of 2-(l-propylpiperidin-4-yl)-lH-benzimidazole-4-carboxamide : A potent inhibitor of poly(ADP-ribose) polymerase (PARP) for the treatment of cancer
PENNING, Thomas D, ZHU, Gui-Dong, XUESONG LIU, YAN SHI, KLINGHOFER, Vered, JOHNSON, Eric F, DONAWHO, Cherrie K, FROST, David J, BONTCHEVA-DIAZ, Velitchka, BOUSKA, Jennifer J, OLSON, Amanda M, MARSH, Kennan C, GANDHI, Viraj B, YAN LUO, ROSENBERG, Saul H, GIRANDA, Vincent L, JIANCHUN GONG, THOMAS, Sheela, LUBISCH, Wilfried, GRANDEL, Roland, WERNET, Wolfgang, PARK, Chang H, FRY, Elizabeth H
Published in Bioorganic & medicinal chemistry (2008)
Get full text
Published in Bioorganic & medicinal chemistry (2008)
Journal Article
Discovery and SAR of 2-(1-propylpiperidin-4-yl)-1 H-benzimidazole-4-carboxamide: A potent inhibitor of poly(ADP-ribose) polymerase (PARP) for the treatment of cancer
Penning, Thomas D., Zhu, Gui-Dong, Gandhi, Viraj B., Gong, Jianchun, Thomas, Sheela, Lubisch, Wilfried, Grandel, Roland, Wernet, Wolfgang, Park, Chang H., Fry, Elizabeth H., Liu, Xuesong, Shi, Yan, Klinghofer, Vered, Johnson, Eric F., Donawho, Cherrie K., Frost, David J., Bontcheva-Diaz, Velitchka, Bouska, Jennifer J., Olson, Amanda M., Marsh, Kennan C., Luo, Yan, Rosenberg, Saul H., Giranda, Vincent L.
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
Get full text
Journal Article