Accessing Diverse Azole Carboxylic Acid Building Blocks via Mild C–H Carboxylation: Parallel, One-Pot Amide Couplings and Machine-Learning-Guided Substrate Scope Design
Felten, Stephanie, He, Cyndi Qixin, Weisel, Mark, Shevlin, Michael, Emmert, Marion H.
Published in Journal of the American Chemical Society (21.12.2022)
Published in Journal of the American Chemical Society (21.12.2022)
Get full text
Journal Article
Quinone-mediated hydrogen anode for non-aqueous reductive electrosynthesis
Twilton, Jack, Johnson, Mathew R., Sidana, Vinayak, Franke, Mareena C., Bottecchia, Cecilia, Lehnherr, Dan, Lévesque, François, Knapp, Spring M. M., Wang, Luning, Gerken, James B., Hong, Cynthia M., Vickery, Thomas P., Weisel, Mark D., Strotman, Neil A., Weix, Daniel J., Root, Thatcher W., Stahl, Shannon S.
Published in Nature (London) (02.11.2023)
Published in Nature (London) (02.11.2023)
Get full text
Journal Article
Nine-Step Stereoselective Synthesis of Islatravir from Deoxyribose
Nawrat, Christopher C, Whittaker, Aaron M, Huffman, Mark A, McLaughlin, Mark, Cohen, Ryan D, Andreani, Teresa, Ding, Bangwei, Li, Hongming, Weisel, Mark, Tschaen, David M
Published in Organic letters (20.03.2020)
Published in Organic letters (20.03.2020)
Get full text
Journal Article
Mechanistic Study of a Re-Catalyzed Monoalkylation of Phenols
Lehnherr, Dan, Wang, Xiao, Peng, Feng, Reibarkh, Mikhail, Weisel, Mark, Maloney, Kevin M
Published in Organometallics (14.01.2019)
Published in Organometallics (14.01.2019)
Get full text
Journal Article
Development of a Commercial Manufacturing Route to 2‑Fluoroadenine, The Key Unnatural Nucleobase of Islatravir
Hong, Cynthia M, Xu, Yingju, Chung, John Y. L, Schultz, Danielle M, Weisel, Mark, Varsolona, Richard J, Zhong, Yong-Li, Purohit, Akasha K, He, Cyndi Q, Gauthier, Donald R, Humphrey, Guy R, Maloney, Kevin M, Lévesque, François, Wang, Zhixun, Whittaker, Aaron M, Sirota, Eric, McMullen, Jonathan P
Published in Organic process research & development (19.03.2021)
Published in Organic process research & development (19.03.2021)
Get full text
Journal Article
An Integrated Approach for Creating Model Diesel Fuels
Androulakis, Ioannis P, Weisel, Mark D, Hsu, Chang S, Qian, Kuangnan, Green, Larry A, Farrell, John T, Nakakita, Kiyomi
Published in Energy & fuels (01.01.2005)
Published in Energy & fuels (01.01.2005)
Get full text
Journal Article
Development and Implementation of an Aluminum-Promoted Phosphorylation in the Uprifosbuvir Manufacturing Route
Liu, Zhuqing, Klapars, Artis, Simmons, Bryon, Bellomo, Ana, Kalinin, Alexei, Weisel, Mark, Hill, Jerry, Silverman, Steven M
Published in Organic process research & development (19.03.2021)
Published in Organic process research & development (19.03.2021)
Get full text
Journal Article
Calcium Dialkylamine Diazeniumdiolates: Synthesis, Stability, and Nitric Oxide Generation
Kauser, Nabeelah I, Weisel, Mark, Zhong, Yong-Li, Lo, Michael Man-Chu, Ali, Amjad
Published in Journal of organic chemistry (03.04.2020)
Published in Journal of organic chemistry (03.04.2020)
Get full text
Journal Article
A mechanistic investigation of an Iridium-catalyzed asymmetric hydrogenation of pyridinium salts
Huang, Yuhua, Liu, Shaodong, Liu, Yizhou, Chen, Yonggang, Weisel, Mark, Williamson, R. Thomas, Davies, Ian W., Zhang, Xumu
Published in Tetrahedron (26.04.2018)
Published in Tetrahedron (26.04.2018)
Get full text
Journal Article
Manufacturing Process Development for Belzutifan, Part 5: A Streamlined Fluorination–Dynamic Kinetic Resolution Process
Wang, Tao, Phillips, Eric M, Dalby, Stephen M, Sirota, Eric, Axnanda, Stephanus, Shultz, C. Scott, Patel, Pratiq, Waldman, Jacob H, Alwedi, Embarek, Wang, Xiao, Zawatzky, Kerstin, Chow, Matthew, Padivitage, Nilusha, Weisel, Mark, Whittington, Michael, Duan, Jianjun, Lu, Taotao
Published in Organic process research & development (18.03.2022)
Published in Organic process research & development (18.03.2022)
Get full text
Journal Article
Improved Preparation of a Key Hydroxylamine Intermediate for Relebactam: Rate Enhancement of Benzyl Ether Hydrogenolysis with DABCO
Yin, Jianguo, Weisel, Mark, Ji, Yining, Liu, Zhijian, Liu, Jinchu, Wallace, Debra J, Xu, Feng, Sherry, Benjamin D, Yasuda, Nobuyoshi
Published in Organic process research & development (16.03.2018)
Published in Organic process research & development (16.03.2018)
Get full text
Journal Article
Enantioselective Hydrogenation of N−H Imines
Hou, Guohua, Gosselin, Francis, Li, Wei, McWilliams, J. Christopher, Sun, Yongkui, Weisel, Mark, O’Shea, Paul D, Chen, Cheng-yi, Davies, Ian W, Zhang, Xumu
Published in Journal of the American Chemical Society (29.07.2009)
Published in Journal of the American Chemical Society (29.07.2009)
Get full text
Journal Article
Enantioselective Synthesis of α‑Methyl-β-cyclopropyldihydrocinnamates
Christensen, Melodie, Nolting, Andrew, Shevlin, Michael, Weisel, Mark, Maligres, Peter E, Lee, Joshua, Orr, Robert K, Plummer, Christopher W, Tudge, Matthew T, Campeau, Louis-Charles, Ruck, Rebecca T
Published in Journal of organic chemistry (05.02.2016)
Published in Journal of organic chemistry (05.02.2016)
Get full text
Journal Article
Development of a Green and Sustainable Manufacturing Process for Gefapixant Citrate (MK-7264) Part 2: Development of a Robust Process for Phenol Synthesis
Peng, Feng, Humphrey, Guy R, Maloney, Kevin M, Lehnherr, Dan, Weisel, Mark, Lévesque, Francois, Naber, John R, Brunskill, Andrew P. J, Larpent, Patrick, Zhang, Si-Wei, Lee, Alfred Y, Arvary, Rebecca A, Lee, Claire H, Bishara, Daniel, Narsimhan, Karthik, Sirota, Eric, Whittington, Michael
Published in Organic process research & development (20.11.2020)
Published in Organic process research & development (20.11.2020)
Get full text
Journal Article
Development of a Scalable and Safer Synthesis of Diazeniumdiolates
Zhong, Yong-Li, Muzzio, Daniel J, Weisel, Mark, Zhang, Li, Humphrey, Guy R, Maloney, Kevin M, Campos, Kevin R
Published in Organic process research & development (18.09.2020)
Published in Organic process research & development (18.09.2020)
Get full text
Journal Article
One-Step Synthesis of 2‑Fluoroadenine Using Hydrogen Fluoride Pyridine in a Continuous Flow Operation
Salehi Marzijarani, Nastaran, Snead, David R, McMullen, Jonathan P, Lévesque, François, Weisel, Mark, Varsolona, Richard J, Lam, Yu-hong, Liu, Zhijian, Naber, John R
Published in Organic process research & development (16.08.2019)
Published in Organic process research & development (16.08.2019)
Get full text
Journal Article
Scalable Synthesis of Diazeniumdiolates: Application to the Preparation of MK-8150
Zhong, Yong-Li, Weisel, Mark, Humphrey, Guy R, Muzzio, Daniel J, Zhang, Li, Huffman, Mark A, Zhong, Wendy, Maloney, Kevin M, Campos, Kevin R
Published in Organic letters (07.06.2019)
Published in Organic letters (07.06.2019)
Get full text
Journal Article
Convergent, Kilogram Scale Synthesis of an Akt Kinase Inhibitor
Grongsaard, Pintipa, Bulger, Paul G, Wallace, Debra J, Tan, Lushi, Chen, Qinghao, Dolman, Sarah J, Nyrop, Jason, Hoerrner, R. Scott, Weisel, Mark, Arredondo, Juan, Itoh, Takahiro, Xie, Chengfu, Wen, Xianghui, Zhao, Dalian, Muzzio, Daniel J, Bassan, Ephraim M, Shultz, C. Scott
Published in Organic process research & development (18.05.2012)
Published in Organic process research & development (18.05.2012)
Get full text
Journal Article