Solvent-Controlled, Site-Selective N‑Alkylation Reactions of Azolo-Fused Ring Heterocycles at N1‑, N2‑, and N3-Positions, Including Pyrazolo[3,4‑d]pyrimidines, Purines, [1,2,3]Triazolo[4,5]pyridines, and Related Deaza-Compounds
Bookser, Brett C, Weinhouse, Michael I, Burns, Aaron C, Valiere, Andrew N, Valdez, Lino J, Stanczak, Pawel, Na, Jim, Rheingold, Arnold L, Moore, Curtis E, Dyck, Brian
Published in Journal of organic chemistry (15.06.2018)
Published in Journal of organic chemistry (15.06.2018)
Get full text
Journal Article
Antimalarial Activities of Novel Synthetic Cysteine Protease Inhibitors
LEE, Belinda J, SINGH, Ajay, CHIANG, Peggy, KEMP, Scott J, GOLDMAN, Erick A, WEINHOUSE, Michael I, VLASUK, George P, ROSENTHAL, Philip J
Published in Antimicrobial Agents and Chemotherapy (01.12.2003)
Published in Antimicrobial Agents and Chemotherapy (01.12.2003)
Get full text
Journal Article
A new family of H3 receptor antagonists based on the natural product Conessine
SANTORA, Vincent J, COVEL, Jonathan A, WEBB, Robert R, SAGE, Carleton, REN, Albert, PEREIRA, Guilherme, KNUDSEN, Jens, EDWARDS, Jeffrey E, SUAREZ, Marissa, FRAZER, John, THOMSEN, William, HAUSER, Erin, HAYASHI, Rena, WHELAN, Kevin, GROTTICK, Andrew J, HOFILENA, Brian J, IBARRA, Jason B, PULLEY, Michelle D, WEINHOUSE, Michael I, SENGUPTA, Dipanjan, DUFFIELD, Jonathan J, SEMPLE, Graeme
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
Get full text
Journal Article
Design and Evaluation of Novel Biphenyl Sulfonamide Derivatives with Potent Histamine H(3) Receptor Inverse Agonist Activity
Covel, Jonathan A., Santora, Vincent J., Smith, Jeffrey M., Hayashi, Rena, Gallardo, Charlemagne, Weinhouse, Michael I., Ibarra, Jason B., Schultz, Jeffrey A., Park, Douglas M., Estrada, Scott A., Hofilena, Brian J., Pulley, Michelle D., Smith, Brian M., Ren, Albert, Suarez, Marissa, Frazer, John, Edwards, Jeffrey, Hauser, Erin K., Lorca, Jodie, Semple, Graeme, Grottick, Andrew J.
Published in Journal of medicinal chemistry (24.09.2009)
Published in Journal of medicinal chemistry (24.09.2009)
Get full text
Journal Article
Design and Evaluation of Novel Biphenyl Sulfonamide Derivatives with Potent Histamine H3 Receptor Inverse Agonist Activity
Covel, Jonathan A., Santora, Vincent J., Smith, Jeffrey M., Hayashi, Rena, Gallardo, Charlemagne, Weinhouse, Michael I., Ibarra, Jason B., Schultz, Jeffrey A., Park, Douglas M., Estrada, Scott A., Hofilena, Brian J., Pulley, Michelle D., Smith, Brian M., Ren, Albert, Suarez, Marissa, Frazer, John, Edwards, Jeffrey, Hauser, Erin K., Lorea, Jodie, Semple, Graeme, Grottick, Andrew J.
Published in Journal of medicinal chemistry (24.09.2009)
Published in Journal of medicinal chemistry (24.09.2009)
Get full text
Journal Article
Immobilized catalytic antibodies in aqueous and organic solvents
Janda, Kim D, Ashley, Jon A, Jones, Teresa M, McLeod, Donald A, Schloeder, Diane M, Weinhouse, Michael I
Published in Journal of the American Chemical Society (01.11.1990)
Published in Journal of the American Chemical Society (01.11.1990)
Get full text
Journal Article
Novel H3 receptor antagonists with improved pharmacokinetic profiles
SANTORA, Vincent J, COVEL, Jonathan A, EDWARDS, Jeffrey E, SUAREZ, Marissa, FRAZER, John, THOMSEN, William, HAUSER, Erin, LOREA, Jodie, GROTTICK, Andrew J, HAYASHI, Rena, HOFILENA, Brian J, IBARRA, Jason B, PULLEY, Michelle D, WEINHOUSE, Michael I, SEMPLE, Graeme, REN, Albert, PEREIRA, Guilherme
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
Get full text
Journal Article
Asymmetric induction via a catalytic antibody
Ikeda, Shoji, Weinhouse, Michael I, Janda, Kim D, Lerner, Richard A, Danishefsky, Samuel J
Published in Journal of the American Chemical Society (01.09.1991)
Published in Journal of the American Chemical Society (01.09.1991)
Get full text
Journal Article
Synthesis and biological activity of peptidyl aldehyde urokinase inhibitors
Tamura, S Y, Weinhouse, M I, Roberts, C A, Goldman, E A, Masukawa, K, Anderson, S M, Cohen, C R, Bradbury, A E, Bernardino, V T, Dixon, S A, Ma, M G, Nolan, T G, Brunck, T K
Published in Bioorganic & medicinal chemistry letters (01.05.2000)
Published in Bioorganic & medicinal chemistry letters (01.05.2000)
Get full text
Journal Article
SUBSTITUTED PYRIDINE AND PYRAZINE COMPOUNDS AS PDE4 INHIBITORS
ZAPF JAMES, BREITENBUCHER JAMES, VICKERS TROY, BOLLU VENKATAIAH, LINDSTROM ANDREW, KAPLAN ALAN, LEMUS ROBERT, WILSON MARK E, WEINHOUSE MICHAEL I
Year of Publication 18.11.2015
Get full text
Year of Publication 18.11.2015
Patent
SUBSTITUTED PYRIDINE AZOLOPYRIMIDINE-5-(6H)-ONE COMPOUNDS
PETERS MARCO, ALLAN AMY, DYCK BRIAN, GOMEZ LAURENT, BRANSTETTER BRYAN, WEINHOUSE MICHAEL I, MARRONE TAMI JO
Year of Publication 08.06.2015
Get full text
Year of Publication 08.06.2015
Patent
Catalytic antibodies with acyl-transfer capabilities: mechanistic and kinetic investigations
Janda, Kim D, Ashley, Jon A, Jones, Teresa M, McLeod, Donald A, Schloeder, Diane M, Weinhouse, Michael I, Lerner, Richard A, Gibbs, Richard A, Benkovic, Patricia A
Published in Journal of the American Chemical Society (1991)
Published in Journal of the American Chemical Society (1991)
Get full text
Journal Article
Metalloselective anti-porphyrin monoclonal antibodies
Schwabacher, Alan W, Weinhouse, Michael I, Auditor, Maria Teresa M, Lerner, Richard A
Published in Journal of the American Chemical Society (01.03.1989)
Published in Journal of the American Chemical Society (01.03.1989)
Get full text
Journal Article
A new family of H 3 receptor antagonists based on the natural product Conessine
Santora, Vincent J., Covel, Jonathan A., Hayashi, Rena, Hofilena, Brian J., Ibarra, Jason B., Pulley, Michelle D., Weinhouse, Michael I., Sengupta, Dipanjan, Duffield, Jonathan J., Semple, Graeme, Webb, Robert R., Sage, Carleton, Ren, Albert, Pereira, Guilherme, Knudsen, Jens, Edwards, Jeffrey E., Suarez, Marissa, Frazer, John, Thomsen, William, Hauser, Erin, Whelan, Kevin, Grottick, Andrew J.
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
Published in Bioorganic & medicinal chemistry letters (15.02.2008)
Get full text
Journal Article
Design and Evaluation of Novel Biphenyl Sulfonamide Derivatives with Potent Histamine H 3 Receptor Inverse Agonist Activity
Covel, Jonathan A., Santora, Vincent J., Smith, Jeffrey M., Hayashi, Rena, Gallardo, Charlemagne, Weinhouse, Michael I., Ibarra, Jason B., Schultz, Jeffrey A., Park, Douglas M., Estrada, Scott A., Hofilena, Brian J., Pulley, Michelle D., Smith, Brian M., Ren, Albert, Suarez, Marissa, Frazer, John, Edwards, Jeffrey, Hauser, Erin K., Lorea, Jodie, Semple, Graeme, Grottick, Andrew J.
Published in Journal of medicinal chemistry (24.09.2009)
Published in Journal of medicinal chemistry (24.09.2009)
Get full text
Journal Article
Novel H 3 receptor antagonists with improved pharmacokinetic profiles
Santora, Vincent J., Covel, Jonathan A., Hayashi, Rena, Hofilena, Brian J., Ibarra, Jason B., Pulley, Michelle D., Weinhouse, Michael I., Semple, Graeme, Ren, Albert, Pereira, Guilherme, Edwards, Jeffrey E., Suarez, Marissa, Frazer, John, Thomsen, William, Hauser, Erin, Lorea, Jodie, Grottick, Andrew J.
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
Published in Bioorganic & medicinal chemistry letters (15.07.2008)
Get full text
Journal Article
Novel H sub(3) receptor antagonists with improved pharmacokinetic profiles
Santora, Vincent J, Covel, Jonathan A, Hayashi, Rena, Hofilena, Brian J, Ibarra, Jason B, Pulley, Michelle D, Weinhouse, Michael I, Semple, Graeme, Ren, Albert, Pereira, Guilherme, Edwards, Jeffrey E, Suarez, Marissa, Frazer, John, Thomsen, William, Hauser, Erin, Lorea, Jodie, Grottick, Andrew J
Published in Bioorganic & medicinal chemistry (01.07.2008)
Published in Bioorganic & medicinal chemistry (01.07.2008)
Get full text
Journal Article
A new family of H sub(3) receptor antagonists based on the natural product Conessine
Santora, Vincent J, Covel, Jonathan A, Hayashi, Rena, Hofilena, Brian J, Ibarra, Jason B, Pulley, Michelle D, Weinhouse, Michael I, Sengupta, Dipanjan, Duffield, Jonathan J, Semple, Graeme, Webb, Robert R, Sage, Carleton, Ren, Albert, Pereira, Guilherme, Knudsen, Jens, Edwards, Jeffrey E, Suarez, Marissa, Frazer, John, Thomsen, William, Hauser, Erin, Whelan, Kevin, Grottick, Andrew J
Published in Bioorganic & medicinal chemistry (01.02.2008)
Published in Bioorganic & medicinal chemistry (01.02.2008)
Get full text
Journal Article