Single-vector inducible lentiviral RNAi system for oncology target validation
Wiederschain, Dmitri, Susan, Wee, Chen, Lin, Loo, Alice, Yang, Guizhi, Huang, Alan, Chen, Yan, Caponigro, Giordano, Yao, Yung-mae, Lengauer, Christoph, Sellers, William R., Benson, John D.
Published in Cell cycle (Georgetown, Tex.) (01.02.2009)
Published in Cell cycle (Georgetown, Tex.) (01.02.2009)
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Journal Article
PTEN-deficient cancers depend on PIK3CB
Wee, Susan, Wiederschain, Dmitri, Maira, Sauveur-Michel, Loo, Alice, Miller, Christine, deBeaumont, Rosalie, Stegmeier, Frank, Yao, Yung-Mae, Lengauer, Christoph
Published in Proceedings of the National Academy of Sciences - PNAS (02.09.2008)
Published in Proceedings of the National Academy of Sciences - PNAS (02.09.2008)
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Journal Article
PI3K pathway activation mediates resistance to MEK inhibitors in KRAS mutant cancers
Wee, Susan, Jagani, Zainab, Xiang, Kay Xiaoqin, Loo, Alice, Dorsch, Marion, Yao, Yung-Mae, Sellers, William R, Lengauer, Christoph, Stegmeier, Frank
Published in Cancer research (Chicago, Ill.) (15.05.2009)
Published in Cancer research (Chicago, Ill.) (15.05.2009)
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Journal Article
Specific apoptosis induction by the dual PI3K/mTor inhibitor NVP-BEZ235 in HER2 amplified and PIK3CA mutant breast cancer cells
Brachmann, Saskia M, Hofmann, Irmgard, Schnell, Christian, Fritsch, Christine, Wee, Susan, Lane, Heidi, Wang, Shaowen, Garcia-Echeverria, Carlos, Maira, Sauveur-Michel
Published in Proceedings of the National Academy of Sciences - PNAS (29.12.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (29.12.2009)
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Journal Article
Sensitivity of Small Cell Lung Cancer to BET Inhibition Is Mediated by Regulation of ASCL1 Gene Expression
Lenhart, Ryan, Kirov, Stefan, Desilva, Heshani, Cao, Jian, Lei, Ming, Johnston, Kathy, Peterson, Russell, Schweizer, Liang, Purandare, Ashok, Ross-Macdonald, Petra, Fairchild, Craig, Wong, Tai, Wee, Susan
Published in Molecular cancer therapeutics (01.10.2015)
Published in Molecular cancer therapeutics (01.10.2015)
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Journal Article
Targeting epigenetic regulators for cancer therapy
Wee, Susan, Dhanak, Dash, Li, Haitao, Armstrong, Scott A., Copeland, Robert A., Sims, Robert, Baylin, Stephen B., Liu, Xiaole Shirley, Schweizer, Liang
Published in Annals of the New York Academy of Sciences (01.02.2014)
Published in Annals of the New York Academy of Sciences (01.02.2014)
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Journal Article
F-Box-Directed CRL Complex Assembly and Regulation by the CSN and CAND1
Schmidt, Michael W., McQuary, Philip R., Wee, Susan, Hofmann, Kay, Wolf, Dieter A.
Published in Molecular cell (11.09.2009)
Published in Molecular cell (11.09.2009)
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Journal Article
BTB/POZ Domain Proteins Are Putative Substrate Adaptors for Cullin 3 Ubiquitin Ligases
Geyer, Rory, Wee, Susan, Anderson, Scott, Yates, John, Wolf, Dieter A.
Published in Molecular cell (01.09.2003)
Published in Molecular cell (01.09.2003)
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Journal Article
CSN facilitates Cullin-RING ubiquitin ligase function by counteracting autocatalytic adapter instability
Wolf, Dieter A, Wee, Susan, Geyer, Rory K, Toda, Takashi
Published in Nature cell biology (01.04.2005)
Published in Nature cell biology (01.04.2005)
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Journal Article
DGKζ exerts greater control than DGKα over CD8 + T cell activity and tumor inhibition
Gu, Junchen, Wang, Cindy, Cao, Carolyn, Huang, Jinwen, Holzhauer, Sandra, Desilva, Heshani, Wesley, Erin M, Evans, Douglas B, Benci, Joseph, Wichroski, Michael, Wee, Susan, Riese, Matthew J
Published in Oncoimmunology (01.01.2021)
Published in Oncoimmunology (01.01.2021)
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Journal Article
PCI proteins eIF3e and eIF3m define distinct translation initiation factor 3 complexes
Zhou, Chunshui, Arslan, Fatih, Wee, Susan, Krishnan, Srinivasan, Ivanov, Alexander R, Oliva, Anna, Leatherwood, Janet, Wolf, Dieter A
Published in BMC biology (17.05.2005)
Published in BMC biology (17.05.2005)
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Journal Article
Why is cancer drug discovery so difficult?
Lengauer, Christoph, Kamb, Alexander, Wee, Susan
Published in Nature reviews. Drug discovery (01.02.2007)
Published in Nature reviews. Drug discovery (01.02.2007)
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Journal Article
Book Review
Inhibition of Casein Kinase 2 Disrupts Differentiation of Myeloid Cells in Cancer and Enhances the Efficacy of Immunotherapy in Mice
Hashimoto, Ayumi, Gao, Chan, Mastio, Jerome, Kossenkov, Andrew, Abrams, Scott I, Purandare, Ashok V, Desilva, Heshani, Wee, Susan, Hunt, John, Jure-Kunkel, Maria, Gabrilovich, Dmitry I
Published in Cancer research (Chicago, Ill.) (01.10.2018)
Published in Cancer research (Chicago, Ill.) (01.10.2018)
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Journal Article
Abstract 936: Regulation of CD8+ T-cell function and antitumor activity by DGKα and DGKζ
Wee, Susan, Gu, Junchen, Wang, Cindy, Cao, Carolyn, Holzhauer, Sandra, Desilva, Heshani, Wesley, Erin, Tsai, Susan, Evans, Douglas, Riese, Matthew
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Journal Article
Discovery of (4-Pyrazolyl)-2-aminopyrimidines as Potent and Selective Inhibitors of Cyclin-Dependent Kinase 2
Hummel, Joshua R., Xiao, Kai-Jiong, Yang, Jeffrey C., Epling, Leslie B., Mukai, Ken, Ye, Qinda, Xu, Meizhong, Qian, Dingquan, Huo, Lu, Weber, Michael, Roman, Valerie, Lo, Yvonne, Drake, Katherine, Stump, Kristine, Covington, Maryanne, Kapilashrami, Kanishk, Zhang, Guofeng, Ye, Min, Diamond, Sharon, Yeleswaram, Swamy, Macarron, Ricardo, Deller, Marc C., Wee, Susan, Kim, Sunkyu, Wang, Xiaozhao, Wu, Liangxing, Yao, Wenqing
Published in Journal of medicinal chemistry (22.02.2024)
Published in Journal of medicinal chemistry (22.02.2024)
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Journal Article
DGKα/ζ inhibitors combine with PD-1 checkpoint therapy to promote T cell-mediated antitumor immunity
Wichroski, Michael, Benci, Joseph, Liu, Si-Qi, Chupak, Louis, Fang, Jie, Cao, Carolyn, Wang, Cindy, Onorato, Joelle, Qiu, Hongchen, Shan, Yongli, Banas, Dana, Powles, Ryan, Locke, Gregory, Witt, Abigail, Stromko, Caitlyn, Qi, Huilin, Zheng, Xiaofan, Martin, Scott, Ding, Min, Gentles, Robert, Meanwell, Nicholas, Velaparthi, Upender, Olson, Richard, Wee, Susan, Tenney, Daniel, Parker, Christopher G, Cravatt, Benjamin F, Lawrence, Michael, Borzilleri, Robert, Lees, Emma
Published in Science translational medicine (25.10.2023)
Published in Science translational medicine (25.10.2023)
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Journal Article
Discovery and Preclinical Pharmacology of an Oral Bromodomain and Extra-Terminal (BET) Inhibitor Using Scaffold-Hopping and Structure-Guided Drug Design
Gavai, Ashvinikumar V, Norris, Derek, Delucca, George, Tortolani, David, Tokarski, John S, Dodd, Dharmpal, O’Malley, Daniel, Zhao, Yufen, Quesnelle, Claude, Gill, Patrice, Vaccaro, Wayne, Huynh, Tram, Ahuja, Vijay, Han, Wen-Ching, Mussari, Christopher, Harikrishnan, Lalgudi, Kamau, Muthoni, Poss, Michael, Sheriff, Steven, Yan, Chunhong, Marsilio, Frank, Menard, Krista, Wen, Mei-Li, Rampulla, Richard, Wu, Dauh-Rurng, Li, Jianqing, Zhang, Huiping, Li, Peng, Sun, Dawn, Yip, Henry, Traeger, Sarah C, Zhang, Yingru, Mathur, Arvind, Zhang, Haiying, Huang, Christine, Yang, Zheng, Ranasinghe, Asoka, Everlof, Gerry, Raghavan, Nirmala, Tye, Ching Kim, Wee, Susan, Hunt, John T, Vite, Gregory, Westhouse, Richard, Lee, Francis Y
Published in Journal of medicinal chemistry (14.10.2021)
Published in Journal of medicinal chemistry (14.10.2021)
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Journal Article
Discovery of Potent, Dual-Inhibitors of Diacylglycerol Kinases Alpha and Zeta Guided by Phenotypic Optimization
Chupak, Louis, Wichroski, Michael, Zheng, Xiaofan, Ding, Min, Martin, Scott, Allard, Christopher, Shi, Jianliang, Gentles, Robert, Meanwell, Nicholas A., Fang, Jie, Tenney, Daniel, Tokarski, John, Cao, Carolyn, Wee, Susan
Published in ACS medicinal chemistry letters (13.07.2023)
Published in ACS medicinal chemistry letters (13.07.2023)
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Journal Article