Concise Formal Synthesis of (−)-Peduncularine via Ring-Closing Metathesis
Washburn, David G, Heidebrecht, Richard W, Martin, Stephen F
Published in Organic letters (18.09.2003)
Published in Organic letters (18.09.2003)
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In Vivo Half-Life Extension of BMP1/TLL Metalloproteinase Inhibitors Using Small-Molecule Human Serum Albumin Binders
Vantourout, Julien C, Mason, Andrew M, Yuen, Josephine, Simpson, Graham L, Evindar, Ghotas, Kuai, Letian, Hobbs, Michael, Edgar, Emma, Needle, Saul, Bai, Xiaopeng, Wilson, Steve, Scott-Stevens, Paul, Traylen, William, Lambert, Kim, Young, Neil, Bunally, Shenaz, Summerfield, Scott G, Snell, Richard, Lad, Rakesh, Shi, Eric, Skinner, Steven, Shewchuk, Lisa, Watson, Allan J.B, Chung, Chun-wa, Pal, Sandeep, Holt, Dennis A, Kallander, Lara S, Prendergast, Joanne, Rivera, Katrina, Washburn, David G, Harpel, Mark R, Arico-Muendel, Christopher, Isidro-Llobet, Albert
Published in Bioconjugate chemistry (17.02.2021)
Published in Bioconjugate chemistry (17.02.2021)
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Journal Article
The discovery of potent blockers of the canonical transient receptor channels, TRPC3 and TRPC6, based on an anilino-thiazole pharmacophore
Washburn, David G., Holt, Dennis A., Dodson, Jason, McAtee, Jeff J., Terrell, Lamont R., Barton, Linda, Manns, Sharada, Waszkiewicz, Anna, Pritchard, Christina, Gillie, Dan J., Morrow, Dwight M., Davenport, Elizabeth A., Lozinskaya, Irina M., Guss, Jeffrey, Basilla, Jonathan B., Negron, Lorena Kallal, Klein, Michael, Willette, Robert N., Fries, Rusty E., Jensen, Timothy C., Xu, Xiaoping, Schnackenberg, Christine G., Marino, Joseph P.
Published in Bioorganic & medicinal chemistry letters (01.09.2013)
Published in Bioorganic & medicinal chemistry letters (01.09.2013)
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Journal Article
Design and synthesis of orally bioavailable serum and glucocorticoid-regulated kinase 1 (SGK1) inhibitors
Hammond, Marlys, Washburn, David G., Hoang, Tram H., Manns, Sharada, Frazee, James S., Nakamura, Hiroko, Patterson, Jaclyn R., Trizna, Walter, Wu, Charlene, Azzarano, Leonard M., Nagilla, Rakesh, Nord, Melanie, Trejo, Rebecca, Head, Martha S., Zhao, Baoguang, Smallwood, Angela M., Hightower, Kendra, Laping, Nicholas J., Schnackenberg, Christine G., Thompson, Scott K.
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
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Journal Article
Asymmetric Total Synthesis of Spongistatins 1 and 2
Crimmins, Michael T, Katz, Jason D, Washburn, David G, Allwein, Shawn P, McAtee, Laura F
Published in Journal of the American Chemical Society (22.05.2002)
Published in Journal of the American Chemical Society (22.05.2002)
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Journal Article
Synthesis and SAR of potent LXR agonists containing an indole pharmacophore
Washburn, David G., Hoang, Tram H., Campobasso, Nino, Smallwood, Angela, Parks, Derek J., Webb, Christine L., Frank, Kelly A., Nord, Melanie, Duraiswami, Chaya, Evans, Christopher, Jaye, Michael, Thompson, Scott K.
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
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Journal Article
Rational design of orally-active, pyrrolidine-based progesterone receptor partial agonists
Thompson, Scott K., Washburn, David G., Frazee, James S., Madauss, Kevin P., Hoang, Tram H., Lapinski, Leahann, Grygielko, Eugene T., Glace, Lindsay E., Trizna, Walter, Williams, Shawn P., Duraiswami, Chaya, Bray, Jeffrey D., Laping, Nicholas J.
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
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Journal Article
Synthesis and SAR of amino acid-derived heterocyclic progesterone receptor full and partial agonists
Hammond, Marlys, Patterson, Jaclyn R., Manns, Sharada, Hoang, Tram H., Washburn, David G., Trizna, Walter, Glace, Lindsay, Grygielko, Eugene T., Nagilla, Rakesh, Nord, Melanie, Fries, Harvey E., Minick, Douglas J., Laping, Nicholas J., Bray, Jeffrey D., Thompson, Scott K.
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
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Journal Article
Improving the developability profile of pyrrolidine progesterone receptor partial agonists
Kallander, Lara S., Washburn, David G., Hoang, Tram H., Frazee, James S., Stoy, Patrick, Johnson, Latisha, Lu, Qing, Hammond, Marlys, Barton, Linda S., Patterson, Jaclyn R., Azzarano, Leonard M., Nagilla, Rakesh, Madauss, Kevin P., Williams, Shawn P., Stewart, Eugene L., Duraiswami, Chaya, Grygielko, Eugene T., Xu, Xiaoping, Laping, Nicholas J., Bray, Jeffrey D., Thompson, Scott K.
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
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Journal Article
Discovery of orally active, pyrrolidinone-based progesterone receptor partial agonists
Washburn, David G., Hoang, Tram H., Frazee, James S., Johnson, Latisha, Hammond, Marlys, Manns, Sharada, Madauss, Kevin P., Williams, Shawn P., Duraiswami, Chaya, Tran, Thuy B., Stewart, Eugene L., Grygielko, Eugene T., Glace, Lindsay E., Trizna, Walter, Nagilla, Rakesh, Bray, Jeffrey D., Thompson, Scott K.
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
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NAV1.8 억제제로서의 2,3-디히드로퀴나졸린 화합물
VIMAL MYTHILY, GUANG JIE, HO MING HSUN, HOANG TRAM H, YING MABEN, MILLER WILLIAM H, ELBAN MARK, WASHBURN DAVID G, DAVIS RODERICK S, ROMANO JOSEPH J
Year of Publication 10.03.2022
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Year of Publication 10.03.2022
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HYDROXY FORMAMIDE DERIVATIVES AND THEIR USE
HOANG TRAM H, LAWHORN BRIAN GRIFFIN, YE GUOSEN, DOWDELL SARAH E, ELBAN MARK, KALLANDER LARA S, WASHBURN DAVID G, PHILP JOANNE, HILFIKER MARK A, MANNS SHARADA, HAMMOND MARLYS, FOX RYAN MICHAEL, EIDAM HILARY SCHENCK
Year of Publication 12.09.2016
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Year of Publication 12.09.2016
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2,3-dihydroquinazolin compounds as NAV1.8 inhibitors
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Year of Publication 14.12.2023
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Year of Publication 14.12.2023
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Compuestos 2,3-dihidroquinazolin como inhibidores nav1 .8
HOANG, Tram H, MILLER, William H, ELBAN, Mark, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 21.04.2023
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Year of Publication 21.04.2023
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2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS
ELBAN, Mark, HOANG, Tram H, MILLER, William H, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 06.04.2023
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Year of Publication 06.04.2023
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2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS
HOANG, Tram H, MILLER, William H, ELBAN, Mark, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 04.05.2022
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Year of Publication 04.05.2022
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COMPOSÉS 2,3-DIHYDROQUINAZOLINE EN TANT QU'INHIBITEURS DE NAV1.8
ELBAN, Mark, HOANG, Tram H, MILLER, William H, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 04.05.2022
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Year of Publication 04.05.2022
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2,3-dihydroquinazolin compounds as NAV1.8 inhibitors
HOANG, Tram H, MILLER, William H, ELBAN, Mark, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 27.01.2022
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Year of Publication 27.01.2022
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2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS
HOANG, Tram H, MILLER, William H, ELBAN, Mark, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 30.12.2020
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Year of Publication 30.12.2020
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