Discovery of a Novel, First-in-Class, Orally Bioavailable Azaindole Inhibitor (VX-787) of Influenza PB2
Clark, Michael P, Ledeboer, Mark W, Davies, Ioana, Byrn, Randal A, Jones, Steven M, Perola, Emanuele, Tsai, Alice, Jacobs, Marc, Nti-Addae, Kwame, Bandarage, Upul K, Boyd, Michael J, Bethiel, Randy S, Court, John J, Deng, Hongbo, Duffy, John P, Dorsch, Warren A, Farmer, Luc J, Gao, Huai, Gu, Wenxin, Jackson, Katrina, Jacobs, Dylan H, Kennedy, Joseph M, Ledford, Brian, Liang, Jianglin, Maltais, François, Murcko, Mark, Wang, Tiansheng, Wannamaker, M. Woods, Bennett, Hamilton B, Leeman, Joshua R, McNeil, Colleen, Taylor, William P, Memmott, Christine, Jiang, Min, Rijnbrand, Rene, Bral, Christopher, Germann, Ursula, Nezami, Azin, Zhang, Yuegang, Salituro, Francesco G, Bennani, Youssef L, Charifson, Paul S
Published in Journal of medicinal chemistry (14.08.2014)
Published in Journal of medicinal chemistry (14.08.2014)
Get full text
Journal Article
Discovery of VX-509 (Decernotinib): A Potent and Selective Janus Kinase 3 Inhibitor for the Treatment of Autoimmune Diseases
Farmer, Luc J, Ledeboer, Mark W, Hoock, Thomas, Arnost, Michael J, Bethiel, Randy S, Bennani, Youssef L, Black, James J, Brummel, Christopher L, Chakilam, Ananthsrinivas, Dorsch, Warren A, Fan, Bin, Cochran, John E, Halas, Summer, Harrington, Edmund M, Hogan, James K, Howe, David, Huang, Hui, Jacobs, Dylan H, Laitinen, Leena M, Liao, Shengkai, Mahajan, Sudipta, Marone, Valerie, Martinez-Botella, Gabriel, McCarthy, Pamela, Messersmith, David, Namchuk, Mark, Oh, Luke, Penney, Marina S, Pierce, Albert C, Raybuck, Scott A, Rugg, Arthur, Salituro, Francesco G, Saxena, Kumkum, Shannon, Dean, Shlyakter, Dina, Swenson, Lora, Tian, Shi-Kai, Town, Christopher, Wang, Jian, Wang, Tiansheng, Wannamaker, M. Woods, Winquist, Raymond J, Zuccola, Harmon J
Published in Journal of medicinal chemistry (24.09.2015)
Published in Journal of medicinal chemistry (24.09.2015)
Get full text
Journal Article
Discovery of Novel Thiophene-Based, Thumb Pocket 2 Allosteric Inhibitors of the Hepatitis C NS5B Polymerase with Improved Potency and Physicochemical Profiles
Court, John J, Poisson, Carl, Ardzinski, Andrzej, Bilimoria, Darius, Chan, Laval, Chandupatla, Kishan, Chauret, Nathalie, Collier, Philip N, Das, Sanjoy Kumar, Denis, Francois, Dorsch, Warren, Iyer, Ganesh, Lauffer, David, L’Heureux, Lucille, Li, Pan, Luisi, Brian S, Mani, Nagraj, Nanthakumar, Suganthi, Nicolas, Olivier, Rao, B. Govinda, Ronkin, Steven, Selliah, Subajini, Shawgo, Rebecca S, Tang, Qing, Waal, Nathan D, Yannopoulos, Constantin G, Green, Jeremy
Published in Journal of medicinal chemistry (14.07.2016)
Published in Journal of medicinal chemistry (14.07.2016)
Get full text
Journal Article
PTERIDINONE COMPOUNDS AND USES THEREOF
GU WENXIN, MARINA PENNEY, LEDFORD BRIAN, MALTAIS FRANCOIS, DAVID DEININGER, NATHAN D WAAL, MARK WILLEM LEDEBOER, LI PAN, DENG HONGBO, LAUFFER DAVID J, GUY BEMIS, RUSSELL R HOOVER, MAC ARTHUR JOHNSON JR, DARIN TAKEMOTO, WANG TIANSHENG, MICHAEL BOYD, WARREN DORSCH
Year of Publication 22.08.2023
Get full text
Year of Publication 22.08.2023
Patent
ANTIPROLIFERATIVE COMPOUNDS AND USES THEREOF
STEVEN RONKIN, TANG QING, CLARKE MICHAEL, MARINA PENNEY, NATHAN D WAAL, LI PAN, DENG HONGBO, DONG HUIJUN, PHILIP COLLIER, LAUFFER DAVID J, GUY BEMIS, RUSSELL R HOOVER, HENRY YU, MAC ARTHUR JOHNSON JR, SHASHANK KUKAMI, DARIN TAKEMOTO, WANG TIANSHENG, MICHAEL BOYD, KISHAN CHANDUPATLA, WARREN DORSCH
Year of Publication 21.07.2023
Get full text
Year of Publication 21.07.2023
Patent
Discovery of Novel Allosteric HCV NS5B Inhibitors. 2. Lactam-Containing Thiophene Carboxylates
Li, Pan, Dorsch, Warren, Lauffer, David J., Bilimoria, Darius, Chauret, Nathalie, Court, John J., Das, Sanjoy Kumar, Denis, Francois, Mani, Nagraj, Nanthakumar, Suganthini, Nicolas, Olivier, Rao, B. Govinda, Ronkin, Steven, Selliah, Subajini, Shawgo, Rebecca S., Stearns, Ralph, Tang, Qing, Waal, Nathan D., Green, Jeremy
Published in ACS medicinal chemistry letters (09.02.2017)
Published in ACS medicinal chemistry letters (09.02.2017)
Get full text
Journal Article
PTERIDINONE COMPOUNDS AND USES THEREOF
Takemoto, Darin, Li, Pan, Gu, Wenxin, Bemis, Guy, Dorsch, Warren, Boyd, Michael, Deng, Hongbo, Wang, Tiansheng, Ledeboer, Mark Willem, Penney, Marina, Ledford, Brian, LAUFFER, David, Maltais, Francois, Deininger, David, Waal, Nathan D, Hoover, Russell R, Johnson, JR., Mac Arthur
Year of Publication 05.10.2023
Get full text
Year of Publication 05.10.2023
Patent
Inhibitors of APOL1 and methods of using same
Sayegh, Camil, Shi, Yi, Nicolas, Olivier, Fortier, Anne, Hamel, Martine, Wang, Tiansheng, Hu, Kan-Nian, Gagnon, Kevin, Witkos, Faith, Rose, Peter, Come, Jon H, Senter, Timothy J, Nanthakumar, Suganthini S, Krueger, Elaine B, Ledford, Brian, Dorsch, Warren A, Denis, Francois, Brodney, Michael, Cao, Jingrong, Shrestha, Muna, Medek, Ales, Dakin, Leslie A
Year of Publication 13.08.2024
Get full text
Year of Publication 13.08.2024
Patent
ANTIPROLIFERATION COMPOUNDS AND USES THEREOF
WANG, Tiansheng, LAUFFER, David J, JOHNSON, Mac, Arthur, JR, WAAL, Nathan, D, YU, Henry, HOOVER, Russell, R, KULKARNI, Shashank, COLLIER, Philip, BEMIS, Guy, TAKEMOTO, Darin, DONG, Huijun, CHANDUPATLA, Kishan, CLARK, Michael, PENNEY, Marina, LI, Pan, DENG, Hongbo, RONKIN, Steven, DORSCH, Warren, BOYD, Michael, TANG, Qing
Year of Publication 05.06.2024
Get full text
Year of Publication 05.06.2024
Patent
INHIBITORS OF APOL1 AND USE OF THE SAME
CAO, Jingrong, WANG, Tiansheng, LEDFORD, Brian, SENTER, Timothy J, SAYEGH, Camil E, DENIS, Francois, FORTIER, Anne, NICOLAS, Olivier, DORSCH, Warren A, COME, Jon H, KRUEGER, Elaine B, HAMEL, Martine, NANTHAKUMAR, Suganthini S, DAKIN, Leslie A, MALTAIS, Francois
Year of Publication 19.04.2023
Get full text
Year of Publication 19.04.2023
Patent