Preparation of Saxagliptin, a Novel DPP-IV Inhibitor
Savage, Scott A, Jones, Gregory S, Kolotuchin, Sergei, Ramrattan, Shelly Ann, Vu, Truc, Waltermire, Robert E
Published in Organic process research & development (20.11.2009)
Published in Organic process research & development (20.11.2009)
Get full text
Journal Article
The Effect of Additives on the Zinc Carbenoid-Mediated Cyclopropanation of a Dihydropyrrole
Ramirez, Antonio, Truc, Vu Chi, Lawler, Michael, Ye, Yun K, Wang, Jianji, Wang, Chenchi, Chen, Steven, Laporte, Thomas, Liu, Nian, Kolotuchin, Sergei, Jones, Scott, Bordawekar, Shailendra, Tummala, Srinivas, Waltermire, Robert E, Kronenthal, David
Published in Journal of organic chemistry (03.07.2014)
Published in Journal of organic chemistry (03.07.2014)
Get full text
Journal Article
Process Development for a Large Scale Stereoselective Synthesis of (Z)-(1-Bromobut-1-ene-1,2-diyl)dibenzene, a Key Intermediate of a Selective Estrogen Receptor Modulator
Cann, Reginald O, Waltermire, Robert E, Chung, Jihchin, Oberholzer, Matthew, Kasparec, Jiri, Ye, Yun K, Wethman, Robert
Published in Organic process research & development (17.09.2010)
Published in Organic process research & development (17.09.2010)
Get full text
Journal Article
Kilogram Synthesis of a Second-Generation LFA-1/ICAM Inhibitor
DelMonte, Albert J, Fan, Yu, Girard, Kevin P, Jones, Gregory S, Waltermire, Robert E, Rosso, Victor, Wang, Xuebao
Published in Organic process research & development (21.01.2011)
Published in Organic process research & development (21.01.2011)
Get full text
Journal Article
The First Kilogram Synthesis of Beclabuvir, an HCV NS5B Polymerase Inhibitor
Bien, Jeffrey, Davulcu, Akin, DelMonte, Albert J, Fraunhoffer, Kenneth J, Gao, Zhinong, Hang, Chao, Hsiao, Yi, Hu, Wenhao, Katipally, Kishta, Littke, Adam, Pedro, Aghogho, Qiu, Yuping, Sandoval, Maria, Schild, Richard, Soltani, Michelle, Tedesco, Anthony, Vanyo, Dale, Vemishetti, Purushotham, Waltermire, Robert E
Published in Organic process research & development (19.10.2018)
Published in Organic process research & development (19.10.2018)
Get full text
Journal Article
Efficient Preparation of a Key Intermediate in the Synthesis of Roxifiban by Enzymatic Dynamic Kinetic Resolution on Large Scale
Pesti, Jaan A, Yin, Jinguao, Zhang, Lin-hua, Anzalone, Luigi, Waltermire, Robert E, Ma, Philip, Gorko, Edward, Confalone, Pat N, Fortunak, Joseph, Silverman, Charlotte, Blackwell, John, Chung, J. C, Hrytsak, Michael D, Cooke, Mary, Powell, Lakisha, Ray, Charles
Published in Organic process research & development (01.01.2004)
Published in Organic process research & development (01.01.2004)
Get full text
Journal Article
Quaternary Chiral Center via Diastereoselective Enolate Amination Enables the Synthesis of an Anti-inflammatory Agent
Magnus, Nicholas A, Campagna, Silvio, Confalone, Pat N, Savage, Scott, Meloni, David J, Waltermire, Robert E, Wethman, Robert G, Yates, Mathew
Published in Organic process research & development (15.01.2010)
Published in Organic process research & development (15.01.2010)
Get full text
Journal Article
Selective deprotection of trialkylsilyl ethers using fluorosilicic acid
Pilcher, Anthony S, Hill, David K, Shimshock, Stephen J, Waltermire, Robert E, DeShong, Philip
Published in Journal of organic chemistry (01.04.1992)
Published in Journal of organic chemistry (01.04.1992)
Get full text
Journal Article
Kilogram Synthesis of a LFA-1/ICAM Inhibitor
DelMonte, Albert J, Waltermire, Robert E, Fan, Yu, McLeod, Douglas D, Gao, Zhinong, Gesenberg, Kirsten D, Girard, Kevin P, Rosingana, Miguel, Wang, Xuebao, Kuehne-Willmore, Jennifer, Braem, Alan D, Castoro, John A
Published in Organic process research & development (21.05.2010)
Published in Organic process research & development (21.05.2010)
Get full text
Journal Article
A general approach to the stereoselective synthesis of spiroketals. A total synthesis of the pheromones of the olive fruit fly and related compounds
DeShong, Philip, Waltermire, Robert E, Ammon, Herman L
Published in Journal of the American Chemical Society (01.03.1988)
Published in Journal of the American Chemical Society (01.03.1988)
Get full text
Journal Article
Synthesis, antiviral activity and pharmacokinetics of P1/P1′ substituted 3-aminoindazole cyclic urea HIV protease inhibitors
Kaltenbach, Robert F, Patel, Mona, Waltermire, Robert E, Harris, Gregory D, Stone, Benjamin R.P, Klabe, Ronald M, Garber, Sena, Bacheler, Lee T, Cordova, Beverly C, Logue, Kelly, Wright, Matthew R, Erickson-Viitanen, Susan, Trainor, George L
Published in Bioorganic & medicinal chemistry letters (24.02.2003)
Published in Bioorganic & medicinal chemistry letters (24.02.2003)
Get full text
Journal Article
Stereoselective Synthesis of HIV-1 Protease Inhibitor, DMP 323
Pierce, Michael E, Harris, Gregory D, Islam, Qamrul, Radesca, Lilian A, Storace, Louis, Waltermire, Robert E, Wat, Ed, Jadhav, Prabhakar K, Emmett, George C
Published in Journal of organic chemistry (26.01.1996)
Published in Journal of organic chemistry (26.01.1996)
Get full text
Journal Article
A total synthesis of (.+-.)-tirandamycin B
Shimshock, Stephen J, Waltermire, Robert E, DeShong, Philip
Published in Journal of the American Chemical Society (01.11.1991)
Published in Journal of the American Chemical Society (01.11.1991)
Get full text
Journal Article
Empirical relationship between chiral selectivity and mobile phase modifier properties
Blackwell, John A., Stringham, Rodger W., Xiang, Dong, Waltermire, Robert E.
Published in Journal of Chromatography A (13.08.1999)
Published in Journal of Chromatography A (13.08.1999)
Get full text
Journal Article
An Efficient Large-Scale Process for the Human Leukocyte Elastase Inhibitor, DMP 777 1
Storace, Louis, Anzalone, Luigi, Confalone, Pat N., Davis, Wayne P., Fortunak, Joseph M., Giangiordano, Mark, Haley, James J., Kamholz, Kenneth, Li, Hui-Yin, Ma, Philip, Nugent, William A., Parsons, Rodney L., Sheeran, Patrick J., Silverman, Charlotte E., Waltermire, Robert E., Wood, Christopher C.
Published in Organic process research & development (01.01.2002)
Published in Organic process research & development (01.01.2002)
Get full text
Journal Article
CRYSTALLINE FORMS AND PROCESS FOR PREPARING SPIRO-HYDANTOIN COMPOUNDS
WEI CHENKOU, MCLEOD DOUGLAS D, DHAR T.G. MURALI, MALLEY MARY F, FAN YU, DELMONTE ALBERT J, WALTERMIRE ROBERT E, GOUGOUTAS JACK Z
Year of Publication 30.10.2008
Get full text
Year of Publication 30.10.2008
Patent
Crystalline forms and process for preparing spiro-hydantoin compounds
DelMonte, Albert J, Dhar, T. G. Murali, Fan, Yu, Gougoutas, Jack Z, Malley, Mary F, McLeod, Douglas D, Waltermire, Robert E, Wei, Chenkou
Year of Publication 03.06.2008
Get full text
Year of Publication 03.06.2008
Patent