Anxiolytic- and Antidepressant-like Effects of the Non-Peptide Vasopressin V1b Receptor Antagonist, SSR149415, Suggest an Innovative Approach for the Treatment of Stress-Related Disorders
Griebel, Guy, Simiand, Jacques, Gal, Claudine Serradeil-Le, Wagnon, Jean, Pascal, Marc, Scatton, Bernard, Maffrand, Jean-Pierre, Soubrié, Philippe
Published in Proceedings of the National Academy of Sciences - PNAS (30.04.2002)
Published in Proceedings of the National Academy of Sciences - PNAS (30.04.2002)
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Characterization of (2S,4R)-1-[5-Chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxy-phenyl)-2-oxo-2,3-dihydro-1H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidine carboxamide (SSR149415), a Selective and Orally Active Vasopressin V1b Receptor Antagonist
Serradeil-Le Gal, Claudine, Wagnon, Jean, Simiand, Jacques, Griebel, Guy, Lacour, Colette, Guillon, Gilles, Barberis, Claude, Brossard, Gabrielle, Soubrié, Philippe, Nisato, Dino, Pascal, Marc, Pruss, Rebecca, Scatton, Bernard, Maffrand, Jean-Pierre, Le Fur, Gérard
Published in The Journal of pharmacology and experimental therapeutics (01.03.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2002)
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Journal Article
Anxiolytic- and antidepressant-like effects of the non-peptide vasopressin V 1b receptor antagonist, SSR149415, suggest an innovative approach for the treatment of stress-related disorders
Griebel, Guy, Simiand, Jacques, Serradeil-Le Gal, Claudine, Wagnon, Jean, Pascal, Marc, Scatton, Bernard, Maffrand, Jean-Pierre, Soubrié, Philippe
Published in Proceedings of the National Academy of Sciences - PNAS (30.04.2002)
Published in Proceedings of the National Academy of Sciences - PNAS (30.04.2002)
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Journal Article
Biological characterization of rodent and human vasopressin V 1b receptors using SSR-149415, a nonpeptide V 1b receptor ligand
Gal, Claudine Serradeil-Le, Raufaste, Danièle, Derick, Sylvain, Blankenstein, Jörg, Allen, John, Pouzet, Brigitte, Pascal, Marc, Wagnon, Jean, Ventura, Maria Angeles
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.08.2007)
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.08.2007)
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Journal Article
Biological characterization of rodent and human vasopressin V sub(1b) receptors using SSR-149415, a nonpeptide V sub(1b) receptor ligand
Gal, Claudine Serradeil-Le, Raufaste, Daniele, Derick, Sylvain, Blankenstein, Joerg, Allen, John, Pouzet, Brigitte, Pascal, Marc, Wagnon, Jean, Ventura, Maria Angeles
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.08.2007)
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Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.08.2007)
Journal Article
Biological characterization of rodent and human vasopressin V1b receptors using SSR-149415, a nonpeptide V1b receptor ligand
SERRADEIL-LE GAL, Claudine, RAUFASTE, Danièle, DERICK, Sylvain, BLANKENSTEIN, Jörg, ALLEN, John, POUZET, Brigitte, PASCAL, Marc, WAGNON, Jean, VENTURA, Maria Angeles
Published in American journal of physiology. Regulatory, integrative and comparative physiology (2007)
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Published in American journal of physiology. Regulatory, integrative and comparative physiology (2007)
Journal Article
Biological characterization of rodent and human vasopressin V1b receptors using SSR-149415, a nonpeptide V1b receptor ligand
Gal, Claudine Serradeil-Le, Raufaste, Daniele, Derick, Sylvain, Blankenstein, Jorg, Allen, John, Pouzet, Brigitte, Pascal, Marc, Wagnon, Jean, Ventura, Maria Angeles
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.08.2007)
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.08.2007)
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Journal Article
Anxiolytic- and antidepressant-like effects of the non-pepetide vasopressin V1b receptor antagonist, SSR149415, suggest an innovative approach for the treatment of stress-related
Griebel, Guy, Simiand, Jacques, Claudine Serradeil-Le Gal, Wagnon, Jean
Published in Proceedings of the National Academy of Sciences - PNAS (30.04.2002)
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Published in Proceedings of the National Academy of Sciences - PNAS (30.04.2002)
Journal Article
An overview of SSR149415, a selective nonpeptide vasopressin V(1b) receptor antagonist for the treatment of stress-related disorders
Serradeil-Le Gal, Claudine, Wagnon, 3rd, Jean, Tonnerre, Bernard, Roux, Richard, Garcia, Georges, Griebel, Guy, Aulombard, Alain
Published in CNS drug reviews (2005)
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Published in CNS drug reviews (2005)
Journal Article
Characterization of (2 S ,4 R )-1-[5-Chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxy-phenyl)-2-oxo-2,3-dihydro-1 H -indol-3-yl]-4-hydroxy- N , N -dimethyl-2-pyrrolidine carboxamide (SSR149415), a Selective and Orally Active Vasopressin V 1b Receptor Antagonist
Gal, Claudine Serradeil-Le, Wagnon, Jean, Simiand, Jacques, Griebel, Guy, Lacour, Colette, Guillon, Gilles, Barberis, Claude, Brossard, Gabrielle, Soubrié, Philippe, Nisato, Dino, Pascal, Marc, Pruss, Rebecca, Scatton, Bernard, Maffrand, Jean-Pierre, Le Fur, Gérard
Published in The Journal of pharmacology and experimental therapeutics (01.03.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.03.2002)
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Journal Article
COMPUESTOS DERIVADOS DE FENIL-(4-FENIL PIRIMIDIN-2-IL)-AMINAS; COMPOSICION FARMACEUTICA QUE COMPRENDE A DICHOS COMPUESTOS ; PROCEDIMIENTO DE PREPARACION DE DICHOS COMPUESTOS; Y SU USO EN ENFERMEDADES INFLAMATORIAS, DIABETES Y CANCER
BOUABOULA MONSIF,CASELLAS PIERRE,DUDA SHERRI,FLUTARD REGINE,NGUEFACK JEAN-FLAUBERT,TONNERRRE BERNARD,WAGNON JEAN,MENDEZ
Year of Publication 16.05.2008
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Year of Publication 16.05.2008
Patent
An Overview of SSR149415, a Selective Nonpeptide Vasopressin V1b Receptor Antagonist for the Treatment of Stress‐Related Disorders
Gal, Claudine Serradeil‐Le, Wagnon, Jean, Tonnerre, Bernard, Roux, Richard, Garcia, Georges, Griebel, Guy, Aulombard, Alain
Published in CNS drug reviews (01.03.2005)
Published in CNS drug reviews (01.03.2005)
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Journal Article