Rational Development of Practical Catalysts for Aromatic Carbon−Nitrogen Bond Formation
Wolfe, John P, Wagaw, Seble, Marcoux, Jean-François, Buchwald, Stephen L
Published in Accounts of chemical research (22.12.1998)
Published in Accounts of chemical research (22.12.1998)
Get full text
Journal Article
Validation of Diacyl Glycerolacyltransferase I as a Novel Target for the Treatment of Obesity and Dyslipidemia Using a Potent and Selective Small Molecule Inhibitor
Zhao, Gang, Souers, Andrew J, Voorbach, Martin, Falls, H. Doug, Droz, Brian, Brodjian, Sevan, Lau, Yau Yi, Iyengar, Rajesh R, Gao, Ju, Judd, Andrew S, Wagaw, Seble H, Ravn, Matthew M, Engstrom, Kenneth M, Lynch, John K, Mulhern, Mathew M, Freeman, Jennifer, Dayton, Brian D, Wang, Xiaojun, Grihalde, Nelson, Fry, Dennis, Beno, David W. A, Marsh, Kennan C, Su, Zhi, Diaz, Gilbert J, Collins, Christine A, Sham, Hing, Reilly, Regina M, Brune, Michael E, Kym, Philip R
Published in Journal of medicinal chemistry (14.02.2008)
Published in Journal of medicinal chemistry (14.02.2008)
Get full text
Journal Article
Development of a Catalytic Enantioselective Conjugate Addition of 1,3-Dicarbonyl Compounds to Nitroalkenes for the Synthesis of Endothelin-A Antagonist ABT-546. Scope, Mechanism, and Further Application to the Synthesis of the Antidepressant Rolipram
Barnes, David M, Ji, Jianguo, Fickes, Michael G, Fitzgerald, Michael A, King, Steven A, Morton, Howard E, Plagge, Frederick A, Preskill, Margo, Wagaw, Seble H, Wittenberger, Steven J, Zhang, Ji
Published in Journal of the American Chemical Society (06.11.2002)
Published in Journal of the American Chemical Society (06.11.2002)
Get full text
Journal Article
A Palladium-Catalyzed Method for the Preparation of Indoles via the Fischer Indole Synthesis
Wagaw, Seble, Yang, Bryant H, Buchwald, Stephen L
Published in Journal of the American Chemical Society (10.11.1999)
Published in Journal of the American Chemical Society (10.11.1999)
Get full text
Journal Article
Development of a Scalable Synthesis of Dipeptidyl Peptidase-4 Inhibitor ABT-279
McDermott, Todd S, Bhagavatula, Lakshmi, Borchardt, Thomas B, Engstrom, Kenneth M, Gandarilla, Jorge, Kotecki, Brian J, Kruger, Albert W, Rozema, Michael J, Sheikh, Ahmad Y, Wagaw, Seble H, Wittenberger, Steven J
Published in Organic process research & development (20.11.2009)
Published in Organic process research & development (20.11.2009)
Get full text
Journal Article
Process Development of a Diacyl Glycerolacyltransferase-1 Inhibitor
Ravn, Matthew M, Wagaw, Seble H, Engstrom, Kenneth M, Mei, Jianzhang, Kotecki, Brian, Souers, Andrew J, Kym, Philip R, Judd, Andrew S, Zhao, Gang
Published in Organic process research & development (19.03.2010)
Published in Organic process research & development (19.03.2010)
Get full text
Journal Article
An Improved Catalyst System for Aromatic Carbon−Nitrogen Bond Formation: The Possible Involvement of Bis(Phosphine) Palladium Complexes as Key Intermediates
Wolfe, John P, Wagaw, Seble, Buchwald, Stephen L
Published in Journal of the American Chemical Society (31.07.1996)
Published in Journal of the American Chemical Society (31.07.1996)
Get full text
Journal Article
Gram Scale Synthesis of the Glucuronide Metabolite of ABT-724
Engstrom, Kenneth M, Daanen, Jerome F, Wagaw, Seble, Stewart, Andrew O
Published in Journal of organic chemistry (27.10.2006)
Published in Journal of organic chemistry (27.10.2006)
Get full text
Journal Article
Screening for Cardiovascular Safety: A Structure−Activity Approach for Guiding Lead Selection of Melanin Concentrating Hormone Receptor 1 Antagonists
Kym, Philip R, Souers, Andrew J, Campbell, Thomas J, Lynch, John K, Judd, Andrew S, Iyengar, Rajesh, Vasudevan, Anil, Gao, Ju, Freeman, Jennifer C, Wodka, Dariusz, Mulhern, Mathew, Zhao, Gang, Wagaw, Seble H, Napier, James J, Brodjian, Sevan, Dayton, Brian D, Reilly, Regina M, Segreti, Jason A, Fryer, Ryan M, Preusser, Lee C, Reinhart, Glenn A, Hernandez, Lisa, Marsh, Kennan C, Sham, Hing L, Collins, Christine A, Polakowski, James S
Published in Journal of medicinal chemistry (06.04.2006)
Published in Journal of medicinal chemistry (06.04.2006)
Get full text
Journal Article
Aminopiperidine indazoles as orally efficacious melanin concentrating hormone receptor-1 antagonists
Vasudevan, Anil, Souers, Andrew J., Freeman, Jennifer C., Verzal, Mary K., Gao, Ju, Mulhern, Mathew M., Wodka, Derek, Lynch, John K., Engstrom, Kenneth M., Wagaw, Seble H., Brodjian, Sevan, Dayton, Brian, Falls, Doug H., Bush, Eugene, Brune, Michael, Shapiro, Robin D., Marsh, Kennan C., Hernandez, Lisa E., Collins, Christine A., Kym, Philip R.
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
Published in Bioorganic & medicinal chemistry letters (01.12.2005)
Get full text
Journal Article
An Efficient, Stereoselective Synthesis of the Hydroxyethylene Dipeptide Isostere Core for the HIV Protease Inhibitor A-792611
Engstrom, Kenneth, Henry, Rodger, Hollis, L. Steven, Kotecki, Brian, Marsden, Ian, Pu, Yu-Ming, Wagaw, Seble, Wang, Weifeng
Published in Journal of organic chemistry (07.07.2006)
Published in Journal of organic chemistry (07.07.2006)
Get full text
Journal Article
Process development of ABT-450 – A first generation NS3/4A protease inhibitor for HCV
Caspi, Daniel D., Cink, Russell D., Clyne, Dean, Diwan, Moiz, Engstrom, Kenneth M., Grieme, Timothy, Mei, Jianzhang, Miller, Robert W., Mitchell, Clifford, Napolitano, José G., Nere, Nandkishor, Ravn, Matthew M., Sheikh, Ahmad, Wagaw, Seble, Zhang, Hongqiang
Published in Tetrahedron (09.08.2019)
Published in Tetrahedron (09.08.2019)
Get full text
Journal Article
Palladium-Catalyzed Coupling of Optically Active Amines with Aryl Bromides
Wagaw, Seble, Rennels, Roger A., Buchwald, Stephen L.
Published in Journal of the American Chemical Society (10.09.1997)
Published in Journal of the American Chemical Society (10.09.1997)
Get full text
Journal Article
Discovery of adamantane ethers as inhibitors of 11β-HSD-1: Synthesis and biological evaluation
Patel, Jyoti R., Shuai, Qi, Dinges, Jurgen, Winn, Marty, Pliushchev, Marina, Fung, Steven, Monzon, Katina, Chiou, William, Wang, Jiahong, Pan, Liping, Wagaw, Seble, Engstrom, Kenneth, Kerdesky, Francis A., Longenecker, Kenton, Judge, Russell, Qin, Wenying, Imade, Hovis M., Stolarik, DeAnne, Beno, David W.A., Brune, Michael, Chovan, Linda E., Sham, Hing L., Jacobson, Peer, Link, J.T.
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
Published in Bioorganic & medicinal chemistry letters (01.02.2007)
Get full text
Journal Article
Chlorination at the 8-Position of a Functionalized Quinolone and the Synthesis of Quinolone Antibiotic ABT-492
Barnes, David M, Christesen, Alan C, Engstrom, Kenneth M, Haight, Anthony R, Hsu, Margaret C, Lee, Elaine C, Peterson, Matthew J, Plata, Daniel J, Raje, Prasad S, Stoner, Eric J, Tedrow, Jason S, Wagaw, Seble
Published in Organic process research & development (21.07.2006)
Published in Organic process research & development (21.07.2006)
Get full text
Journal Article