Exploring protein hotspots by optimized fragment pharmacophores
Bajusz, Dávid, Wade, Warren S, Satała, Grzegorz, Bojarski, Andrzej J, Ilaš, Janez, Ebner, Jessica, Grebien, Florian, Papp, Henrietta, Jakab, Ferenc, Douangamath, Alice, Fearon, Daren, von Delft, Frank, Schuller, Marion, Ahel, Ivan, Wakefield, Amanda, Vajda, Sándor, Gerencsér, János, Pallai, Péter, Keserű, György M
Published in Nature communications (27.05.2021)
Published in Nature communications (27.05.2021)
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Journal Article
Central nervous system origins of the sympathetic nervous system outflow to white adipose tissue
Bamshad, Maryam, Aoki, Victor T, Adkison, M. Gregory, Warren, Wade S, Bartness, Timothy J
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.07.1998)
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.07.1998)
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Journal Article
Pharmacological Characterization of CXC Chemokine Receptor 3 Ligands and a Small Molecule Antagonist
Heise, Christopher E, Pahuja, Anil, Hudson, Sarah C, Mistry, Monica S, Putnam, Amy L, Gross, Molly M, Gottlieb, Peter A, Wade, Warren S, Kiankarimi, Mehrak, Schwarz, David, Crowe, Paul, Zlotnik, Albert, Alleva, David G
Published in The Journal of pharmacology and experimental therapeutics (01.06.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2005)
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Journal Article
Structure and ligand recognition of the phosphotyrosine binding domain of Shc
Zhou, Ming-Ming, Ravichandran, Kodimangalam S, Olejniczak, Edward T, Petros, Andrew M, Meadows, Robert P, Sattler, Michael, Harlan, John E, Wade, Warren S, Burakoff, Steven J, Fesik, Stephen W
Published in Nature (London) (07.12.1995)
Published in Nature (London) (07.12.1995)
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Journal Article
Synthesis and structure–activity relationships of selective norepinephrine reuptake inhibitors (sNRI) with a heterocyclic ring constraint
Hudson, Sarah, Kiankarimi, Mehrak, Eccles, Wendy, Mostofi, Yalda S., Genicot, Marc J., Dwight, Wesley, Fleck, Beth A., Gogas, Kathleen, Wade, Warren S.
Published in Bioorganic & medicinal chemistry (15.08.2008)
Published in Bioorganic & medicinal chemistry (15.08.2008)
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Journal Article
Discovery of a potent, selective, and less flexible selective norepinephrine reuptake inhibitor (sNRI)
Wu, Dongpei, Pontillo, Joseph, Ching, Brett, Hudson, Sarah, Gao, Yinghong, Fleck, Beth A., Gogas, Kathleen, Wade, Warren S.
Published in Bioorganic & medicinal chemistry (15.07.2008)
Published in Bioorganic & medicinal chemistry (15.07.2008)
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Journal Article
모노아실글리세롤 리파아제 조절제로서의 아릴 피페리딘
AMERIKS MICHAEL K, BERRY CYNTHIA B, SAMANT ANDREW V, BIRO KRISZTIAN, GARCIA REYNAGA PABLO, WADE WARREN S
Year of Publication 29.11.2022
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Year of Publication 29.11.2022
Patent
Synthesis and structure-activity relationships of selective norepinephrine reuptake inhibitors (sNRI) with improved pharmaceutical characteristics
PONTILLO, Joseph, DONGPEI WU, HUA WANG, WEN, Jenny, WADE, Warren S, CHINGA, Brett, HUDSON, Sarah, GENICOTA, Marc J, YINGHONG GAO, EWING, Todd, FLECK, Beth A, GOGAS, Kathleen, APARICIO, Anna
Published in Bioorganic & medicinal chemistry (01.12.2008)
Published in Bioorganic & medicinal chemistry (01.12.2008)
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Journal Article
Structure–activity relationships of chiral selective norepinephrine reuptake inhibitors (sNRI) with increased oxidative stability
Hudson, Sarah, Kiankarimi, Mehrak, Eccles, Wendy, Dwight, Wesley, Mostofi, Yalda S., Genicot, Marc J., Fleck, Beth A., Gogas, Kathleen, Aparicio, Anna, Wang, Hua, Wen, Jenny, Wade, Warren S.
Published in Bioorganic & medicinal chemistry (15.08.2008)
Published in Bioorganic & medicinal chemistry (15.08.2008)
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Journal Article
Synthesis and structure–activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 2
Hudson, Sarah, Kiankarimi, Mehrak, Rowbottom, Martin W., Vickers, Troy D., Wu, Dongpei, Pontillo, Joseph, Ching, Brett, Dwight, Wesley, Goodfellow, Val S., Schwarz, David, Heise, Christopher E., Madan, Ajay, Wen, Jenny, Ban, William, Wang, Hua, Wade, Warren S.
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
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Journal Article
Synthesis and structure–activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 1
Rowbottom, Martin W., Vickers, Troy D., Dyck, Brian, Grey, Jonathan, Tamiya, Junko, Zhang, Mingzhu, Kiankarimi, Mehrak, Wu, Dongpei, Dwight, Wesley, Wade, Warren S., Schwarz, David, Heise, Christopher E., Madan, Ajay, Fisher, Andrew, Petroski, Robert, Goodfellow, Val S.
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
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Journal Article
A high-throughput chemotaxis assay for pharmacological characterization of chemokine receptors: Utilization of U937 monocytic cells
Ott, Thomas R., Pahuja, Anil, Lio, Francisco M., Mistry, Monica S., Gross, Molly, Hudson, Sarah C., Wade, Warren S., Simpson, Pedro B., Struthers, R. Scott, Alleva, David G.
Published in Journal of pharmacological and toxicological methods (01.03.2005)
Published in Journal of pharmacological and toxicological methods (01.03.2005)
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Journal Article
Application of Base Cleavable Safety Catch Linkers to Solid Phase Library Production
Wade, Warren S, Yang, Fan, Sowin, Thomas J
Published in Journal of combinatorial chemistry (01.05.2000)
Published in Journal of combinatorial chemistry (01.05.2000)
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Journal Article
Engineering metal coordination sites into the antibody light chain
Wade, Warren S, Koh, Jong S, Han, Nianhe, Hoekstra, Denise M, Lerner, Richard A
Published in Journal of the American Chemical Society (01.06.1993)
Published in Journal of the American Chemical Society (01.06.1993)
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