Genome-wide association analysis identifies genetic correlates of immune infiltrates in solid tumors
Siemers, Nathan O, Holloway, James L, Chang, Han, Chasalow, Scott D, Ross-MacDonald, Petra B, Voliva, Charles F, Szustakowski, Joseph D
Published in PloS one (27.07.2017)
Published in PloS one (27.07.2017)
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Identification and characterization of NVP-BKM120, an orally available pan-class I PI3-kinase inhibitor
Maira, Sauveur-Michel, Pecchi, Sabina, Huang, Alan, Burger, Matthew, Knapp, Mark, Sterker, Dario, Schnell, Christian, Guthy, Daniel, Nagel, Tobi, Wiesmann, Marion, Brachmann, Saskia, Fritsch, Christine, Dorsch, Marion, Chène, Patrick, Shoemaker, Kevin, De Pover, Alain, Menezes, Daniel, Martiny-Baron, Georg, Fabbro, Doriano, Wilson, Christopher J, Schlegel, Robert, Hofmann, Francesco, García-Echeverría, Carlos, Sellers, William R, Voliva, Charles F
Published in Molecular cancer therapeutics (01.02.2012)
Published in Molecular cancer therapeutics (01.02.2012)
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Identification of NVP-BKM120 as a Potent, Selective, Orally Bioavailable Class I PI3 Kinase Inhibitor for Treating Cancer
Burger, Matthew T, Pecchi, Sabina, Wagman, Allan, Ni, Zhi-Jie, Knapp, Mark, Hendrickson, Thomas, Atallah, Gordana, Pfister, Keith, Zhang, Yanchen, Bartulis, Sarah, Frazier, Kelly, Ng, Simon, Smith, Aaron, Verhagen, Joelle, Haznedar, Joshua, Huh, Kay, Iwanowicz, Ed, Xin, Xiaohua, Menezes, Daniel, Merritt, Hanne, Lee, Isabelle, Wiesmann, Marion, Kaufman, Susan, Crawford, Kenneth, Chin, Michael, Bussiere, Dirksen, Shoemaker, Kevin, Zaror, Isabel, Maira, Sauveur-Michel, Voliva, Charles F
Published in ACS medicinal chemistry letters (13.10.2011)
Published in ACS medicinal chemistry letters (13.10.2011)
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Journal Article
Synthesis and in Vitro and in Vivo Evaluation of Phosphoinositide-3-kinase Inhibitors
Burger, Matthew T, Knapp, Mark, Wagman, Allan, Ni, Zhi-Jie, Hendrickson, Thomas, Atallah, Gordana, Zhang, Yanchen, Frazier, Kelly, Verhagen, Joelle, Pfister, Keith, Ng, Simon, Smith, Aaron, Bartulis, Sarah, Merrit, Hanne, Weismann, Marion, Xin, Xiaohua, Haznedar, Joshua, Voliva, Charles F, Iwanowicz, Ed, Pecchi, Sabina
Published in ACS medicinal chemistry letters (13.01.2011)
Published in ACS medicinal chemistry letters (13.01.2011)
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Journal Article
RAF-Mutant Melanomas Differentially Depend on ERK2 Over ERK1 to Support Aberrant MAPK Pathway Activation and Cell Proliferation
Crowe, Matthew S, Zavorotinskaya, Tatiana, Voliva, Charles F, Shirley, Matthew D, Wang, Yanqun, Ruddy, David A, Rakiec, Daniel P, Engelman, Jeffery A, Stuart, Darrin D, Freeman, Alyson K
Published in Molecular cancer research (01.06.2021)
Published in Molecular cancer research (01.06.2021)
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Journal Article
Discovery of imidazo[1,2-a]-pyridine inhibitors of pan-PI3 kinases that are efficacious in a mouse xenograft model
Han, Wooseok, Menezes, Daniel L., Xu, Yongjin, Knapp, Mark S., Elling, Robert, Burger, Matthew T., Ni, Zhi-Jie, Smith, Aaron, Lan, Jiong, Williams, Teresa E., Verhagen, Joelle, Huh, Kay, Merritt, Hanne, Chan, John, Kaufman, Susan, Voliva, Charles F., Pecchi, Sabina
Published in Bioorganic & medicinal chemistry letters (01.02.2016)
Published in Bioorganic & medicinal chemistry letters (01.02.2016)
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Journal Article
Identification and structure–activity relationship of 2-morpholino 6-(3-hydroxyphenyl) pyrimidines, a class of potent and selective PI3 kinase inhibitors
Pecchi, Sabina, Renhowe, Paul A., Taylor, Clarke, Kaufman, Susan, Merritt, Hanne, Wiesmann, Marion, Shoemaker, Kevin R., Knapp, Mark S., Ornelas, Elizabeth, Hendrickson, Thomas F., Fantl, Wendy, Voliva, Charles F.
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
Published in Bioorganic & medicinal chemistry letters (01.12.2010)
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Journal Article
Structure guided optimization of a fragment hit to imidazopyridine inhibitors of PI3K
Pecchi, Sabina, Ni, Zhi-Jie, Han, Wooseok, Smith, Aaron, Lan, Jiong, Burger, Matthew, Merritt, Hanne, Wiesmann, Marion, Chan, John, Kaufman, Susan, Knapp, Mark S., Janssen, Johanna, Huh, Kay, Voliva, Charles F.
Published in Bioorganic & medicinal chemistry letters (15.08.2013)
Published in Bioorganic & medicinal chemistry letters (15.08.2013)
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Journal Article
Recognition Properties of Antibodies to PAMAM Dendrimers and Their Use in Immune Detection of Dendrimers
Lee, Stephen C, Parthasarathy, Ranjani, Duffin, Tiffany D, Botwin, Kelly, Zobel, James, Beck, Theresa, Lange, Gary, Kunneman, David, Janssen, Robert, Rowold, Edwin, Voliva, Charles F
Published in Biomedical microdevices (01.03.2001)
Published in Biomedical microdevices (01.03.2001)
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Abstract 1140: A novel MTA non-competitive PRMT5 inhibitor
Malik, Rohit, Park, Peter K., Barbieri, Christopher M., Blat, Yuval, Sheriff, Steven, Weigelt, Carolyn A., Kopcho, Lisa M., Celiktas, Muge, Ruzanov, Max, Naglich, Joseph G., Price, Jennifer L., Harner, Mary, Omalley, Kevin M., Deng, JIngjing, Schmitz, William, Li, Guo, Ruan, Zheming, Qin, Lan-ying, Duke, Gerald J., Rodrigo, Iyoncy, Witmer, Mark R., Harden, David G., Demes, Shilpa, Arey, Brian J., Soars, Matt, Fink, Brian E., Gavai, Ashvinikumar V., Vite, Gregory D., Voliva, Charles F.
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Abstract 4497: NVP-BKM120, a novel inhibitor of phosphoinosotide 3-kinase in Phase I/II clinical trials, shows significant antitumor activity in xenograft and primary tumor models
Maira, Michel, Menezes, Daniel, Pecchi, Sabina, Shoemaker, Kevin, Burger, Matthew, Schnell, christian, Fritsch, christine, Brachmann, Saskia, Nagel, Tobi, Sellers, William R., Garcia-Echeverria, Carlos, Wiesmann, Marion, Voliva, charles F.
Published in Cancer research (Chicago, Ill.) (15.04.2010)
Published in Cancer research (Chicago, Ill.) (15.04.2010)
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Abstract 4498: Biological characterization of NVP-BKM120, a novel inhibitor of phosphoinosotide 3-kinase in Phase I/II clinical trials
Voliva, charles F., Pecchi, Sabina, Burger, Matthew, Nagel, Tobi, Schnell, Christian, Fritsch, christine, Brachmann, saskia, Menezes, Daniel, Knapp, Mark, Shoemaker, Kevin, Wiesmann, Marion, Huh, kay, Zaror, Isabel, Dorsch, Marion, Sellers, William R., Garcia-Echeverria, Carlos, Maira, Michel
Published in Cancer research (Chicago, Ill.) (15.04.2010)
Published in Cancer research (Chicago, Ill.) (15.04.2010)
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Journal Article
Conservation throughout mammalia and extensive protein-encoding capacity of the highly repeated DNA long interspersed sequence one
Burton, Frank H., Loeb, Daniel D., Voliva, Charles F., Martin, Sandra L., Edgell, Marshall H., Hutchison, Clyde A.
Published in Journal of molecular biology (20.01.1986)
Published in Journal of molecular biology (20.01.1986)
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Journal Article
DNA sequence organization of the β-globin complex in the BALB/c mouse
Jahn, Carolyn L., Hutchison, Clyde A., Phillips, Sandra J., Weaver, Steven, Haigwood, Nancy L., Voliva, Charles F., Edgell, Marshall H.
Published in Cell (01.08.1980)
Published in Cell (01.08.1980)
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A Large Interspersed Repeat Found in Mouse DNA Contains a Long Open Reading Frame That Evolves as If It Encodes a Protein
Martin, Sandra L., Voliva, Charles F., Burton, Frank H., Edgell, Marshall H., Hutchison, Clyde A.
Published in Proceedings of the National Academy of Sciences - PNAS (01.04.1984)
Published in Proceedings of the National Academy of Sciences - PNAS (01.04.1984)
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