Selecting the first chemical molecule inhibitor of HSP110 for colorectal cancer therapy
Gozzi, Gustavo J., Gonzalez, Daniel, Boudesco, Christophe, Dias, Alexandre M. M., Gotthard, Guillaume, Uyanik, Burhan, Dondaine, Lucile, Marcion, Guillaume, Hermetet, François, Denis, Camille, Hardy, Laurianne, Suzanne, Peggy, Douhard, Romain, Jego, Gaetan, Dubrez, Laurence, Demidov, Oleg N., Neiers, Fabrice, Briand, Loïc, Sopková-de Oliveira Santos, Jana, Voisin-Chiret, Anne-Sophie, Garrido, Carmen
Published in Cell death and differentiation (01.01.2020)
Published in Cell death and differentiation (01.01.2020)
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Synthesis of Pyridoclax Analogues: Insight into Their Druggability by Investigating Their Physicochemical Properties and Interactions with Membranes
De Pascale, Martina, Iacopetta, Domenico, Since, Marc, Corvaisier, Sophie, Vie, Véronique, Paboeuf, Gilles, Hennequin, Didier, Perato, Serge, De Giorgi, Marcella, Sinicropi, Maria Stefania, Sopkova‐De Oliveira Santos, Jana, Voisin‐Chiret, Anne‐Sophie, Malzert‐Freon, Aurélie
Published in ChemMedChem (07.01.2020)
Published in ChemMedChem (07.01.2020)
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Microplate assay for lipophilicity determination using intrinsic fluorescence of drugs: Application to a promising anticancer lead, pyridoclax
Smeralda, Willy, Since, Marc, Corvaisier, Sophie, Legay, Rémi, Voisin-Chiret, Anne-Sophie, Malzert-Freon, Aurélie
Published in European journal of pharmaceutical sciences (01.04.2019)
Published in European journal of pharmaceutical sciences (01.04.2019)
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Nutrient Requirements during Pregnancy and Lactation
Jouanne, Marie, Oddoux, Sarah, Noël, Antoine, Voisin-Chiret, Anne Sophie
Published in Nutrients (01.02.2021)
Published in Nutrients (01.02.2021)
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First Identification of Boronic Species as Novel Potential Inhibitors of the Staphylococcus aureus NorA Efflux Pump
Fontaine, Fanny, Hequet, Arnaud, Voisin-Chiret, Anne-Sophie, Bouillon, Alexandre, Lesnard, Aurélien, Cresteil, Thierry, Jolivalt, Claude, Rault, Sylvain
Published in Journal of medicinal chemistry (27.03.2014)
Published in Journal of medicinal chemistry (27.03.2014)
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Estrogen Receptor-α Targeting: PROTACs, SNIPERs, Peptide-PROTACs, Antibody Conjugated PROTACs and SNIPERs
Negi, Arvind, Kesari, Kavindra Kumar, Voisin-Chiret, Anne Sophie
Published in Pharmaceutics (01.11.2022)
Published in Pharmaceutics (01.11.2022)
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Boronic species as promising inhibitors of the Staphylococcus aureus NorA efflux pump: Study of 6-substituted pyridine-3-boronic acid derivatives
Fontaine, Fanny, Héquet, Arnaud, Voisin-Chiret, Anne-Sophie, Bouillon, Alexandre, Lesnard, Aurélien, Cresteil, Thierry, Jolivalt, Claude, Rault, Sylvain
Published in European journal of medicinal chemistry (05.05.2015)
Published in European journal of medicinal chemistry (05.05.2015)
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Light-Activating PROTACs in Cancer: Chemical Design, Challenges, and Applications
Negi, Arvind, Kesari, Kavindra Kumar, Voisin-Chiret, Anne Sophie
Published in Applied sciences (01.10.2022)
Published in Applied sciences (01.10.2022)
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Synthesis of 3,3-Diarylazetidines by Calcium(II)-Catalyzed Friedel–Crafts Reaction of Azetidinols with Unexpected Cbz Enhanced Reactivity
Denis, Camille, Dubois, Maryne A. J, Voisin-Chiret, Anne Sophie, Bureau, Ronan, Choi, Chulho, Mousseau, James J, Bull, James A
Published in Organic letters (04.01.2019)
Published in Organic letters (04.01.2019)
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Toward Understanding Mcl‑1 Promiscuous and Specific Binding Mode
Fogha, Jade, Marekha, Bogdan, De Giorgi, Marcella, Voisin-Chiret, Anne Sophie, Rault, Sylvain, Bureau, Ronan, Sopkova-de Oliveira Santos, Jana
Published in Journal of chemical information and modeling (27.11.2017)
Published in Journal of chemical information and modeling (27.11.2017)
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Sequential one pot double C-H heteroarylation of thiophene using bromopyridines to synthesize unsymmetrical 2,5-bipyridylthiophenes
Kieffer, Charline, Babin, Victor, Jouanne, Marie, Slimani, Ikram, Berhault, Yohann, Legay, Remi, Santos, Jana Sopkova-de Oliveira, Rault, Sylvain, Voisin-Chiret, Anne Sophie
Published in Tetrahedron (01.09.2017)
Published in Tetrahedron (01.09.2017)
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Structure-guided design of pyridoclax derivatives based on Noxa / Mcl-1 interaction mode
Hedir, Siham, De Giorgi, Marcella, Fogha, Jade, De Pascale, Martina, Weiswald, Louis-Bastien, Brotin, Emilie, Marekha, Bogdan, Denoyelle, Christophe, Denis, Camille, Suzanne, Peggy, Gautier, Fabien, Juin, Philippe, Ligat, Laetitia, Lopez, Frédéric, Carlier, Ludovic, Legay, Rémi, Bureau, Ronan, Rault, Sylvain, Poulain, Laurent, Oliveira Santos, Jana Sopková-de, Voisin-Chiret, Anne Sophie
Published in European journal of medicinal chemistry (05.11.2018)
Published in European journal of medicinal chemistry (05.11.2018)
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Catalytic Friedel‐Crafts Reactions on Saturated Heterocycles and Small Rings for sp3‐sp2 Coupling of Medicinally Relevant Fragments
Croft, Rosemary A., Dubois, Maryne A. J., Boddy, Alexander J., Denis, Camille, Lazaridou, Anna, Voisin‐Chiret, Anne Sophie, Bureau, Ronan, Choi, Chulho, Mousseau, James J., Bull, James A.
Published in European journal of organic chemistry (01.09.2019)
Published in European journal of organic chemistry (01.09.2019)
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