Access to 2,6-Disubstituted Piperidines: Control of the Diastereoselectivity, Scope, and Limitations. Applications to the Stereoselective Synthesis of (−)-Solenopsine A and Alkaloid (+)-241D
Abrunhosa-Thomas, Isabelle, Plas, Aurélie, Vogrig, Alexandre, Kandepedu, Nishanth, Chalard, Pierre, Troin, Yves
Published in Journal of organic chemistry (15.03.2013)
Published in Journal of organic chemistry (15.03.2013)
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Synthesis and evaluation of bidentate ligands designed to interact with PDZ domains
Boucherle, Benjamin, Vogrig, Alexandre, Deokar, Hemantkumar, Bouzidi, Naoual, Ripoche, Isabelle, Thomas, Isabelle, Marin, Philippe, Ducki, Sylvie
Published in Bioorganic & medicinal chemistry (15.07.2011)
Published in Bioorganic & medicinal chemistry (15.07.2011)
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Structure-Based Design of PDZ Ligands as Inhibitors of 5‑HT2A Receptor/PSD-95 PDZ1 Domain Interaction Possessing Anti-hyperalgesic Activity
Vogrig, Alexandre, Dorr, Liam, Bouzidi, Naoual, Boucherle, Benjamin, Wattiez, Anne-Sophie, Cassier, Elisabeth, Vallon, Gary, Ripoche, Isabelle, Abrunhosa-Thomas, Isabelle, Marin, Philippe, Nauton, Lionel, Thery, Vincent, Courteix, Christine, Lian, Lu-Yun, Ducki, Sylvie
Published in ACS chemical biology (18.10.2013)
Published in ACS chemical biology (18.10.2013)
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Identification of PDZ ligands by docking-based virtual screening for the development of novel analgesic agents
Bouzidi, Naoual, Deokar, Hemantkumar, Vogrig, Alexandre, Boucherle, Benjamin, Ripoche, Isabelle, Abrunhosa-Thomas, Isabelle, Dorr, Liam, Wattiez, Anne-Sophie, Lian, Lu-Yun, Marin, Philippe, Courteix, Christine, Ducki, Sylvie
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
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NMR evaluation of interactions between substituted-indole and PDZ1 domain of PSD-95
Vogrig, Alexandre, Boucherle, Benjamin, Deokar, Hemantkumar, Thomas, Isabelle, Ripoche, Isabelle, Lian, Lu-Yun, Ducki, Sylvie
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
Published in Bioorganic & medicinal chemistry letters (01.06.2011)
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Structure-Based Design of PDZ Ligands as Inhibitors of 5-HT 2A Receptor/PSD-95 PDZ1 Domain Interaction Possessing Anti-hyperalgesic Activity
Vogrig, Alexandre, Dorr, Liam, Bouzidi, Naoual, Boucherle, Benjamin, Wattiez, Anne-Sophie, Cassier, Elisabeth, Vallon, Gary, Ripoche, Isabelle, Abrunhosa-Thomas, Isabelle, Marin, Philippe, Nauton, Lionel, Thery, Vincent, Courteix, Christine, Lian, Lu-Yun, Ducki, Sylvie
Published in ACS chemical biology (18.10.2013)
Published in ACS chemical biology (18.10.2013)
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Structure-based design of PDZ ligands as inhibitors of 5-HT(2A) receptor/PSD-95 PDZ1 domain interaction possessing anti-hyperalgesic activity
Vogrig, Alexandre, Dorr, Liam, Bouzidi, Naoual, Boucherle, Benjamin, Wattiez, Anne-Sophie, Cassier, Elisabeth, Vallon, Gary, Ripoche, Isabelle, Abrunhosa-Thomas, Isabelle, Marin, Philippe, Nauton, Lionel, Thery, Vincent, Courteix, Christine, Lian, Lu-Yun, Ducki, Sylvie
Published in ACS chemical biology (18.10.2013)
Published in ACS chemical biology (18.10.2013)
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ChemInform Abstract: Access to 2,6-Disubstituted Piperidines: Control of the Diastereoselectivity, Scope, and Limitations. Applications to the Stereoselective Synthesis of (-)-Solenopsine A and Alkaloid (+)-241D
Abrunhosa-Thomas, Isabelle, Plas, Aurelie, Vogrig, Alexandre, Kandepedu, Nishanth, Chalard, Pierre, Troin, Yves
Published in ChemInform (23.07.2013)
Published in ChemInform (23.07.2013)
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