Molecular Field Extrema as Descriptors of Biological Activity: Definition and Validation
Cheeseright, Tim, Mackey, Mark, Rose, Sally, Vinter, Andy
Published in Journal of chemical information and modeling (01.03.2006)
Published in Journal of chemical information and modeling (01.03.2006)
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Journal Article
How computational chemistry develops: a tribute to Peter Goodford
Cruciani, Gabriele, Martin, Yvonne, Vinter, Andy, Lewis, Richard, Gago, Federico, Stouch, Terry R.
Published in Journal of computer-aided molecular design (01.08.2019)
Published in Journal of computer-aided molecular design (01.08.2019)
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Journal Article
Modulation of 11β-hydroxysteroid dehydrogenase type 1 activity by 1,5-substituted 1H-tetrazoles
Webster, Scott P., Binnie, Margaret, McConnell, Kirsty M.M., Sooy, Karen, Ward, Peter, Greaney, Michael F., Vinter, Andy, Pallin, T. David, Dyke, Hazel J., Gill, Matthew I.A., Warner, Ines, Seckl, Jonathan R., Walker, Brian R.
Published in Bioorganic & medicinal chemistry letters (01.06.2010)
Published in Bioorganic & medicinal chemistry letters (01.06.2010)
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An efficient asymmetric synthesis of the potent β-blocker ICI-118,551 allows the determination of enantiomer dependency on biological activityWe would like to dedicate this paper to the memory of Sir James Black who instigated this work as part of a larger βAR study at UCL.Electronic supplementary information (ESI) available: Full experimental details are provided. See DOI: 10.1039/c0cc00142b
Baker, James R, Hothersall, J. Daniel, Fitzmaurice, Richard J, Tucknott, Matthew, Vinter, Andy, Tinker, Andrew, Caddick, Stephen
Year of Publication 14.06.2010
Year of Publication 14.06.2010
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Journal Article
Discovery and biological evaluation of adamantyl amide 11β-HSD1 inhibitors
Webster, Scott P., Ward, Peter, Binnie, Margaret, Craigie, Eilidh, McConnell, Kirsty M.M., Sooy, Karen, Vinter, Andy, Seckl, Jonathan R., Walker, Brian R.
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
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Journal Article
An efficient asymmetric synthesis of the potent beta-blocker ICI-118,551 allows the determination of enantiomer dependency on biological activity
Baker, James R., Hothersall, J. Daniel, Fitzmaurice, Richard J., Tucknott, Matthew, Vinter, Andy, Tinker, Andrew, Caddick, Stephen
Published in Chemical communications (Cambridge, England) (14.06.2010)
Published in Chemical communications (Cambridge, England) (14.06.2010)
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Journal Article
Modulation of 11b-hydroxysteroid dehydrogenase type 1 activity by 1,5-substituted 1H-tetrazoles
Webster, Scott P, Binnie, Margaret, McConnell, Kirsty MM, Sooy, Karen, Ward, Peter, Greaney, Michael F, Vinter, Andy, Pallin, TDavid, Dyke, Hazel J, Gill, Matthew IA, Warner, Ines, Seckl, Jonathan R, Walker, Brian R
Published in Bioorganic & medicinal chemistry letters (01.06.2010)
Published in Bioorganic & medicinal chemistry letters (01.06.2010)
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Journal Article
Discovery and biological evaluation of adamantyl amide 11beta-HSD1 inhibitors
Webster, Scott P, Ward, Peter, Binnie, Margaret, Craigie, Eilidh, McConnell, Kirsty M M, Sooy, Karen, Vinter, Andy, Seckl, Jonathan R, Walker, Brian R
Published in Bioorganic & medicinal chemistry letters (15.05.2007)
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Published in Bioorganic & medicinal chemistry letters (15.05.2007)
Journal Article
Peptides to non-peptides: leads from structureless virtual screening
Cheeseright, Tim, Mackey, Mark, Vinter, Andy
Published in Drug Discovery Today: Biosilico (01.03.2004)
Published in Drug Discovery Today: Biosilico (01.03.2004)
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Book Review
Journal Article
Modulation of 11beta-hydroxysteroid dehydrogenase type 1 activity by 1,5-substituted 1H-tetrazoles
Webster, Scott P, Binnie, Margaret, McConnell, Kirsty M M, Sooy, Karen, Ward, Peter, Greaney, Michael F, Vinter, Andy, Pallin, T David, Dyke, Hazel J, Gill, Matthew I A, Warner, Ines, Seckl, Jonathan R, Walker, Brian R
Published in Bioorganic & medicinal chemistry letters (01.06.2010)
Published in Bioorganic & medicinal chemistry letters (01.06.2010)
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Journal Article
Editorial
Marshall, Garland R, Vinter, Andy
Published in Journal of computer-aided molecular design (01.01.1997)
Published in Journal of computer-aided molecular design (01.01.1997)
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ChemInform Abstract: An Efficient Asymmetric Synthesis of the Potent β-Blocker ICI-118,551 Allows the Determination of Enantiomer Dependency on Biological Activity
Baker, James R., Hothersall, J. Daniel, Fitzmaurice, Richard J., Tucknott, Matthew, Vinter, Andy, Tinker, Andrew, Caddick, Stephen
Published in ChemInform (26.10.2010)
Published in ChemInform (26.10.2010)
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