A possible improvement for structure-based drug design illustrated by the discovery of a Tat HIV-1 inhibitor
Montembault, Mickaël, Vo-Thanh, Giang, Deyine, Abdallah, Fargeas, Valérie, Villiéras, Monique, Adjou, Ané, Dubreuil, Didier, Esquieu, Didier, Grégoire, Catherine, Opi, Sandrine, Péloponèse, Jean-Marie, Campbell, Grant, Watkins, Jennifer, de Mareuil, Jean, Aubertin, Anne-Marie, Bailly, Christian, Loret, Erwann, Lebreton, Jacques
Published in Bioorganic & medicinal chemistry letters (22.03.2004)
Published in Bioorganic & medicinal chemistry letters (22.03.2004)
Get full text
Journal Article
Copper(I) mediated highly diastereoselective conjugate addition of Grignard reagents to functionalised cycloalkenols: a general and efficient route for the stereoselective synthesis of 5-and 6-membered ring trisubstituted cycloalkanols
Dambrin, Villieras, M, Janvier, P, Toupet, L, Amri, H, Lebreton, J, Villieras, J
Published in Tetrahedron (10.03.2001)
Published in Tetrahedron (10.03.2001)
Get full text
Journal Article
A new and efficient method for the isomerization of secondary functional allylic alcohols into their primary isomers
Beltaief, Hbaieb, S, Besbes, R, Amri, H, Villieras, M, Villieras, J
Published in Synthesis (Stuttgart) (01.12.1998)
Published in Synthesis (Stuttgart) (01.12.1998)
Get more information
Journal Article
Copper (I) mediated highly diastereoselective conjugate addition of Grignard reagents to functionalised 6-membered ring cycloalkenols. Synthesis of cyclohexanes derivatives substituted on three contiguous atoms
Dambrin, Valéry, Villiéras, Monique, Lebreton, Jacques, Toupet, Loïc, Amri, Hassen, Villiéras, Jean
Published in Tetrahedron letters (29.01.1999)
Published in Tetrahedron letters (29.01.1999)
Get full text
Journal Article
Porphyrin dyes for TiO2 sensitization
ODOBEL, Fabrice, BLART, Errol, LAGREE, Marie, VILLIERAS, Monique, BOUJTITA, Hamada, NABIL EL MURR, CARAMORI, Stefano, BIGNOZZI, Carlo Alberto
Published in Journal of materials chemistry (20.02.2003)
Published in Journal of materials chemistry (20.02.2003)
Get full text
Journal Article
Discovery of a Tat HIV‐1 Inhibitor through Computer‐Aided Drug Design
Esquieu, Didier, Péloponèse, Jean-Marie, Opi, Sandrine, Gregoire, Catherine, de Mareuil, Jean, Watkins, Jennifer, Campbell, Grant, Dunot, Jean-Pierre, Sturgis, James, Witvrouw, Myriam, Pannecouque, Christophe, de Clercq, Erik, Montembault, Mickaël, Giang, Vo-Thanh, Villiéras, Monique, Fargeas, Valérie, Lebreton, Jacques, Loret, Erwann P.
Published in Journal of spectroscopy (Hindawi) (01.01.2003)
Published in Journal of spectroscopy (Hindawi) (01.01.2003)
Get full text
Journal Article