Synthesis of a sugar-based thiosemicarbazone series and structure-activity relationship versus the parasite cysteine proteases rhodesain, cruzain, and Schistosoma mansoni cathepsin B1
Fonseca, Nayara Cristina, da Cruz, Luana Faria, da Silva Villela, Filipe, do Nascimento Pereira, Glaécia Aparecida, de Siqueira-Neto, Jair Lage, Kellar, Danielle, Suzuki, Brian M, Ray, Debalina, de Souza, Thiago Belarmino, Alves, Ricardo José, Sales Júnior, Policarpo Ademar, Romanha, Alvaro José, Murta, Silvane Maria Fonseca, McKerrow, James H, Caffrey, Conor R, de Oliveira, Renata Barbosa, Ferreira, Rafaela Salgado
Published in Antimicrobial agents and chemotherapy (01.05.2015)
Published in Antimicrobial agents and chemotherapy (01.05.2015)
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Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond
Van Voorhis, Wesley C, Adams, John H, Adelfio, Roberto, Alday, Aintzane, Alsibaee, Aishah, Alzualde, Ainhoa, Avery, Simon V, Avery, Vicky M, Baker, Mark, Ben Mamoun, Choukri, Bhatia, Sangeeta, Bowling, Tana, Bosch, Jürgen, Boucher, Lauren E, Boyom, Fabrice F, Brea, Jose, Brennan, Marian, Burton, Audrey, Caffrey, Conor R, Carter, Dee, Belen Cassera, Maria, Chih-Chien Cheng, Ken, Corbett, Yolanda, Cowan, Noemi, D'Alessandro, Sarah, Delves, Michael, DeRisi, Joseph L, Du, Alan Y, Fernández Robledo, José A, Florent, Isabelle, Fokou, Patrick V T, Galstian, Ani, Gamo, Francisco Javier, Gokool, Suzanne, Golub, Todd, Guiguemde, W Armand, Guy, R Kiplin, Horii, Takaaki, Horrocks, Paul, Hughes, Tyler B, Huston, Christopher, Igarashi, Ikuo, Ingram-Sieber, Katrin, Jadhav, Ajit, Jensen, Laran T, Keiser, Jennifer, Ketas, Thomas, Kumar, Vidya P, Kyle, Dennis E, Lafuente, Maria Jose, Landfear, Scott, Lee, Sukjun, Li, Fengwu, Little, David, Liu, Liqiong, Lubar, Aristea, Mansour, Nuha R, March, Sandra, McGowan, Sheena, Medina Vera, Iset, Mestres, Jordi, Morais Rodrigues da Costa, Francielly, Muriana, Arantza, Nare, Bakela, Papadatos, George, Parapini, Silvia, Patra, Kailash, Prats, Sarah, Poulsen, Sally-Ann, Quinn, Ronald J, Rice, Christopher A, Ruecker, Andrea, Salgado Ferreira, Rafaela, Samra, Jasmeet, Schlecht, Ulrich, Silva Villela, Filipe, Silvestrini, Francesco, Sinden, Robert, Soldati, Thierry, Spitzmüller, Andreas, Stamm, Serge Maximilian, Sullivan, David J, Sullivan, William, Swamidass, S Joshua, Taramelli, Donatella, Tripathi, Abhai K, Trofimov, Valentin, Udenze, Kenneth O, Vigil, Edgar, Voong Vinh, Phat, Vu, Hoan, Watanabe, Nao-Aki, Weatherby, Kate, White, Pamela M, Yokoyama, Naoaki, Abla, Nada, Laleu, Benoît, Leroy, Didier, Spangenberg, Thomas, Willis, Paul A
Published in PLoS pathogens (01.07.2016)
Published in PLoS pathogens (01.07.2016)
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Synthesis and structure–activity relationship study of a new series of antiparasitic aryloxyl thiosemicarbazones inhibiting Trypanosoma cruzi cruzain
Espíndola, José Wanderlan Pontes, Cardoso, Marcos Veríssimo de Oliveira, Filho, Gevanio Bezerra de Oliveira, Oliveira e Silva, Dayane Albuquerque, Moreira, Diogo Rodrigo Magalhaes, Bastos, Tanira Matutino, Simone, Carlos Alberto de, Soares, Milena Botelho Pereira, Villela, Filipe Silva, Ferreira, Rafaela Salgado, Castro, Maria Carolina Accioly Brelaz de, Pereira, Valéria Rego Alves, Murta, Silvane Maria Fonseca, Sales Junior, Policarpo Ademar, Romanha, Alvaro José, Leite, Ana Cristina Lima
Published in European journal of medicinal chemistry (28.08.2015)
Published in European journal of medicinal chemistry (28.08.2015)
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2-(phenylthio)ethylidene derivatives as anti-Trypanosoma cruzi compounds: Structural design, synthesis and antiparasitic activity
Cardoso, Marcos Veríssimo de Oliveira, Oliveira Filho, Gevanio Bezerra de, Siqueira, Lucianna Rabelo Pessoa de, Espíndola, José Wanderlan Pontes, Silva, Elany Barbosa da, Mendes, Andresa Pereira de Oliveira, Pereira, Valéria Rêgo Alves, Castro, Maria Carolina Accioly Brelaz de, Ferreira, Rafaela Salgado, Villela, Filipe Silva, Costa, Francielly Morais Rodrigues da, Meira, Cássio Santana, Moreira, Diogo Rodrigo Magalhães, Soares, Milena Botelho Pereira, Leite, Ana Cristina Lima
Published in European journal of medicinal chemistry (15.10.2019)
Published in European journal of medicinal chemistry (15.10.2019)
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Conformational restriction of aryl thiosemicarbazones produces potent and selective anti-Trypanosoma cruzi compounds which induce apoptotic parasite death
Magalhaes Moreira, Diogo Rodrigo, de Oliveira, Ana Daura Travassos, Teixeira de Moraes Gomes, Paulo André, de Simone, Carlos Alberto, Villela, Filipe Silva, Ferreira, Rafaela Salgado, da Silva, Aline Caroline, dos Santos, Thiago André Ramos, Brelaz de Castro, Maria Carolina Accioly, Pereira, Valéria Rego Alves, Leite, Ana Cristina Lima
Published in European journal of medicinal chemistry (21.03.2014)
Published in European journal of medicinal chemistry (21.03.2014)
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