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Gomez, Laurent, Massari, Mark Eben, Vickers, Troy, Freestone, Graeme, Vernier, William, Ly, Kiev, Xu, Rui, McCarrick, Margaret, Marrone, Tami, Metz, Markus, Yan, Yingzhou G, Yoder, Zachary W, Lemus, Robert, Broadbent, Nicola J, Barido, Richard, Warren, Noelle, Schmelzer, Kara, Neul, David, Lee, Dong, Andersen, Carsten B, Sebring, Kristen, Aertgeerts, Kathleen, Zhou, Xianbo, Tabatabaei, Ali, Peters, Marco, Breitenbucher, J. Guy
Published in Journal of medicinal chemistry (09.03.2017)
Published in Journal of medicinal chemistry (09.03.2017)
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Discovery of Highly Potent and Selective Pan-Aurora Kinase Inhibitors with Enhanced in Vivo Antitumor Therapeutic Index
Liu, Gang, Abraham, Sunny, Tran, Lan, Vickers, Troy D, Xu, Shimin, Hadd, Michael J, Quiambao, Sheena, Holladay, Mark W, Hua, Helen, Ford Pulido, Julia M, Gunawardane, Ruwanthi N, Davis, Mindy I, Eichelberger, Shawn R, Apuy, Julius L, Gitnick, Dana, Gardner, Michael F, James, Joyce, Breider, Mike A, Belli, Barbara, Armstrong, Robert C, Treiber, Daniel K
Published in Journal of medicinal chemistry (12.04.2012)
Published in Journal of medicinal chemistry (12.04.2012)
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Studies on the structure–activity relationship of bicifadine analogs as monoamine transporter inhibitors
Zhang, Mingzhu, Jovic, Florence, Vickers, Troy, Dyck, Brian, Tamiya, Junko, Grey, Jonathan, Tran, Joe A., Fleck, Beth A., Pick, Rebecca, Foster, Alan C., Chen, Chen
Published in Bioorganic & medicinal chemistry (01.07.2008)
Published in Bioorganic & medicinal chemistry (01.07.2008)
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Identification of 1S,2R-milnacipran analogs as potent norepinephrine and serotonin transporter inhibitors
TAMIYA, Junko, DYCK, Brian, FOSTER, Alan C, CHEN CHEN, MINGZHU ZHANG, PHAN, Kasey, FLECK, Beth A, APARICIO, Anna, JOVIC, Florence, TRAN, Joe A, VICKERS, Troy, GREY, Jonathan
Published in Bioorganic & medicinal chemistry (01.06.2008)
Published in Bioorganic & medicinal chemistry (01.06.2008)
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Thienopyrimidinone bis-aminopyrrolidine ureas as potent melanin-concentrating hormone receptor-1 (MCH-R1) antagonists
Zhang, Mingzhu, Tamiya, Junko, Nguyen, Linh, Rowbottom, Martin W., Dyck, Brian, Vickers, Troy D., Grey, Jonathan, Schwarz, David A., Heise, Christopher E., Haelewyn, Jason, Mistry, Monica S., Goodfellow, Val S.
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
Published in Bioorganic & medicinal chemistry letters (01.05.2007)
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Studies on the SAR and pharmacophore of milnacipran derivatives as monoamine transporter inhibitors
Chen, Chen, Dyck, Brian, Fleck, Beth A., Foster, Alan C., Grey, Jonathan, Jovic, Florence, Mesleh, Michael, Phan, Kasey, Tamiya, Junko, Vickers, Troy, Zhang, Mingzhu
Published in Bioorganic & medicinal chemistry (15.02.2008)
Published in Bioorganic & medicinal chemistry (15.02.2008)
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Studies on a series of milnacipran analogs containing a heteroaromatic group as potent norepinephrine and serotonin transporter inhibitors
Vickers, Troy, Dyck, Brian, Tamiya, Junko, Zhang, Mingzhu, Jovic, Florence, Grey, Jonathan, Fleck, Beth A., Aparicio, Anna, Johns, Michael, Jin, Liping, Tang, Hui, Foster, Alan C., Chen, Chen
Published in Bioorganic & medicinal chemistry (01.06.2008)
Published in Bioorganic & medicinal chemistry (01.06.2008)
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Synthesis and structure–activity relationships of spirohydantoin-derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1)
Rowbottom, Martin W., Vickers, Troy D., Tamiya, Junko, Zhang, Mingzhu, Dyck, Brian, Grey, Jonathan, Schwarz, David, Heise, Christopher E., Hedrick, Michael, Wen, Jenny, Tang, Hui, Wang, Hua, Fisher, Andrew, Aparicio, Anna, Saunders, John, Goodfellow, Val S.
Published in Bioorganic & medicinal chemistry letters (15.04.2007)
Published in Bioorganic & medicinal chemistry letters (15.04.2007)
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Synthesis and structure–activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 2
Hudson, Sarah, Kiankarimi, Mehrak, Rowbottom, Martin W., Vickers, Troy D., Wu, Dongpei, Pontillo, Joseph, Ching, Brett, Dwight, Wesley, Goodfellow, Val S., Schwarz, David, Heise, Christopher E., Madan, Ajay, Wen, Jenny, Ban, William, Wang, Hua, Wade, Warren S.
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
Published in Bioorganic & medicinal chemistry letters (15.09.2006)
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Bis(aminopyrrolidine)-derived ureas (APUs) as potent MCH1 receptor antagonists
Grey, Jonathan, Dyck, Brian, Rowbottom, Martin W, Tamiya, Junko, Vickers, Troy D, Zhang, Mingzhu, Zhao, Liren, Heise, Christopher E, Schwarz, David, Saunders, John, Goodfellow, Val S
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
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Journal Article
Synthesis and structure–activity relationships of retro bis-aminopyrrolidine urea (rAPU) derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1). Part 1
Rowbottom, Martin W., Vickers, Troy D., Dyck, Brian, Grey, Jonathan, Tamiya, Junko, Zhang, Mingzhu, Kiankarimi, Mehrak, Wu, Dongpei, Dwight, Wesley, Wade, Warren S., Schwarz, David, Heise, Christopher E., Madan, Ajay, Fisher, Andrew, Petroski, Robert, Goodfellow, Val S.
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
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Synthesis and structure–activity relationships of biarylcarboxamide bis-aminopyrrolidine urea derived small-molecule antagonists of the melanin-concentrating hormone receptor-1 (MCH-R1)
Rowbottom, Martin W., Vickers, Troy D., Dyck, Brian, Tamiya, Junko, Zhang, Mingzhu, Zhao, Liren, Grey, Jonathan, Provencal, David, Schwarz, David, Heise, Christopher E., Mistry, Monica, Fisher, Andrew, Dong, Teresa, Hu, Tao, Saunders, John, Goodfellow, Val S.
Published in Bioorganic & medicinal chemistry letters (15.07.2005)
Published in Bioorganic & medicinal chemistry letters (15.07.2005)
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HADIDA RUAH SARA SABINA, PIERRE FABRICE, MCCARTNEY JASON, DWIGHT TIMOTHY A, PARASELLI PRASUNA, KHATUYA HARIPADA, UY JOHNNY, FANNING LEV TYLER DEWEY, SILINA ALINA, VICKERS TROY, ARUMUGAM VIJAYALAKSMI, GROOTENHUIS PETER, ANDERSON COREY DON, COON TIMOTHY RICHARD, FRIEMAN BRYAN A, GULEVICH ANTON V, ZHOU JINGLAN, VALDEZ LINO, ABRAHAM SUNNY, MELILLO VITO, TRAN JOE A, CHAU JACLYN, CLEVELAND THOMAS, ABELA ALEXANDER RUSSELL, MILLER MARK THOMAS, CLEMENS JEREMY, KRENITSKY PAUL, ISHIHARA YOSHIHIRO
Year of Publication 17.07.2023
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Novel series of pyrrolotriazine analogs as highly potent pan-Aurora kinase inhibitors
Abraham, Sunny, Hadd, Michael J., Tran, Lan, Vickers, Troy, Sindac, Janice, Milanov, Zdravko V., Holladay, Mark W., Bhagwat, Shripad S., Hua, Helen, Ford Pulido, Julia M., Cramer, Merryl D., Gitnick, Dana, James, Joyce, Dao, Alan, Belli, Barbara, Armstrong, Robert C., Treiber, Daniel K., Liu, Gang
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
Published in Bioorganic & medicinal chemistry letters (15.09.2011)
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A Thienopyridazinone-Based Melanin-Concentrating Hormone Receptor 1 Antagonist with Potent in Vivo Anorectic Properties
Dyck, Brian, Markison, Stacy, Zhao, Liren, Tamiya, Junko, Grey, Jonathan, Rowbottom, Martin W, Zhang, Mingzhu, Vickers, Troy, Sorensen, Katie, Norton, Christi, Wen, Jenny, Heise, Christopher E, Saunders, John, Conlon, Paul, Madan, Ajay, Schwarz, David, Goodfellow, Val S
Published in Journal of medicinal chemistry (29.06.2006)
Published in Journal of medicinal chemistry (29.06.2006)
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SUBSTITUTED PYRIDINE AND PYRAZINE COMPOUNDS AS PDE4 INHIBITORS
ZAPF JAMES, BREITENBUCHER JAMES, VICKERS TROY, BOLLU VENKATAIAH, LINDSTROM ANDREW, KAPLAN ALAN, LEMUS ROBERT, WILSON MARK E, WEINHOUSE MICHAEL I
Year of Publication 18.11.2015
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Year of Publication 18.11.2015
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SUBSTITUTED THIOPHENE- AND FURAN-FUSED AZOLOPYRIMIDINE-5-(6H)-ONE COMPOUNDS
BREITENBUCHER JAMES, PETERS MARCO, VICKERS TROY, DYCK BRIAN, HUDSON ANDREW RICHARD, GOMEZ LAURENT, BRANSTETTER BRYAN, MARRONE TAMI JO
Year of Publication 08.06.2015
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Year of Publication 08.06.2015
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Characterization of Thien-2-yl 1S,2R-Milnacipran Analogues as Potent Norepinephrine/Serotonin Transporter Inhibitors for the Treatment of Neuropathic Pain
Dyck, Brian, Tamiya, Junko, Jovic, Florence, Pick, Rebecca R, Bradbury, Margaret J, O’Brien, Julie, Wen, Jenny, Johns, Michael, Madan, Ajay, Fleck, Beth A, Foster, Alan C, Li, Binfeng, Zhang, Mingzhu, Tran, Joe A, Vickers, Troy, Grey, Jonathan, Saunders, John, Chen, Chen
Published in Journal of medicinal chemistry (27.11.2008)
Published in Journal of medicinal chemistry (27.11.2008)
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