Inhibition of Acetyl-CoA Carboxylase 1 (ACC1) and 2 (ACC2) Reduces Proliferation and De Novo Lipogenesis of EGFRvIII Human Glioblastoma Cells
Jones, Jessica E C, Esler, William P, Patel, Rushi, Lanba, Adhiraj, Vera, Nicholas B, Pfefferkorn, Jeffrey A, Vernochet, Cecile
Published in PloS one (01.01.2017)
Published in PloS one (01.01.2017)
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Adipocyte OGT governs diet-induced hyperphagia and obesity
Li, Min-Dian, Vera, Nicholas B, Yang, Yunfan, Zhang, Bichen, Ni, Weiming, Ziso-Qejvanaj, Enida, Ding, Sheng, Zhang, Kaisi, Yin, Ruonan, Wang, Simeng, Zhou, Xu, Fang, Ethan X, Xu, Tian, Erion, Derek M, Yang, Xiaoyong
Published in Nature communications (30.11.2018)
Published in Nature communications (30.11.2018)
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Pharmacologic inhibition of ketohexokinase prevents fructose-induced metabolic dysfunction
Gutierrez, Jemy A., Liu, Wei, Perez, Sylvie, Xing, Gang, Sonnenberg, Gabriele, Kou, Kou, Blatnik, Matt, Allen, Richard, Weng, Yan, Vera, Nicholas B., Chidsey, Kristin, Bergman, Arthur, Somayaji, Veena, Crowley, Collin, Clasquin, Michelle F., Nigam, Anu, Fulham, Melissa A., Erion, Derek M., Ross, Trenton T., Esler, William P., Magee, Thomas V., Pfefferkorn, Jeffrey A., Bence, Kendra K., Birnbaum, Morris J., Tesz, Gregory J.
Published in Molecular metabolism (Germany) (01.06.2021)
Published in Molecular metabolism (Germany) (01.06.2021)
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The hepatoselective glucokinase activator PF-04991532 ameliorates hyperglycemia without causing hepatic steatosis in diabetic rats
Erion, Derek M, Lapworth, Amanda, Amor, Paul A, Bai, Guoyun, Vera, Nicholas B, Clark, Ronald W, Yan, Qingyun, Zhu, Yimin, Ross, Trenton T, Purkal, Julie, Gorgoglione, Matthew, Zhang, Guodong, Bonato, Vinicius, Baker, Levenia, Barucci, Nicole, D'Aquila, Theresa, Robertson, Alan, Aiello, Robert J, Yan, Jiangli, Trimmer, Jeff, Rolph, Timothy P, Pfefferkorn, Jeffrey A
Published in PloS one (23.05.2014)
Published in PloS one (23.05.2014)
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Growth differentiation factor 15 neutralization does not impact anorexia or survival in lipopolysaccharide-induced inflammation
Breen, Danna M., Jagarlapudi, Srinath, Patel, Anita, Zou, Chang, Joaquim, Stephanie, Li, Xiangping, Kang, Liya, Pang, Jincheng, Hales, Katherine, Ziso-Qejvanaj, Enida, Vera, Nicholas B., Bennett, Donald, He, Tao, Lambert, Matthew, Kelleher, Kerry, Wu, Zhidan, Zhang, Bei B., Lin, Laura, Seeley, Randy J., Bezy, Olivier
Published in iScience (25.06.2021)
Published in iScience (25.06.2021)
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Human sebum requires de novo lipogenesis, which is increased in acne vulgaris and suppressed by acetyl-CoA carboxylase inhibition
Esler, William P, Tesz, Gregory J, Hellerstein, Marc K, Beysen, Carine, Sivamani, Raja, Turner, Scott M, Watkins, Steven M, Amor, Paul A, Carvajal-Gonzalez, Santos, Geoly, Frank J, Biddle, Kathleen E, Purkal, Julie J, Fitch, Mark, Buckeridge, Clare, Silvia, Annette M, Griffith, David A, Gorgoglione, Matthew, Hassoun, Lauren, Bosanac, Suzana S, Vera, Nicholas B, Rolph, Timothy P, Pfefferkorn, Jeffrey A, Sonnenberg, Gabriele E
Published in Science translational medicine (15.05.2019)
Published in Science translational medicine (15.05.2019)
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Characterization of a Novel Intestinal Glycerol-3-phosphate Acyltransferase Pathway and Its Role in Lipid Homeostasis
Khatun, Irani, Clark, Ronald W., Vera, Nicholas B., Kou, Kou, Erion, Derek M., Coskran, Timothy, Bobrowski, Walter F., Okerberg, Carlin, Goodwin, Bryan
Published in The Journal of biological chemistry (05.02.2016)
Published in The Journal of biological chemistry (05.02.2016)
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Adipocyte JAK2 Regulates Hepatic Insulin Sensitivity Independently of Body Composition, Liver Lipid Content, and Hepatic Insulin Signaling
Corbit, Kevin C, Camporez, João Paulo G, Edmunds, Lia R, Tran, Jennifer L, Vera, Nicholas B, Erion, Derek M, Deo, Rahul C, Perry, Rachel J, Shulman, Gerald I, Jurczak, Michael J, Weiss, Ethan J
Published in Diabetes (New York, N.Y.) (01.02.2018)
Published in Diabetes (New York, N.Y.) (01.02.2018)
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Quantitation of Urinary Acylcarnitines by DMS-MS/MS Uncovers the Effects of Total Body Irradiation in Cancer Patients
Vera, Nicholas B, Coy, Stephen L, Laiakis, Evagelia C, Fornace, Albert J, Clasquin, Michelle, Barker, Christopher A, Pfefferkorn, Jeffrey A, Vouros, Paul
Published in Journal of the American Society for Mass Spectrometry (04.03.2020)
Published in Journal of the American Society for Mass Spectrometry (04.03.2020)
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Discovery and characterization of novel inhibitors of the sodium-coupled citrate transporter (NaCT or SLC13A5)
Huard, Kim, Brown, Janice, Jones, Jessica C, Cabral, Shawn, Futatsugi, Kentaro, Gorgoglione, Matthew, Lanba, Adhiraj, Vera, Nicholas B, Zhu, Yimin, Yan, Qingyun, Zhou, Yingjiang, Vernochet, Cecile, Riccardi, Keith, Wolford, Angela, Pirman, David, Niosi, Mark, Aspnes, Gary, Herr, Michael, Genung, Nathan E, Magee, Thomas V, Uccello, Daniel P, Loria, Paula, Di, Li, Gosset, James R, Hepworth, David, Rolph, Timothy, Pfefferkorn, Jeffrey A, Erion, Derek M
Published in Scientific reports (01.12.2015)
Published in Scientific reports (01.12.2015)
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Differential mobility spectrometry (DMS) reveals the elevation of urinary acetylcarnitine in non‐human primates (NHPs) exposed to radiation
Vera, Nicholas B., Chen, Zhidan, Pannkuk, Evan, Laiakis, Evagelia C., Fornace, Albert J., Erion, Derek M., Coy, Stephen L., Pfefferkorn, Jeffrey A., Vouros, Paul
Published in Journal of mass spectrometry. (01.07.2018)
Published in Journal of mass spectrometry. (01.07.2018)
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Optimization of a Dicarboxylic Series for in Vivo Inhibition of Citrate Transport by the Solute Carrier 13 (SLC13) Family
Huard, Kim, Gosset, James R, Montgomery, Justin I, Gilbert, Adam, Hayward, Matthew M, Magee, Thomas V, Cabral, Shawn, Uccello, Daniel P, Bahnck, Kevin, Brown, Janice, Purkal, Julie, Gorgoglione, Matthew, Lanba, Adhiraj, Futatsugi, Kentaro, Herr, Michael, Genung, Nathan E, Aspnes, Gary, Polivkova, Jana, Garcia-Irizarry, Carmen N, Li, Qifang, Canterbury, Daniel, Niosi, Mark, Vera, Nicholas B, Li, Zhenhong, Khunte, Bhagyashree, Siderewicz, Jaclyn, Rolph, Timothy, Erion, Derek M
Published in Journal of medicinal chemistry (11.02.2016)
Published in Journal of medicinal chemistry (11.02.2016)
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De novo lipogenesis is essential for platelet production in humans
Kelly, Kenneth L, Reagan, William J, Sonnenberg, Gabriele E, Clasquin, Michelle, Hales, Katherine, Asano, Shoh, Amor, Paul A, Carvajal-Gonzalez, Santos, Shirai, Norimitsu, Matthews, Marcy D, Li, Kelvin W, Hellerstein, Marc K, Vera, Nicholas B, Ross, Trenton T, Cappon, Gregg, Bergman, Arthur, Buckeridge, Clare, Sun, Zhongyuan, Qejvanaj, Enida Ziso, Schmahai, Theodore, Beebe, David, Pfefferkorn, Jeffrey A, Esler, William P
Published in Nature metabolism (01.10.2020)
Published in Nature metabolism (01.10.2020)
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Discovery of a Selective Covalent Inhibitor of Lysophospholipase-like 1 (LYPLAL1) as a Tool to Evaluate the Role of this Serine Hydrolase in Metabolism
Ahn, Kay, Boehm, Markus, Brown, Matthew F, Calloway, Jessica, Che, Ye, Chen, Jinshan, Fennell, Kimberly F, Geoghegan, Kieran F, Gilbert, Adam M, Gutierrez, Jemy A, Kalgutkar, Amit S, Lanba, Adhiraj, Limberakis, Chris, Magee, Thomas V, O’Doherty, Inish, Oliver, Robert, Pabst, Brandon, Pandit, Jayvardhan, Parris, Kevin, Pfefferkorn, Jeffrey A, Rolph, Timothy P, Patel, Rushi, Schuff, Brandon, Shanmugasundaram, Veerabahu, Starr, Jeremy T, Varghese, Alison H, Vera, Nicholas B, Vernochet, Cecile, Yan, Jiangli
Published in ACS chemical biology (16.09.2016)
Published in ACS chemical biology (16.09.2016)
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Adipocyte JAK2 mediates spontaneous metabolic liver disease and hepatocellular carcinoma
Corbit, Kevin C, Wilson, Camella G, Lowe, Dylan, Tran, Jennifer L, Vera, Nicholas B, Clasquin, Michelle, Mattis, Aras N, Weiss, Ethan J
Published in JCI insight (05.09.2019)
Published in JCI insight (05.09.2019)
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Inhibition of Acetyl-CoA Carboxylase 1 Reduces Proliferation and De Novo Lipogenesis of EGFRvIII Human Glioblastoma Cells
Jones, Jessica E. C, Esler, William P, Patel, Rushi, Lanba, Adhiraj, Vera, Nicholas B, Pfefferkorn, Jeffrey A, Vernochet, Cecile
Published in PloS one (12.01.2017)
Published in PloS one (12.01.2017)
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Journal Article
Inhibition of Acetyl-CoA Carboxylase 1
Jones, Jessica E. C, Esler, William P, Patel, Rushi, Lanba, Adhiraj, Vera, Nicholas B, Pfefferkorn, Jeffrey A, Vernochet, Cecile
Published in PloS one (12.01.2017)
Published in PloS one (12.01.2017)
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