GPCR activation mechanisms across classes and macro/microscales
Hauser, Alexander S, Kooistra, Albert J, Munk, Christian, Heydenreich, Franziska M, Veprintsev, Dmitry B, Bouvier, Michel, Babu, M Madan, Gloriam, David E
Published in Nature structural & molecular biology (01.11.2021)
Published in Nature structural & molecular biology (01.11.2021)
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Journal Article
Diverse activation pathways in class A GPCRs converge near the G-protein-coupling region
Venkatakrishnan, A J, Deupi, Xavier, Lebon, Guillaume, Heydenreich, Franziska M, Flock, Tilman, Miljus, Tamara, Balaji, Santhanam, Bouvier, Michel, Veprintsev, Dmitry B, Tate, Christopher G, Schertler, Gebhard F X, Babu, M Madan
Published in Nature (London) (25.08.2016)
Published in Nature (London) (25.08.2016)
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Journal Article
Hsp90-Tau Complex Reveals Molecular Basis for Specificity in Chaperone Action
Karagöz, G. Elif, Duarte, Afonso M.S., Akoury, Elias, Ippel, Hans, Biernat, Jacek, Morán Luengo, Tania, Radli, Martina, Didenko, Tatiana, Nordhues, Bryce A., Veprintsev, Dmitry B., Dickey, Chad A., Mandelkow, Eckhard, Zweckstetter, Markus, Boelens, Rolf, Madl, Tobias, Rüdiger, Stefan G.D.
Published in Cell (27.02.2014)
Published in Cell (27.02.2014)
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A new inhibitor of the β-arrestin/AP2 endocytic complex reveals interplay between GPCR internalization and signalling
Beautrait, Alexandre, Paradis, Justine S, Zimmerman, Brandon, Giubilaro, Jenna, Nikolajev, Ljiljana, Armando, Sylvain, Kobayashi, Hiroyuki, Yamani, Lama, Namkung, Yoon, Heydenreich, Franziska M, Khoury, Etienne, Audet, Martin, Roux, Philippe P, Veprintsev, Dmitry B, Laporte, Stéphane A, Bouvier, Michel
Published in Nature communications (18.04.2017)
Published in Nature communications (18.04.2017)
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Journal Article
Distinct G protein-coupled receptor phosphorylation motifs modulate arrestin affinity and activation and global conformation
Mayer, Daniel, Damberger, Fred F, Samarasimhareddy, Mamidi, Feldmueller, Miki, Vuckovic, Ziva, Flock, Tilman, Bauer, Brian, Mutt, Eshita, Zosel, Franziska, Allain, Frédéric H T, Standfuss, Jörg, Schertler, Gebhard F X, Deupi, Xavier, Sommer, Martha E, Hurevich, Mattan, Friedler, Assaf, Veprintsev, Dmitry B
Published in Nature communications (19.03.2019)
Published in Nature communications (19.03.2019)
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Journal Article
Targeted rescue of a destabilized mutant of p53 by an in silico screened drug
Boeckler, Frank M, Joerger, Andreas C, Jaggi, Gaurav, Rutherford, Trevor J, Veprintsev, Dmitry B, Fersht, Alan R
Published in Proceedings of the National Academy of Sciences - PNAS (29.07.2008)
Published in Proceedings of the National Academy of Sciences - PNAS (29.07.2008)
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Journal Article
High-throughput mutagenesis using a two-fragment PCR approach
Heydenreich, Franziska M, Miljuš, Tamara, Jaussi, Rolf, Benoit, Roger, Milić, Dalibor, Veprintsev, Dmitry B
Published in Scientific reports (28.07.2017)
Published in Scientific reports (28.07.2017)
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Journal Article
Molecular recognition of an odorant by the murine trace amine-associated receptor TAAR7f
Gusach, Anastasiia, Lee, Yang, Khoshgrudi, Armin Nikpour, Mukhaleva, Elizaveta, Ma, Ning, Koers, Eline J, Chen, Qingchao, Edwards, Patricia C, Huang, Fanglu, Kim, Jonathan, Mancia, Filippo, Veprintsev, Dmitry B, Vaidehi, Nagarajan, Weyand, Simone N, Tate, Christopher G
Published in Nature communications (30.08.2024)
Published in Nature communications (30.08.2024)
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Journal Article
Modulation of the Oligomerization State of p53 by Differential Binding of Proteins of the S100 Family to p53 Monomers and Tetramers
van Dieck, Jan, Fernandez-Fernandez, Maria R., Veprintsev, Dmitry B., Fersht, Alan R.
Published in The Journal of biological chemistry (15.05.2009)
Published in The Journal of biological chemistry (15.05.2009)
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Journal Article
Stabilization of G protein-coupled receptors by point mutations
Heydenreich, Franziska M, Vuckovic, Ziva, Matkovic, Milos, Veprintsev, Dmitry B
Published in Frontiers in pharmacology (20.04.2015)
Published in Frontiers in pharmacology (20.04.2015)
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Journal Article
Development of a membrane-based Gi-CASE biosensor assay for profiling compounds at cannabinoid receptors
Scott-Dennis, Morgan, Rafani, Fikri A., Yi, Yicheng, Perera, Themiya, Harwood, Clare R., Guba, Wolfgang, Rufer, Arne C., Grether, Uwe, Veprintsev, Dmitry B., Sykes, David A.
Published in Frontiers in pharmacology (11.08.2023)
Published in Frontiers in pharmacology (11.08.2023)
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Journal Article
Acetylation of lysine 120 of p53 endows DNA-binding specificity at effective physiological salt concentration
Arbely, Eyal, Natan, Eviatar, Brandt, Tobias, Allen, Mark D., Veprintsev, Dmitry B., Robinson, Carol V., Chin, Jason W., Joerger, Andreas C., Fersht, Alan R.
Published in Proceedings of the National Academy of Sciences - PNAS (17.05.2011)
Published in Proceedings of the National Academy of Sciences - PNAS (17.05.2011)
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Journal Article
Structural Evolution of p53, p63, and p73: Implication for Heterotetramer Formation
Joerger, Andreas C., Rajagopalan, Sridharan, Natan, Eviatar, Veprintsev, Dmitry B., Robinson, Carol V., Fersht, Alan R.
Published in Proceedings of the National Academy of Sciences - PNAS (20.10.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (20.10.2009)
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Journal Article
Lithocholic acid is an endogenous inhibitor of MDM4 and MDM2
Vogel, Simon M, Bauer, Matthias R, Joerger, Andreas C, Wilcken, Rainer, Brandt, Tobias, Veprintsev, Dmitry B, Rutherford, Trevor J, Fersht, Alan R, Boeckler, Frank M
Published in Proceedings of the National Academy of Sciences - PNAS (16.10.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (16.10.2012)
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Journal Article
Cooperative Binding of Tetrameric p53 to DNA
Weinberg, Richard L., Veprintsev, Dmitry B., Fersht, Alan R.
Published in Journal of molecular biology (27.08.2004)
Published in Journal of molecular biology (27.08.2004)
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