Structures of aminoarabinose transferase ArnT suggest a molecular basis for lipid A glycosylation
Petrou, Vasileios I., Herrera, Carmen M., Schultz, Kathryn M., Clarke, Oliver B., Vendome, Jérémie, Tomasek, David, Banerjee, Surajit, Rajashankar, Kanagalaghatta R., Dufrisne, Meagan Belcher, Kloss, Brian, Kloppmann, Edda, Rost, Burkhard, Klug, Candice S., Trent, M. Stephen, Shapiro, Lawrence, Mancia, Filippo
Published in Science (American Association for the Advancement of Science) (05.02.2016)
Published in Science (American Association for the Advancement of Science) (05.02.2016)
Get full text
Journal Article
Molecular Modeling of Wild-Type and D816V c-Kit Inhibition Based on ATP-Competitive Binding of Ellipticine Derivatives to Tyrosine Kinases
Vendôme, Jérémie, Letard, Sébastien, Martin, Frédéric, Svinarchuk, Fedor, Dubreuil, Patrice, Auclair, Christian, Le Bret, Marc
Published in Journal of medicinal chemistry (06.10.2005)
Published in Journal of medicinal chemistry (06.10.2005)
Get full text
Journal Article
The Extracellular Architecture of Adherens Junctions Revealed by Crystal Structures of Type I Cadherins
Harrison, Oliver J., Jin, Xiangshu, Hong, Soonjin, Bahna, Fabiana, Ahlsen, Goran, Brasch, Julia, Wu, Yinghao, Vendome, Jeremie, Felsovalyi, Klara, Hampton, Cheri M., Troyanovsky, Regina B., Ben-Shaul, Avinoam, Frank, Joachim, Troyanovsky, Sergey M., Shapiro, Lawrence, Honig, Barry
Published in Structure (London) (09.02.2011)
Published in Structure (London) (09.02.2011)
Get full text
Journal Article
Nectin ectodomain structures reveal a canonical adhesive interface
Harrison, Oliver J, Vendome, Jeremie, Brasch, Julia, Jin, Xiangshu, Hong, Soonjin, Katsamba, Phinikoula S, Ahlsen, Goran, Troyanovsky, Regina B, Troyanovsky, Sergey M, Honig, Barry, Shapiro, Lawrence
Published in Nature structural & molecular biology (01.09.2012)
Published in Nature structural & molecular biology (01.09.2012)
Get full text
Journal Article
Structural and energetic determinants of adhesive binding specificity in type I cadherins
Vendome, Jeremie, Felsovalyi, Klara, Song, Hang, Yang, Zhongyu, Jin, Xiangshu, Brasch, Julia, Harrison, Oliver J., Ahlsen, Goran, Bahna, Fabiana, Kaczynska, Anna, Katsamba, Phinikoula S., Edmond, Darwin, Hubbell, Wayne L., Shapiro, Lawrence, Honig, Barry
Published in Proceedings of the National Academy of Sciences - PNAS (07.10.2014)
Published in Proceedings of the National Academy of Sciences - PNAS (07.10.2014)
Get full text
Journal Article
Evidence for the early emergence of piperaquine-resistant Plasmodium falciparum malaria and modeling strategies to mitigate resistance
Small-Saunders, Jennifer L, Hagenah, Laura M, Wicht, Kathryn J, Dhingra, Satish K, Deni, Ioanna, Kim, Jonathan, Vendome, Jeremie, Gil-Iturbe, Eva, Roepe, Paul D, Mehta, Monica, Mancia, Filippo, Quick, Matthias, Eppstein, Margaret J, Fidock, David A
Published in PLoS pathogens (07.02.2022)
Published in PLoS pathogens (07.02.2022)
Get full text
Journal Article
The mechanism of patellamide macrocyclization revealed by the characterization of the PatG macrocyclase domain
Koehnke, Jesko, Bent, Andrew, Houssen, Wael E, Zollman, David, Morawitz, Falk, Shirran, Sally, Vendome, Jeremie, Nneoyiegbe, Ada F, Trembleau, Laurent, Botting, Catherine H, Smith, Margaret C M, Jaspars, Marcel, Naismith, James H
Published in Nature structural & molecular biology (01.08.2012)
Published in Nature structural & molecular biology (01.08.2012)
Get full text
Journal Article
Structure and Substrate Recognition of the Bottromycin Maturation Enzyme BotP
Mann, Greg, Huo, Liujie, Adam, Sebastian, Nardone, Brunello, Vendome, Jeremie, Westwood, Nicholas James, Müller, Rolf, Koehnke, Jesko
Published in Chembiochem : a European journal of chemical biology (02.12.2016)
Published in Chembiochem : a European journal of chemical biology (02.12.2016)
Get full text
Journal Article
Loop L5 Acts as a Conformational Latch in the Mitotic Kinesin Eg5
Behnke-Parks, William M., Vendome, Jeremie, Honig, Barry, Maliga, Zoltan, Moores, Carolyn, Rosenfeld, Steven S.
Published in The Journal of biological chemistry (18.02.2011)
Published in The Journal of biological chemistry (18.02.2011)
Get full text
Journal Article
Shape-Based Virtual Screening of a Billion-Compound Library Identifies Mycobacterial Lipoamide Dehydrogenase Inhibitors
Michino, Mayako, Beautrait, Alexandre, Boyles, Nicholas A., Nadupalli, Aparna, Dementiev, Alexey, Sun, Shan, Ginn, John, Baxt, Leigh, Suto, Robert, Bryk, Ruslana, Jerome, Steven V., Huggins, David J., Vendome, Jeremie
Published in ACS bio & med chem au (20.12.2023)
Published in ACS bio & med chem au (20.12.2023)
Get full text
Journal Article
The Discovery of New Cyanobactins from Cyanothece PCC 7425 Defines a New Signature for Processing of Patellamides
Houssen, Wael E., Koehnke, Jesko, Zollman, David, Vendome, Jeremie, Raab, Andrea, Smith, Margaret C. M., Naismith, James H., Jaspars, Marcel
Published in Chembiochem : a European journal of chemical biology (21.12.2012)
Published in Chembiochem : a European journal of chemical biology (21.12.2012)
Get full text
Journal Article
Crystal structures of Drosophila N-cadherin ectodomain regions reveal a widely used class of Ca2+-free interdomain linkers
Jin, Xiangshu, Walker, Melissa A, Felsövályi, Klára, Vendome, Jeremie, Bahna, Fabiana, Mannepalli, Seetha, Cosmanescu, Filip, Ahlsen, Goran, Honig, Barry, Shapiro, Lawrence
Published in Proceedings of the National Academy of Sciences - PNAS (17.01.2012)
Published in Proceedings of the National Academy of Sciences - PNAS (17.01.2012)
Get full text
Journal Article
Characterization of Biochemical Properties of Bacillus subtilis RecQ Helicase
Qin, Wei, Liu, Na-Nv, Wang, Lijun, Zhou, Min, Ren, Hua, Bugnard, Elisabeth, Liu, Jie-Lin, Zhang, Lin-Hu, Vendôme, Jeremie, Hu, Jin-Shan, Xi, Xu Guang
Published in Journal of bacteriology (01.12.2014)
Published in Journal of bacteriology (01.12.2014)
Get full text
Journal Article
Transforming binding affinities from three dimensions to two with application to cadherin clustering
Wu, Yinghao, Vendome, Jeremie, Shapiro, Lawrence, Ben-Shaul, Avinoam, Honig, Barry
Published in Nature (London) (28.07.2011)
Published in Nature (London) (28.07.2011)
Get full text
Journal Article
Enhancing Hit Discovery in Virtual Screening through Absolute Protein–Ligand Binding Free-Energy Calculations
Chen, Wei, Cui, Di, Jerome, Steven V., Michino, Mayako, Lenselink, Eelke B., Huggins, David J., Beautrait, Alexandre, Vendome, Jeremie, Abel, Robert, Friesner, Richard A., Wang, Lingle
Published in Journal of chemical information and modeling (22.05.2023)
Published in Journal of chemical information and modeling (22.05.2023)
Get full text
Journal Article
Structure and drug resistance of the Plasmodium falciparum transporter PfCRT
Kim, Jonathan, Tan, Yong Zi, Wicht, Kathryn J., Erramilli, Satchal K., Dhingra, Satish K., Okombo, John, Vendome, Jeremie, Hagenah, Laura M., Giacometti, Sabrina I., Warren, Audrey L., Nosol, Kamil, Roepe, Paul D., Potter, Clinton S., Carragher, Bridget, Kossiakoff, Anthony A., Quick, Matthias, Fidock, David A., Mancia, Filippo
Published in Nature (London) (12.12.2019)
Published in Nature (London) (12.12.2019)
Get full text
Journal Article
Identification of a Novel 1,2,3,4-Tetrahydrobenzo[b][1,6]naphthyridine Analogue as a Potent Phosphodiesterase 5 Inhibitor with Improved Aqueous Solubility for the Treatment of Alzheimer’s Disease
Fiorito, Jole, Vendome, Jeremie, Saeed, Faisal, Staniszewski, Agnieszka, Zhang, Hong, Yan, Shijun, Deng, Shi-Xian, Arancio, Ottavio, Landry, Donald W
Published in Journal of medicinal chemistry (09.11.2017)
Published in Journal of medicinal chemistry (09.11.2017)
Get full text
Journal Article
Induced-Fit Docking Enables Accurate Free Energy Perturbation Calculations in Homology Models
Xu, Tianchuan, Zhu, Kai, Beautrait, Alexandre, Vendome, Jeremie, Borrelli, Kenneth W., Abel, Robert, Friesner, Richard A., Miller, Edward B.
Published in Journal of chemical theory and computation (13.09.2022)
Published in Journal of chemical theory and computation (13.09.2022)
Get full text
Journal Article
Fine Sampling of Sequence Space for Membrane Protein Structural Biology
Loukeris, Michael, Sanghai, Zahra Assur, Vendome, Jeremie, Hendrickson, Wayne A., Kloss, Brian, Mancia, Filippo
Published in Journal of molecular biology (23.07.2021)
Published in Journal of molecular biology (23.07.2021)
Get full text
Journal Article
Silencing c-Myc translation as a therapeutic strategy through targeting PI3Kδ and CK1ε in hematological malignancies
Deng, Changchun, Lipstein, Mark R., Scotto, Luigi, Jirau Serrano, Xavier O., Mangone, Michael A., Li, Shirong, Vendome, Jeremie, Hao, Yun, Xu, Xiaoming, Deng, Shi-Xian, Realubit, Ronald B., Tatonetti, Nicholas P., Karan, Charles, Lentzsch, Suzanne, Fruman, David A., Honig, Barry, Landry, Donald W., O'Connor, Owen A.
Published in Blood (05.01.2017)
Published in Blood (05.01.2017)
Get full text
Journal Article