Selective cytotoxic activity and DNA damage by an epoxyalkyl galactopyranoside
Burgos‐Morón, Estefanía, Pastor, Nuria, Orta, Manuel Luis, Jiménez‐Alonso, Julio José, Vega‐Holm, Margarita, Vega‐Pérez, José Manuel, Iglesias‐Guerra, Fernando, Mateos, Santiago, López‐Lázaro, Miguel, Calderón‐Montaño, José Manuel
Published in Drug development research (01.12.2018)
Published in Drug development research (01.12.2018)
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Journal Article
Synthesis of New Chiral Ketones from D-Glucose Derivatives and Their Use in the Enantioselective Epoxidation of Arylalkenes
Vega-Pérez, José Manuel, Vega Holm, Margarita, Martínez, M. Luisa, Blanco, Eugenia, Iglesias-Guerra, Fernando
Published in European Journal of Organic Chemistry (01.12.2009)
Published in European Journal of Organic Chemistry (01.12.2009)
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Book Review
Journal Article
Repurposing Study of 4-Acyl-1-phenylaminocarbonyl-2-substituted-piperazine Derivatives as Potential Anticancer Agents-In Vitro Evaluation against Breast Cancer Cells
Guillén-Mancina, Emilio, García-Lozano, María Del Rosario, Burgos-Morón, Estefanía, Mazzotta, Sarah, Martínez-Aguado, Pablo, Calderón-Montaño, José Manuel, Vega-Pérez, José Manuel, López-Lázaro, Miguel, Iglesias-Guerra, Fernando, Vega-Holm, Margarita
Published in International journal of molecular sciences (01.12.2023)
Published in International journal of molecular sciences (01.12.2023)
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Journal Article
New 4‑Acyl-1-phenylaminocarbonyl-2-phenylpiperazine Derivatives as Potential Inhibitors of Adenovirus Infection. Synthesis, Biological Evaluation, and Structure–activity Relationships
Sánchez-Céspedes, Javier, Martínez-Aguado, Pablo, Vega-Holm, Margarita, Serna-Gallego, Ana, Candela, José Ignacio, Marrugal-Lorenzo, José Antonio, Pachón, Jerónimo, Iglesias-Guerra, Fernando, Vega-Pérez, José Manuel
Published in Journal of medicinal chemistry (09.06.2016)
Published in Journal of medicinal chemistry (09.06.2016)
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Journal Article
Serinol-Based Benzoic Acid Esters as New Scaffolds for the Development of Adenovirus Infection Inhibitors: Design, Synthesis, and In Vitro Biological Evaluation
Mazzotta, Sarah, Berastegui-Cabrera, Judith, Carullo, Gabriele, Vega-Holm, Margarita, Carretero-Ledesma, Marta, Mendolia, Lara, Aiello, Francesca, Iglesias-Guerra, Fernando, Pachón, Jerónimo, Vega-Pérez, José Manuel, Sánchez-Céspedes, Javier
Published in ACS infectious diseases (11.06.2021)
Published in ACS infectious diseases (11.06.2021)
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Journal Article
In Vitro Anticancer Activity and Mechanism of Action of an Aziridinyl Galactopyranoside
Burgos-Morón, Estefanía, Pastor, Nuria, Orta, Manuel Luis, Jiménez-Alonso, Julio José, Palo-Nieto, Carlos, Vega-Holm, Margarita, Vega-Pérez, José Manuel, Iglesias-Guerra, Fernando, Mateos, Santiago, López-Lázaro, Miguel, Calderón-Montaño, José Manuel
Published in Biomedicines (01.01.2022)
Published in Biomedicines (01.01.2022)
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Journal Article
Optimization of piperazine-derived ureas privileged structures for effective antiadenovirus agents
Mazzotta, Sarah, Marrugal-Lorenzo, José Antonio, Vega-Holm, Margarita, Serna-Gallego, Ana, Álvarez-Vidal, Jaime, Berastegui-Cabrera, Judith, Pérez del Palacio, José, Díaz, Caridad, Aiello, Francesca, Pachón, Jerónimo, Iglesias-Guerra, Fernando, Vega-Pérez, José Manuel, Sánchez-Céspedes, Javier
Published in European journal of medicinal chemistry (01.01.2020)
Published in European journal of medicinal chemistry (01.01.2020)
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Journal Article
Exploration of piperazine-derived thioureas as antibacterial and anti-inflammatory agents. In vitro evaluation against clinical isolates of colistin-resistant Acinetobacter baumannii
Mazzotta, Sarah, Cebrero-Cangueiro, Tania, Frattaruolo, Luca, Vega-Holm, Margarita, Carretero-Ledesma, Marta, Sánchez-Céspedes, Javier, Cappello, Anna Rita, Aiello, Francesca, Pachón, Jerónimo, Vega-Pérez, José Manuel, Iglesias-Guerra, Fernando, Pachón-Ibáñez, María Eugenia
Published in Bioorganic & medicinal chemistry letters (15.09.2020)
Published in Bioorganic & medicinal chemistry letters (15.09.2020)
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Journal Article
GPR120/FFAR4 Pharmacology: Focus on Agonists in Type 2 Diabetes Mellitus Drug Discovery
Carullo, Gabriele, Mazzotta, Sarah, Vega-Holm, Margarita, Iglesias-Guerra, Fernando, Vega-Pérez, José Manuel, Aiello, Francesca, Brizzi, Antonella
Published in Journal of medicinal chemistry (22.04.2021)
Published in Journal of medicinal chemistry (22.04.2021)
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Journal Article
Design, synthesis and in vitro biological evaluation of a novel class of anti-adenovirus agents based on 3-amino-1,2-propanediol
Mazzotta, Sarah, Berastegui-Cabrera, Judith, Vega-Holm, Margarita, García-Lozano, María del Rosario, Carretero-Ledesma, Marta, Aiello, Francesca, Vega-Pérez, José Manuel, Pachón, Jerónimo, Iglesias-Guerra, Fernando, Sánchez-Céspedes, Javier
Published in Bioorganic chemistry (01.09.2021)
Published in Bioorganic chemistry (01.09.2021)
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Journal Article
The Pharmacy Practice Classroom project in Pharmacy Degree of the University of Seville
Guerrero, Concepción Pérez, Perales, Ma Carmen Monedero, Carrillo, Antonio Ramos, Jimenez, Javier Escamilla, Rubio, Ma José Peral, Pérez, José Manuel Vega, de Sotomayor, María Alvarez
Published in FarmaJournal (01.02.2019)
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Published in FarmaJournal (01.02.2019)
Journal Article
Piperazine-derived small molecules as potential Flaviviridae NS3 protease inhibitors. In vitro antiviral activity evaluation against Zika and Dengue viruses
del Rosario García-Lozano, María, Dragoni, Filippo, Gallego, Paloma, Mazzotta, Sarah, López-Gómez, Alejandro, Boccuto, Adele, Martínez-Cortés, Carlos, Rodríguez-Martínez, Alejandro, Pérez-Sánchez, Horacio, Manuel Vega-Pérez, José, Antonio Del Campo, José, Vicenti, Ilaria, Vega-Holm, Margarita, Iglesias-Guerra, Fernando
Published in Bioorganic chemistry (01.04.2023)
Published in Bioorganic chemistry (01.04.2023)
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Journal Article
PIPERAZINE DERIVATIVES AS ANTIVIRAL AGENTS WITH INCREASED THERAPEUTIC ACTIVITY
SÁNCHEZ CÉSPEDES, Javier, PACHÓN IBÁÑEZ, María Eugenia, PACHÓN DÍAZ, Jerónimo, MARTÍNEZ AGUADO, Pablo, IGLESIAS GUERRA, Fernando, CEBRERO CANGUEIRO, Tania, MAZZOTTA, Sarah, VEGA PÉREZ, José Manuel, VEGA HOLM, Margarita, CANDELA LENA, José Ignacio
Year of Publication 10.10.2019
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Year of Publication 10.10.2019
Patent
PIPERAZINE DERIVATIVES AS ANTIVIRAL AGENTS WITH INCREASED THERAPEUTIC ACTIVITY
SÁNCHEZ CÉSPEDES, Javier, PACHÓN IBÁÑEZ, María Eugenia, PACHÓN DÍAZ, Jerónimo, MARTÍNEZ AGUADO, Pablo, IGLESIAS GUERRA, Fernando, CEBRERO CANGUEIRO, Tania, MAZZOTTA, Sarah, VEGA PÉREZ, José Manuel, VEGA HOLM, Margarita, CANDELA LENA, José Ignacio
Year of Publication 02.01.2019
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Year of Publication 02.01.2019
Patent
PIPERAZINE DERIVATIVES AS ANTIVIRAL AGENTS WITH INCREASED THERAPEUTIC ACTIVITY
SÁNCHEZ CÉSPEDES, Javier, PACHÓN IBÁÑEZ, María Eugenia, PACHÓN DÍAZ, Jerónimo, MARTÍNEZ AGUADO, Pablo, IGLESIAS GUERRA, Fernando, CEBRERO CANGUEIRO, Tania, MAZZOTTA, Sarah, VEGA PÉREZ, José Manuel, VEGA HOLM, Margarita, CANDELA LENA, José Ignacio
Year of Publication 31.08.2017
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Year of Publication 31.08.2017
Patent
USO DE COMPUESTO N-FENIL-N'-(3-METIL-2-BUTENIL)TIOUREA PARA LA ELABORACION DE MEDICAMENTOS DESTINADOS AL TRATAMIENTO DE LA ENCEFALOPATIA HEPATICA
VEGA PEREZ, JOSE MANUEL, ROMERO GOMEZ, MANUEL, PERINAN DOMINGUEZ, IGNACIO, DIAZ HERRERO, MARIA DEL MAR, JOVER COBOS, MARIA, BAUTISTA PALOMAS, JUAN DIONISIO, IGLESIIAS GUERRA, FERNANDO
Year of Publication 22.05.2012
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Year of Publication 22.05.2012
Patent
USE OF THE COMPOUND N-PHENYL-N'-(3-METHYL-2-BUTENYL)THIOUREA FOR PRODUCING MEDICAMENTS FOR THE TREATMENT OF HEPATIC ENCEPHALOPATHY
VEGA PEREZ, JOSE MANUEL, ROMERO GOMEZ, MANUEL, PERINAN DOMINGUEZ, IGNACIO, DIAZ HERRERO, MARIA DEL MAR, IGLESIAS GUERRA, FERNANDO, JOVER COBOS, MARIA, BAUTISTA PALOMAS, JUAN DIONISIO
Year of Publication 30.06.2011
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Year of Publication 30.06.2011
Patent
USE OF THE COMPOUND N-PHENYL-N'-(3-METHYL-2-BUTENYL)THIOUREA FOR PRODUCING MEDICAMENTS FOR THE TREATMENT OF HEPATIC ENCEPHALOPATHY
VEGA PEREZ, JOSE MANUEL, ROMERO GOMEZ, MANUEL, PERINAN DOMINGUEZ, IGNACIO, DIAZ HERRERO, MARIA DEL MAR, JOVER COBOS, MARIA, BAUTISTA PALOMAS, JUAN DIONISIO, IGLESIIAS GUERRA, FERNANDO
Year of Publication 13.07.2011
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Year of Publication 13.07.2011
Patent