The highly selective and oral phosphoinositide 3-kinase delta (PI3K-δ) inhibitor roginolisib induces apoptosis in mesothelioma cells and increases immune effector cell composition
Kalla, Claudia, Ott, German, Finotello, Francesca, Niewola-Staszkowska, Karolina, Conza, Giusy Di, Lahn, Michael, van der Veen, Lars, Schüler, Julia, Falkenstern-Ge, Roger, Kopecka, Joanna, Riganti, Chiara
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Published in Translational oncology (01.05.2024)
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469 Combining a safe PI3Kd inhibitor with chemotherapy and anti-PD1 in immunotherapy-refractory NSCLC: a proof-of-concept study to allow clinical trial design
Riganti, Chiara, Scagliotti, Giorgio, Novello, Silvia, Tabbo, Fabrizio, Righi, Luisella, Neff, Laurence, Lahn, Michael, Veen, Lars Van der, Conza, Giusy Di
Published in Journal for immunotherapy of cancer (01.11.2023)
Published in Journal for immunotherapy of cancer (01.11.2023)
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922 A novel autotaxin inhibitor, IOA-289, modulates tumor, immune and stromal cell function and has monotherapy activity in fibrotic cancer models
Deken, Marcel, Niewola, Karolina, Matas-Rico, Elisa, Medhi, Ragini, Carruthers, Alan, Cheasty, Anne, Peyruchaud, Olivier, Fraser, Amy, Shah, Pritom, Moolenaar, Wouter, Veen, Lars van der, Lahn, Michael, Johnson, Zoe
Published in Journal for immunotherapy of cancer (01.11.2021)
Published in Journal for immunotherapy of cancer (01.11.2021)
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Origin of the Bite Angle Effect on Rhodium Diphosphine Catalyzed Hydroformylation
van der Veen, Lars A, Keeven, Peter H, Schoemaker, Gerard C, Reek, Joost N. H, Kamer, Paul C. J, van Leeuwen, Piet W. N. M, Lutz, Martin, Spek, Anthony L
Published in Organometallics (06.03.2000)
Published in Organometallics (06.03.2000)
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Electronic Effect on Rhodium Diphosphine Catalyzed Hydroformylation: The Bite Angle Effect Reconsidered
van der Veen, Lars A, Boele, Maarten D. K, Bregman, Frank R, Kamer, Paul C. J, van Leeuwen, Piet W. N. M, Goubitz, Kees, Fraanje, Jan, Schenk, Henk, Bo, Carles
Published in Journal of the American Chemical Society (18.11.1998)
Published in Journal of the American Chemical Society (18.11.1998)
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New Phosphacyclic Diphosphines for Rhodium-Catalyzed Hydroformylation
van der Veen, Lars A, Kamer, Paul C. J, van Leeuwen, Piet W. N. M
Published in Organometallics (08.11.1999)
Published in Organometallics (08.11.1999)
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P1114: HIGHLY SELECTIVE ALLOSTERIC MODULATOR OF THE PHOSPHOINOSITIDE 3‐KINASE DELTA (PI3KΔ) ROGINOLISIB (IOA‐244) IN A DOSE ESCALATION STUDY OF PATIENTS WITH REFRACTORY/RELAPSED FOLLICULAR LYMPHOMA (FL)
Carlo‐Stella, Carmelo, Lahn, Michael, Hammett, Tracey, Veen, Lars, Zorrilla, Rebeca, Pickering, Catherine, Santoro, Armando
Published in HemaSphere (08.08.2023)
Published in HemaSphere (08.08.2023)
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Catalytic asymmetric hydrogenation of heterocyclic ketone-derived hydrazones, pronounced solvent effect on the inversion of configuration
Haddad, Nizar, Qu, Bo, Rodriguez, Sonia, van der Veen, Lars, Reeves, Diana C., Gonnella, Nina C., Lee, Heewon, Grinberg, Nelu, Ma, Shengli, Krishnamurthy, Dhileepkumar, Wunberg, Tobias, Senanayake, Chris H.
Published in Tetrahedron letters (20.07.2011)
Published in Tetrahedron letters (20.07.2011)
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A Robust, Environmentally Benign Catalyst for Highly Selective Hydroformylation
Sandee, Albertus J., van der Veen, Lars A., Reek, Joost N. H., Kamer, Paul C. J., Lutz, Martin, Spek, Anthony L., van Leeuwen, Piet W. N. M.
Published in Angewandte Chemie (International ed.) (02.11.1999)
Published in Angewandte Chemie (International ed.) (02.11.1999)
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Hydroxycarbonylation of styrene with palladium catalysts: The influence of the mono- and bidentate phosphorus ligand
del Rı́o, Inmaculada, Ruiz, Nuria, Claver, Carmen, van der Veen, Lars A., van Leeuwen, Piet W.N.M.
Published in Journal of molecular catalysis. A, Chemical (06.11.2000)
Published in Journal of molecular catalysis. A, Chemical (06.11.2000)
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Chiral Cooperativity in Diastereomeric Diphosphite Ligands: Effects on the Rhodium-Catalyzed Enantioselective Hydroformylation of Styrene
Buisman, Godfried J. H, van der Veen, Lars A, Klootwijk, Angélique, de Lange, Wim G. J, Kamer, Paul C. J, van Leeuwen, Piet W. N. M, Vogt, Dieter
Published in Organometallics (24.06.1997)
Published in Organometallics (24.06.1997)
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A novel orally available type IV autotaxin inhibitor, IOA-289, ameliorates steatosis and fibrosis in a preclinical model of non-alcoholic steatohepatitis
ten Hove, Marit, Di Conza, Giusy, Niewola, Karolina, Deken, Marcel, van der Veen, Lars, Bansal, Ruchi
Published in Journal of hepatology (01.06.2023)
Published in Journal of hepatology (01.06.2023)
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WED-441 - A novel orally available type IV autotaxin inhibitor, IOA-289, ameliorates steatosis and fibrosis in a preclinical model of non-alcoholic steatohepatitis
ten Hove, Marit, Di Conza, Giusy, Niewola, Karolina, Deken, Marcel, van der Veen, Lars, Bansal, Ruchi
Published in Journal of hepatology (01.06.2023)
Published in Journal of hepatology (01.06.2023)
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Roginolisib a Highly Selective Allosteric Modulator of the Phosphoinositide 3-Kinase Delta (PI3Kδ) in Patients with Refractory/Relapsed Follicular Lymphoma
Carlo-Stella, Carmelo, Lahn, Michael, Hammett, Tracey, Kaur, Paramjit, Zorrilla, Rebeca, Di Conza, Giusy, van der Veen, Lars, Pickering, Catherine, Santoro, Armando
Published in Blood (02.11.2023)
Published in Blood (02.11.2023)
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Novel Pi3kδ Inhibitor Roginolisib Synergizes with the Bcl-2 Inhibitor Venetoclax in Hematological Malignancies
Kandathilparambil Sasi, Binu, Tarantelli, Chiara, Civanelli, Elisa, Cannas, Eleonora, Fernandes, Stacey M, Shupe, Samantha J., Lahn, Michael, van der Veen, Lars, Di Conza, Giusy, Bertoni, Francesco, Brown, Jennifer R.
Published in Blood (02.11.2023)
Published in Blood (02.11.2023)
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