Distinct In Vitro Binding Profile of the Somatostatin Receptor Subtype 2 Antagonist [ 177 Lu]Lu-OPS201 Compared to the Agonist [ 177 Lu]Lu-DOTA-TATE
Mansi, Rosalba, Plas, Pascale, Vauquelin, Georges, Fani, Melpomeni
Published in Pharmaceuticals (Basel, Switzerland) (04.12.2021)
Published in Pharmaceuticals (Basel, Switzerland) (04.12.2021)
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Mechanisms of PDZ domain scaffold assembly illuminated by use of supported cell membrane sheets
Erlendsson, Simon, Thorsen, Thor Seneca, Vauquelin, Georges, Ammendrup-Johnsen, Ina, Wirth, Volker, Martinez, Karen L, Teilum, Kaare, Gether, Ulrik, Madsen, Kenneth Lindegaard
Published in eLife (03.01.2019)
Published in eLife (03.01.2019)
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The Role of Binding Kinetics in GPCR Drug Discovery
Swinney, David C, Haubrich, Brad A, Van Liefde, Isabelle, Vauquelin, Georges
Published in Current topics in medicinal chemistry (01.01.2015)
Published in Current topics in medicinal chemistry (01.01.2015)
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A study of the molecular mechanism of binding kinetics and long residence times of human CCR5 receptor small molecule allosteric ligands
Swinney, David C, Beavis, Paul, Chuang, Kai‐Ting, Zheng, Yue, Lee, Ina, Gee, Peter, Deval, Jerome, Rotstein, David M, Dioszegi, Marianna, Ravendran, Palani, Zhang, Jun, Sankuratri, Surya, Kondru, Rama, Vauquelin, Georges
Published in British journal of pharmacology (01.07.2014)
Published in British journal of pharmacology (01.07.2014)
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Pressor and renal hemodynamic effects of the novel angiotensin A peptide are angiotensin II type 1A receptor dependent
Yang, Rui, Smolders, Ilse, Vanderheyden, Patrick, Demaegdt, Heidi, Van Eeckhaut, Ann, Vauquelin, Georges, Lukaszuk, Aneta, Tourwé, Dirk, Chai, Siew Yeen, Albiston, Anthony L, Nahmias, Clara, Walther, Thomas, Dupont, Alain G
Published in Hypertension (Dallas, Tex. 1979) (01.05.2011)
Published in Hypertension (Dallas, Tex. 1979) (01.05.2011)
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Neurokinin 1 Receptor Antagonists: Correlation between in Vitro Receptor Interaction and in Vivo Efficacy
Lindström, Erik, von Mentzer, Bengt, Påhlman, Ingrid, Ahlstedt, Ingela, Uvebrant, Anna, Kristensson, Elin, Martinsson, Rakel, Novén, Anna, de Verdier, Jennie, Vauquelin, Georges
Published in The Journal of pharmacology and experimental therapeutics (01.09.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2007)
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Involvement of the AT₁ receptor subtype in the effects of angiotensin IV and LVV-haemorphin 7 on hippocampal neurotransmitter levels and spatial working memory
De Bundel, Dimitri, Demaegdt, Heidi, Lahoutte, Tony, Caveliers, Vicky, Kersemans, Ken, Ceulemans, Ann-Gaelle, Vauquelin, Georges, Clinckers, Ralph, Vanderheyden, Patrick, Michotte, Yvette, Smolders, Ilse
Published in Journal of neurochemistry (01.03.2010)
Published in Journal of neurochemistry (01.03.2010)
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