tracerDB: a crowdsourced fluorescent tracer database for target engagement analysis
Dopfer, Johannes, Vasta, James D, Müller, Susanne, Knapp, Stefan, Robers, Matthew B, Schwalm, Martin P
Published in Nature communications (05.07.2024)
Published in Nature communications (05.07.2024)
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Quantifying CDK inhibitor selectivity in live cells
Wells, Carrow I, Vasta, James D, Corona, Cesear R, Wilkinson, Jennifer, Zimprich, Chad A, Ingold, Morgan R, Pickett, Julie E, Drewry, David H, Pugh, Kathryn M, Schwinn, Marie K, Hwang, Byounghoon Brian, Zegzouti, Hicham, Huber, Kilian V M, Cong, Mei, Meisenheimer, Poncho L, Willson, Timothy M, Robers, Matthew B
Published in Nature communications (02.06.2020)
Published in Nature communications (02.06.2020)
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Development of Cell Permeable NanoBRET Probes for the Measurement of PLK1 Target Engagement in Live Cells
Yang, Xuan, Smith, Jeffery L, Beck, Michael T, Wilkinson, Jennifer M, Michaud, Ani, Vasta, James D, Robers, Matthew B, Willson, Timothy M
Published in Molecules (Basel, Switzerland) (25.03.2023)
Published in Molecules (Basel, Switzerland) (25.03.2023)
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Dual targeting of the androgen receptor and PI3K/AKT/mTOR pathways in prostate cancer models improves antitumor efficacy and promotes cell apoptosis
Sugawara, Tatsuo, Nevedomskaya, Ekaterina, Heller, Simon, Böhme, Annika, Lesche, Ralf, Ahsen, Oliver, Grünewald, Sylvia, Nguyen, Holly M., Corey, Eva, Baumgart, Simon J., Georgi, Victoria, Pütter, Vera, Fernández‐Montalván, Amaury, Vasta, James D., Robers, Matthew B., Politz, Oliver, Mumberg, Dominik, Haendler, Bernard
Published in Molecular oncology (01.03.2024)
Published in Molecular oncology (01.03.2024)
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A Toolbox for the Generation of Chemical Probes for Baculovirus IAP Repeat Containing Proteins
Schwalm, Martin P., Berger, Lena M., Meuter, Maximilian N., Vasta, James D., Corona, Cesear R., Röhm, Sandra, Berger, Benedict-Tilman, Farges, Frederic, Beinert, Sebastian M., Preuss, Franziska, Morasch, Viktoria, Rogov, Vladimir V., Mathea, Sebastian, Saxena, Krishna, Robers, Matthew B., Müller, Susanne, Knapp, Stefan
Published in Frontiers in cell and developmental biology (26.05.2022)
Published in Frontiers in cell and developmental biology (26.05.2022)
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Quantitative Live-Cell Kinetic Degradation and Mechanistic Profiling of PROTAC Mode of Action
Riching, Kristin M, Mahan, Sarah, Corona, Cesear R, McDougall, Mark, Vasta, James D, Robers, Matthew B, Urh, Marjeta, Daniels, Danette L
Published in ACS chemical biology (21.09.2018)
Published in ACS chemical biology (21.09.2018)
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Journal Article
KRAS is vulnerable to reversible switch-II pocket engagement in cells
Vasta, James D, Peacock, D Matthew, Zheng, Qinheng, Walker, Joel A, Zhang, Ziyang, Zimprich, Chad A, Thomas, Morgan R, Beck, Michael T, Binkowski, Brock F, Corona, Cesear R, Robers, Matthew B, Shokat, Kevan M
Published in Nature chemical biology (01.06.2022)
Published in Nature chemical biology (01.06.2022)
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Journal Article
Quantitative, Wide-Spectrum Kinase Profiling in Live Cells for Assessing the Effect of Cellular ATP on Target Engagement
Vasta, James D., Corona, Cesear R., Wilkinson, Jennifer, Zimprich, Chad A., Hartnett, James R., Ingold, Morgan R., Zimmerman, Kristopher, Machleidt, Thomas, Kirkland, Thomas A., Huwiler, Kristin G., Ohana, Rachel Friedman, Slater, Michael, Otto, Paul, Cong, Mei, Wells, Carrow I., Berger, Benedict-Tilman, Hanke, Thomas, Glas, Carina, Ding, Ke, Drewry, David H., Huber, Kilian V.M., Willson, Timothy M., Knapp, Stefan, Müller, Susanne, Meisenheimer, Poncho L., Fan, Frank, Wood, Keith V., Robers, Matthew B.
Published in Cell chemical biology (15.02.2018)
Published in Cell chemical biology (15.02.2018)
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Journal Article
Binding Kinetics Survey of the Drugged Kinome
Georgi, Victoria, Schiele, Felix, Berger, Benedict-Tilman, Steffen, Andreas, Marin Zapata, Paula A, Briem, Hans, Menz, Stephan, Preusse, Cornelia, Vasta, James D, Robers, Matthew B, Brands, Michael, Knapp, Stefan, Fernández-Montalván, Amaury
Published in Journal of the American Chemical Society (21.11.2018)
Published in Journal of the American Chemical Society (21.11.2018)
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Discovery of a selective inhibitor of doublecortin like kinase 1
Ferguson, Fleur M, Nabet, Behnam, Raghavan, Srivatsan, Liu, Yan, Leggett, Alan L, Kuljanin, Miljan, Kalekar, Radha L, Yang, Annan, He, Shuning, Wang, Jinhua, Ng, Raymond W S, Sulahian, Rita, Li, Lianbo, Poulin, Emily J, Huang, Ling, Koren, Jost, Dieguez-Martinez, Nora, Espinosa, Sergio, Zeng, Zhiyang, Corona, Cesear R, Vasta, James D, Ohi, Ryoma, Sim, Taebo, Kim, Nam Doo, Harshbarger, Wayne, Lizcano, Jose M, Robers, Matthew B, Muthaswamy, Senthil, Lin, Charles Y, Look, A Thomas, Haigis, Kevin M, Mancias, Joseph D, Wolpin, Brian M, Aguirre, Andrew J, Hahn, William C, Westover, Kenneth D, Gray, Nathanael S
Published in Nature chemical biology (01.06.2020)
Published in Nature chemical biology (01.06.2020)
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Protomer selectivity of type II RAF inhibitors within the RAS/RAF complex
Vasta, James D., Michaud, Ani, Zimprich, Chad A., Beck, Michael T., Swiatnicki, Matthew R., Zegzouti, Hicham, Thomas, Morgan R., Wilkinson, Jennifer, Crapster, J. Aaron, Robers, Matthew B.
Published in Cell chemical biology (16.11.2023)
Published in Cell chemical biology (16.11.2023)
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DELs enable the development of BRET probes for target engagement studies in cells
Teske, Kelly A, Su, Wenji, Corona, Cesear R, Wen, Jing, Deng, Jason, Ping, Yan, Zhang, Zaihong, Zhang, Qi, Wilkinson, Jennifer, Beck, Michael T, Nealey, Kendra R, Vasta, James D, Cong, Mei, Meisenheimer, Poncho L, Kuai, Letian, Robers, Matthew B
Published in Cell chemical biology (17.08.2023)
Published in Cell chemical biology (17.08.2023)
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Journal Article
Design of a “Two-in-One” Mutant-Selective Epidermal Growth Factor Receptor Inhibitor That Spans the Orthosteric and Allosteric Sites
Wittlinger, Florian, Heppner, David E, To, Ciric, Günther, Marcel, Shin, Bo Hee, Rana, Jaimin K, Schmoker, Anna M, Beyett, Tyler S, Berger, Lena M, Berger, Benedict-Tilman, Bauer, Nicolas, Vasta, James D, Corona, Cesear R, Robers, Matthew B, Knapp, Stefan, Jänne, Pasi A, Eck, Michael J, Laufer, Stefan A
Published in Journal of medicinal chemistry (27.01.2022)
Published in Journal of medicinal chemistry (27.01.2022)
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