Synthesis and multifaceted pharmacological activity of novel quinazoline NHE-1 inhibitors
Spasov, Alexander, Ozerov, Alexander, Vassiliev, Pavel, Kosolapov, Vadim, Gurova, Natalia, Kucheryavenko, Aida, Naumenko, Ludmila, Babkov, Denis, Sirotenko, Viktor, Taran, Alena, Litvinov, Roman, Borisov, Alexander, Klochkov, Vladlen, Merezhkina, Darya, Miroshnikov, Mikhail, Uskov, Georgy, Ovsyankina, Nadezhda
Published in Scientific reports (21.12.2021)
Published in Scientific reports (21.12.2021)
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Journal Article
Computational Analysis of CD46 Protein Interaction with SARS-CoV-2 Structural Proteins: Elucidating a Putative Viral Entry Mechanism into Human Cells
Vassiliev, Pavel, Gusev, Evgenii, Komelkova, Maria, Kochetkov, Andrey, Dobrynina, Maria, Sarapultsev, Alexey
Published in Viruses (23.11.2023)
Published in Viruses (23.11.2023)
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Immunomodulatory Action of Substituted 1,3,4-Thiadiazines on the Course of Myocardial Infarction
Sarapultsev, Alexey P, Vassiliev, Pavel M, Sarapultsev, Petr A, Chupakhin, Oleg N, Ianalieva, Laura R, Sidorova, Larisa P
Published in Molecules (Basel, Switzerland) (02.07.2018)
Published in Molecules (Basel, Switzerland) (02.07.2018)
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Journal Article
Design, Synthesis and Pharmacological Evaluation of Novel C2,C3-Quinoxaline Derivatives as Promising Anxiolytic Agents
Maltsev, Dmitriy V., Skripka, Maria O., Spasov, Alexander A., Vassiliev, Pavel M., Perfiliev, Maxim A., Divaeva, Lyudmila N., Zubenko, Alexander A., Morkovnik, Anatolii S., Klimenko, Alexander I., Miroshnikov, Mikhail V., Klochkov, Vladlen G., Ianalieva, Laura R.
Published in International journal of molecular sciences (19.11.2022)
Published in International journal of molecular sciences (19.11.2022)
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Journal Article
Synthesis and Pharmacological Evaluation of Novel 2,3,4,5-tetrahydro[1,3]diazepino[1,2-a]benzimidazole Derivatives as Promising Anxiolytic and Analgesic Agents
Maltsev, Dmitriy V., Spasov, Alexander A., Vassiliev, Pavel M., Skripka, Maria O., Miroshnikov, Mikhail V., Kochetkov, Andrey N., Eliseeva, Nataliya V., Lifanova, Yuliya V., Kuzmenko, Tatyana A., Divaeva, Lyudmila N., Morkovnik, Anatolii S.
Published in Molecules (Basel, Switzerland) (06.10.2021)
Published in Molecules (Basel, Switzerland) (06.10.2021)
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Journal Article
Consensus Ensemble Multitarget Neural Network Model of Anxiolytic Activity of Chemical Compounds and Its Use for Multitarget Pharmacophore Design
Vassiliev, Pavel M, Maltsev, Dmitriy V, Spasov, Alexander A, Perfilev, Maxim A, Skripka, Maria O, Kochetkov, Andrey N
Published in Pharmaceuticals (Basel, Switzerland) (11.05.2023)
Published in Pharmaceuticals (Basel, Switzerland) (11.05.2023)
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Role of TGF-β1/SMADs signalling pathway in resveratrol-induced reduction of extracellular matrix deposition by dexamethasone-treated human trabecular meshwork cells
Bakar, Amy Suzana Abu, Razali, Norhafiza, Agarwal, Renu, Iezhitsa, Igor, Perfilev, Maxim A., Vassiliev, Pavel M.
Published in The Korean journal of physiology & pharmacology (01.07.2024)
Published in The Korean journal of physiology & pharmacology (01.07.2024)
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Journal Article
Antimicrobial Activity of Substituted Benzopentathiepin-6-amines
Khomenko, Tatyana M., Korchagina, Dina, Baev, Dmitry S., Vassiliev, Pavel M., Volcho, Konstantin P., Salakhutdinov, Nariman F.
Published in Journal of antibiotics (01.08.2019)
Published in Journal of antibiotics (01.08.2019)
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Journal Article
Searching for new anxiolytic agents among derivatives of 11-dialkylaminoethyl-2,3,4,5-tetrahydrodiazepino[1,2-a]benzimidazole
Maltsev, Dmitriy V., Spasov, Alexander A., Yakovlev, Dmitriy S., Vassiliev, Pavel M., Skripka, Maria O., Miroshnikov, Mikhail V., Sultanova, Kira T., Kochetkov, Andrey N., Divaeva, Lyudmila N., Kuzmenko, Tatyana A., Morkovnik, Anatolii S.
Published in European journal of pharmaceutical sciences (01.06.2021)
Published in European journal of pharmaceutical sciences (01.06.2021)
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Journal Article
Combined In Silico, Ex Vivo, and In Vivo Assessment of L-17, a Thiadiazine Derivative with Putative Neuro- and Cardioprotective and Antidepressant Effects
Sarapultsev, Alexey, Vassiliev, Pavel, Grinchii, Daniil, Kiss, Alexander, Mach, Mojmir, Osacka, Jana, Balloova, Alexandra, Paliokha, Ruslan, Kochetkov, Andrey, Sidorova, Larisa, Sarapultsev, Petr, Chupakhin, Oleg, Rantsev, Maxim, Spasov, Alexander, Dremencov, Eliyahu
Published in International journal of molecular sciences (20.12.2021)
Published in International journal of molecular sciences (20.12.2021)
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Journal Article
Bornyl Derivatives of p-(Benzyloxy)Phenylpropionic Acid: In Vivo Evaluation of Antidiabetic Activity
Kuranov, Sergey, Luzina, Olga, Khvostov, Mikhail, Baev, Dmitriy, Kuznetsova, Darya, Zhukova, Nataliya, Vassiliev, Pavel, Kochetkov, Andrey, Tolstikova, Tatyana, Salakhutdinov, Nariman
Published in Pharmaceuticals (Basel, Switzerland) (19.11.2020)
Published in Pharmaceuticals (Basel, Switzerland) (19.11.2020)
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Journal Article
Pyridoxine dipharmacophore derivatives as potent glucokinase activators for the treatment of type 2 diabetes mellitus
Dzyurkevich, Mikhail S, Babkov, Denis A, Shtyrlin, Nikita V, Mayka, Olga Yu, Iksanova, Alfiya G, Vassiliev, Pavel M, Balakin, Konstantin V, Spasov, Alexander A, Tarasov, Vadim V, Barreto, George, Shtyrlin, Yurii G, Aliev, Gjumrakch
Published in Scientific reports (22.11.2017)
Published in Scientific reports (22.11.2017)
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Journal Article
Synthesis and Evaluation of Novel [1,2,4]Triazolo[5,1‐c][1,2,4]‐triazines and Pyrazolo[5,1‐c][1,2,4]triazines as Potential Antidiabetic Agents
Rusinov, Vladimir L., Sapozhnikova, Irina M., Bliznik, Anastasiya M., Chupakhin, Oleg N., Charushin, Valery N., Spasov, Alexander A., Vassiliev, Pavel M., Kuznetsova, Valentina A., Rashchenko, Andrey I., Babkov, Denis A.
Published in Archiv der Pharmazie (Weinheim) (01.05.2017)
Published in Archiv der Pharmazie (Weinheim) (01.05.2017)
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Journal Article
Hypoglycemic potential of cyclic guanidine derivatives
Spasov, Alexander A., Vassiliev, Pavel M., Lenskaya, Karina V., Anisimova, Vera A., Kuzmenko, Tatyana A., Morkovnik, Anatolii S., Kosolapov, Vadim A., Babkov, Denis A.
Published in Pure and applied chemistry (01.08.2017)
Published in Pure and applied chemistry (01.08.2017)
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Journal Article
Author Correction: Pyridoxine dipharmacophore derivatives as potent glucokinase activators for the treatment of type 2 diabetes mellitus
Dzyurkevich, Mikhail S, Babkov, Denis A, Shtyrlin, Nikita V, Mayka, Olga Yu, Iksanova, Alfiya G, Vassiliev, Pavel M, Balakin, Konstantin V, Spasov, Alexander A, Tarasov, Vadim V, Barreto, George, Shtyrlin, Yurii G, Aliev, Gjumrakch
Published in Scientific reports (19.04.2018)
Published in Scientific reports (19.04.2018)
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Journal Article
3-Amino(azido)-4,6-aryl(hetaryl)thieno[2,3-b]pyridines and benzo(furo,thieno)[c]thieno[2,3,4-i,j]-2,7-naphthyridines on their basis: synthesis, spectral properties, and prediction of biological activity
Vasilin, Vladimir K., Kanishcheva, Eugeniya A., Stroganova, Tat’yana А., Volynkin, Vitaly А., Gizhinskaya, Anzhelika V., Vassiliev, Pavel M., Krapivin, Gennady D.
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.08.2020)
Published in Chemistry of heterocyclic compounds (New York, N.Y. 1965) (01.08.2020)
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Journal Article
Unusual Oxidative Dimerization in the 3‑Aminothieno[2,3‑b]pyridine-2-carboxamide Series
Stroganova, Tatyana A, Vasilin, Vladimir K, Dotsenko, Victor V, Aksenov, Nicolai A, Morozov, Pavel G, Vassiliev, Pavel M, Volynkin, Vitaly A, Krapivin, Gennady D
Published in ACS omega (08.06.2021)
Published in ACS omega (08.06.2021)
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Journal Article
Design, Synthesis and Pharmacological Evaluation of Novel C 2 ,C 3 -Quinoxaline Derivatives as Promising Anxiolytic Agents
Maltsev, Dmitriy V, Skripka, Maria O, Spasov, Alexander A, Vassiliev, Pavel M, Perfiliev, Maxim A, Divaeva, Lyudmila N, Zubenko, Alexander A, Morkovnik, Anatolii S, Klimenko, Alexander I, Miroshnikov, Mikhail V, Klochkov, Vladlen G, Ianalieva, Laura R
Published in International journal of molecular sciences (19.11.2022)
Published in International journal of molecular sciences (19.11.2022)
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Journal Article
Data on the effects of imidazo[1,2-a]benzimidazole and pyrimido[1,2-a]benzimidazole compounds on intraocular pressure of ocular normotensive rats
Marcus, Adrian Julian, Iezhitsa, Igor, Agarwal, Renu, Vassiliev, Pavel, Spasov, Alexander, Zhukovskaya, Olga, Anisimova, Vera, Mohd Ismail, Nafeeza
Published in Data in brief (01.06.2018)
Published in Data in brief (01.06.2018)
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Journal Article
Relationship between intraocular pressure lowering effect and chemical structure of imidazo[1,2-a]benzimidazole and pyrimido[1,2-a]benzimidazole derivatives
Vassiliev, Pavel, Iezhitsa, Igor, Agarwal, Renu, Marcus, Adrian Julian, Spasov, Alexander, Zhukovskaya, Olga, Anisimova, Vera
Published in Data in brief (01.06.2018)
Published in Data in brief (01.06.2018)
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