Opportunities and Challenges for the Development of MRCK Kinases Inhibitors as Potential Cancer Chemotherapeutics
Ruscetta, Vanessa M, Seaton, Taj J, Shakeel, Aleen, Vasconcelos, Stanley N S, Viirre, Russell D, Adler, Marc J, Olson, Michael F
Published in Cells (Basel, Switzerland) (01.02.2023)
Published in Cells (Basel, Switzerland) (01.02.2023)
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Journal Article
Discovery of a Potent Dual SLK/STK10 Inhibitor Based on a Maleimide Scaffold
Serafim, Ricardo A. M, Sorrell, Fiona J, Berger, Benedict-Tilman, Collins, Ross J, Vasconcelos, Stanley N. S, Massirer, Katlin B, Knapp, Stefan, Bennett, James, Fedorov, Oleg, Patel, Hitesh, Zuercher, William J, Elkins, Jonathan M
Published in Journal of medicinal chemistry (23.09.2021)
Published in Journal of medicinal chemistry (23.09.2021)
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Journal Article
One-pot Fluorination and Organocatalytic Robinson Annulation for Asymmetric Synthesis of Mono- and Difluorinated Cyclohexenones
Huang, Xin, Zhao, Weizhao, Zhang, Xiaofeng, Liu, Miao, Vasconcelos, Stanley N S, Zhang, Wei
Published in Molecules (Basel, Switzerland) (04.09.2018)
Published in Molecules (Basel, Switzerland) (04.09.2018)
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Journal Article
Development of Pyridine-based Inhibitors for the Human Vaccinia-related Kinases 1 and 2
Serafim, Ricardo A. M, de Souza Gama, Fernando H, Dutra, Luiz A, dos Reis, Caio V, Vasconcelos, Stanley N. S, da Silva Santiago, André, Takarada, Jéssica E, Di Pillo, Fúlvia, Azevedo, Hatylas, Mascarello, Alessandra, Elkins, Jonathan M, Massirer, Katlin B, Gileadi, Opher, Guimarães, Cristiano R. W, Couñago, Rafael M
Published in ACS medicinal chemistry letters (12.09.2019)
Published in ACS medicinal chemistry letters (12.09.2019)
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Journal Article
Synthesis, molecular and crystal structure analysis of 1-(4-Methylbenzenesulfonyl)indole-3-carbaldehyde and DFT investigation of its rotational conformers
Zukerman-Schpector, Julio, Madureira, Lucas Sousa, Wulf, Glaudeston Dutra, Stefani, Hélio A, Vasconcelos, Stanley N S, Ng, Seik Weng, Tiekink, Edward R T
Published in Molecules (Basel, Switzerland) (13.02.2014)
Published in Molecules (Basel, Switzerland) (13.02.2014)
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Journal Article
Synthesis of 5-Organotellanyl-1H-1,2,3-triazoles: Functionalization of the 5-Position Scaffold by the Sonogashira Cross-Coupling Reaction
Stefani, Hélio A., Vasconcelos, Stanley N. S., Manarin, Flávia, Leal, Daiana M., Souza, Frederico B., Madureira, Lucas Sousa, Zukerman-Schpector, Julio, Eberlin, Marcos N., Godoi, Marla N., de Souza Galaverna, Renan
Published in European journal of organic chemistry (01.06.2013)
Published in European journal of organic chemistry (01.06.2013)
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Journal Article
Discovery of pyrazolo[3,4-d]pyrimidines as novel mitogen-activated protein kinase kinase 3 (MKK3) inhibitors
Takarada, Jessica E., Cunha, Micael R., Almeida, Vitor M., Vasconcelos, Stanley N. S., Santiago, Andre S., Godoi, Paulo H., Salmazo, Anita, Ramos, Priscila Z., Fala, Angela M., De Souza, Lucas R., Da Silva, Italo E. P., Bengtson, Mario H., Massirer, Katlin B., Counago, Rafael M.
Published in Bioorganic & medicinal chemistry (15.01.2024)
Published in Bioorganic & medicinal chemistry (15.01.2024)
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Journal Article
Stereoselective Oxa‐Michael Addition of Tyrosine to Propargyl Aldehyde/Esters: Formation of Benzofurans and Flavones
Vasconcelos, Stanley N. S., Oliveira, Isadora Maria, Shamim, Anwar, Zukerman‐Schpector, Julio, Pimenta, Daniel C., Stefani, Hélio A.
Published in Advanced synthesis & catalysis (17.09.2019)
Published in Advanced synthesis & catalysis (17.09.2019)
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Journal Article
A Target Engagement Assay to Assess Uptake, Potency, and Retention of Antibiotics in Living Bacteria
Fanti, Rebeka C., Vasconcelos, Stanley N. S., Catta-Preta, Carolina M. C., Sullivan, Jaryd R., Riboldi, Gustavo P., dos Reis, Caio V., Ramos, Priscila Z., Edwards, Aled M., Behr, Marcel A., Couñago, Rafael M.
Published in ACS infectious diseases (12.08.2022)
Published in ACS infectious diseases (12.08.2022)
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Journal Article
3-Alkenyltyrosines Accessed by Suzuki-Miyaura Coupling: A Key Intermediate in the Synthesis and Mechanistic Study of Povarov Multicomponent Reactions
Vasconcelos, Stanley N. S., Menezes da Silva, Vitor H., Braga, Ataualpa A. C., Shamim, Anwar, Souza, Frederico B., Pimenta, Daniel C., Stefani, Helio A.
Published in Asian journal of organic chemistry (01.07.2017)
Published in Asian journal of organic chemistry (01.07.2017)
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Journal Article
Synthesis of symmetrical biaryl compounds by homocoupling reaction
Vasconcelos, Stanley N.S., Reis, Joel S., de Oliveira, Isadora M., Balfour, Michael N., Stefani, Hélio A.
Published in Tetrahedron (29.03.2019)
Published in Tetrahedron (29.03.2019)
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Journal Article
Ligand and copper free Sonogashira coupling to achieve 2-alkynyl d-glucal derivatives: regioselective electrophile promoted nucleophilic 5-endo-dig cyclization
Shamim, Anwar, Vasconcelos, Stanley N.S., Ali, Bakhat, Madureira, Lucas Sousa, Zukerman-Schpector, J., Stefani, Hélio A.
Published in Tetrahedron letters (21.10.2015)
Published in Tetrahedron letters (21.10.2015)
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Journal Article
ChemInform Abstract: Synthesis and Applications of 4-Substituted 1-(4-Iodophenyl)pyrrolidine-2,5-diones
Ali, Bakhat, Shamim, Anwar, Vasconcelos, Stanley N. S., Stefani, Helio A.
Published in ChemInform (01.11.2015)
Published in ChemInform (01.11.2015)
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