New RNA Purine Building Blocks, 4′-Selenopurine Nucleosides: First Synthesis and Unusual Mixture of Sugar Puckerings
Yu, Jinha, Kim, Jin-Hee, Lee, Hyuk Woo, Alexander, Varughese, Ahn, Hee-Chul, Choi, Won Jun, Choi, Jungwon, Jeong, Lak Shin
Published in Chemistry : a European journal (26.04.2013)
Published in Chemistry : a European journal (26.04.2013)
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Structure–activity relationships of 2′-modified-4′-selenoarabinofuranosyl-pyrimidines as anticancer agents
Kim, Jin-Hee, Yu, Jinha, Alexander, Varughese, Choi, Jung Hee, Song, Jayoung, Lee, Hyuk Woo, Kim, Hea Ok, Choi, Jungwon, Lee, Sang Kook, Jeong, Lak Shin
Published in European journal of medicinal chemistry (18.08.2014)
Published in European journal of medicinal chemistry (18.08.2014)
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Journal Article
Synthesis and biological evaluation of 2′-substituted-4′-selenoribofuranosyl pyrimidines as antitumor agents
Alexander, Varughese, Song, Jayoung, Yu, Jinha, Choi, Jung Hee, Kim, Jin-Hee, Lee, Sang Kook, Choi, Won Jun, Jeong, Lak Shin
Published in Archives of pharmacal research (01.06.2015)
Published in Archives of pharmacal research (01.06.2015)
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Improved synthesis of a DNA-dependent protein kinase inhibitor IC86621
Chandra, Girish, Alexander, Varughese, Lee, Hyuk Woo, Jeong, Lak Shin
Published in Archives of pharmacal research (01.04.2012)
Published in Archives of pharmacal research (01.04.2012)
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Structure–Activity Relationships of Truncated C2- or C8-Substituted Adenosine Derivatives as Dual Acting A2A and A3 Adenosine Receptor Ligands
Hou, Xiyan, Majik, Mahesh S, Kim, Kyunglim, Pyee, Yuna, Lee, Yoonji, Alexander, Varughese, Chung, Hwa-Jin, Lee, Hyuk Woo, Chandra, Girish, Lee, Jin Hee, Park, Seul-gi, Choi, Won Jun, Kim, Hea Ok, Phan, Khai, Gao, Zhan-Guo, Jacobson, Kenneth A, Choi, Sun, Lee, Sang Kook, Jeong, Lak Shin
Published in Journal of medicinal chemistry (12.01.2012)
Published in Journal of medicinal chemistry (12.01.2012)
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Journal Article
Discovery of A New Human A2A Adenosine Receptor Agonist, Truncated 2-Hexynyl-4′-thioadenosine
Hou, Xiyan, Kim, Hea Ok, Alexander, Varughese, Kim, Kyunglim, Choi, Sun, Park, Seul-gi, Lee, Jin Hee, Yoo, Lena S, Gao, Zhan-Guo, Jacobson, Kenneth A, Jeong, Lak Shin
Published in ACS medicinal chemistry letters (09.12.2010)
Published in ACS medicinal chemistry letters (09.12.2010)
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Synthesis of 2,3-unsaturated glycopyranosides by ferrier rearrangement in FeCl3 based ionic liquid
TILVE, Rutuja D, VARUGHESE ALEXANDER, M, KHANDEKAR, Amit C, SAMANT, Sriniwas D, KANETKAR, Vinod R
Published in Journal of molecular catalysis. A, Chemical (01.12.2004)
Published in Journal of molecular catalysis. A, Chemical (01.12.2004)
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Conference Proceeding
Journal Article
Subtle Chemical Changes Cross the Boundary between Agonist and Antagonist: New A 3 Adenosine Receptor Homology Models and Structural Network Analysis Can Predict This Boundary
Lee, Yoonji, Hou, Xiyan, Lee, Jin Hee, Nayak, Akshata, Alexander, Varughese, Sharma, Pankaz K, Chang, Hyerim, Phan, Khai, Gao, Zhan-Guo, Jacobson, Kenneth A, Choi, Sun, Jeong, Lak Shin
Published in Journal of medicinal chemistry (09.09.2021)
Published in Journal of medicinal chemistry (09.09.2021)
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Journal Article
Subtle Chemical Changes Cross the Boundary between Agonist and Antagonist: New A3 Adenosine Receptor Homology Models and Structural Network Analysis Can Predict This Boundary
Lee, Yoonji, Hou, Xiyan, Lee, Jin Hee, Nayak, Akshata, Alexander, Varughese, Sharma, Pankaz K, Chang, Hyerim, Phan, Khai, Gao, Zhan-Guo, Jacobson, Kenneth A, Choi, Sun, Jeong, Lak Shin
Published in Journal of medicinal chemistry (09.09.2021)
Published in Journal of medicinal chemistry (09.09.2021)
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Journal Article
Synthesis and biological evaluation of 20-substituted-40- selenoribofuranosyl pyrimidines as antitumor agents
Varughese Alexander, 송자영, 유진하, 최정희, 김진희, 이상국, 최원준, 정낙신
Published in Archives of pharmacal research (01.06.2015)
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Published in Archives of pharmacal research (01.06.2015)
Journal Article
Fluorocyclopentenyl-cytosine with Broad Spectrum and Potent Antitumor Activity
Choi, Won Jun, Chung, Hwa-Jin, Chandra, Girish, Alexander, Varughese, Zhao, Long Xuan, Lee, Hyuk Woo, Nayak, Akshata, Majik, Mahesh S, Kim, Hea Ok, Kim, Jin-Hee, Lee, Young B, Ahn, Chang H, Lee, Sang Kook, Jeong, Lak Shin
Published in Journal of medicinal chemistry (10.05.2012)
Published in Journal of medicinal chemistry (10.05.2012)
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Journal Article
Structure–Activity Relationships of Truncated C2- or C8-Substituted Adenosine Derivatives as Dual Acting A 2A and A 3 Adenosine Receptor Ligands
Hou, Xiyan, Majik, Mahesh S., Kim, Kyunglim, Pyee, Yuna, Lee, Yoonji, Alexander, Varughese, Chung, Hwa-Jin, Lee, Hyuk Woo, Chandra, Girish, Lee, Jin Hee, Park, Seul-gi, Choi, Won Jun, Kim, Hea Ok, Phan, Khai, Gao, Zhan-Guo, Jacobson, Kenneth A., Choi, Sun, Lee, Sang Kook, Jeong, Lak Shin
Published in Journal of medicinal chemistry (12.01.2012)
Published in Journal of medicinal chemistry (12.01.2012)
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Journal Article
Structure-Activity Relationships of Truncated C2- or C8-Substituted Adenosine Derivatives as Dual Acting A(2A) and A(3) Adenosine Receptor Ligands
Hou, Xiyan, Majik, Mahesh S., Kim, Kyunglim, Pyee, Yuna, Lee, Yoonji, Alexander, Varughese, Chung, Hwa-Jin, Lee, Hyuk Woo, Chandra, Girish, Lee, Jin Hee, Park, Seul-gi, Choi, Won Jun, Kim, Hea Ok, Phan, Khai, Gao, Zhan-Guo, Jacobson, Kenneth A., Choi, Sun, Lee, Sang Kook, Jeong, Lak Shin
Published in Journal of medicinal chemistry (12.01.2012)
Published in Journal of medicinal chemistry (12.01.2012)
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Journal Article
2'-플루오로-6'-메틸렌-탄소환식 아데노신(FMCA) 및 2'-플루오로-6'-메틸렌-탄소환식 구아노신(FMCG)의 합성
SINGH UMA SHARAN, CHU CHUNG K, MISHRA RAM C, MULAMOOTTIL VARUGHESE ALEXANDER
Year of Publication 18.12.2018
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Year of Publication 18.12.2018
Patent
A simpler and greener protocol for the preparation of β-acetylamino ketones by a one-pot reaction of aryl aldehydes, enolisable ketones, acetyl chloride and acetonitrile in the presence of zeolite Hβ as a reusable catalyst
Bhat, Ramakrishna P., Raje, Vivek P., Alexander, Varughese M., Patil, Sachin B., Samant, Shriniwas D.
Published in Tetrahedron letters (11.07.2005)
Published in Tetrahedron letters (11.07.2005)
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Journal Article
A New DNA Building Block, 4′-Selenothymidine: Synthesis and Modification to 4′-Seleno-AZT as a Potential Anti-HIV Agent
Alexander, Varughese, Choi, Won Jun, Chun, Jeongha, Kim, Hea Ok, Jeon, Ji Hye, Tosh, Dilip K, Lee, Hyuk Woo, Chandra, Girish, Choi, Jungwon, Jeong, Lak Shin
Published in Organic letters (21.05.2010)
Published in Organic letters (21.05.2010)
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Journal Article
Iodination of activated arenes using silfen: an improved protocol
Tilve, Rutuja D., Alexander, Varughese M., Khadilkar, Bhushan M.
Published in Tetrahedron letters (16.12.2002)
Published in Tetrahedron letters (16.12.2002)
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Journal Article