Islatravir Case Study for Enhanced Screening of Thermodynamically Stable Crystalline Anhydrate Phases in Pharmaceutical Process Development by Hot Melt Extrusion
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Published in Molecular pharmaceutics (03.08.2020)
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Development of a Large Scale Asymmetric Synthesis of the Glucocorticoid Agonist BI 653048 BS H3PO4
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Crystallization Process Development for the Final Step of the Biocatalytic Synthesis of Islatravir: Comprehensive Crystal Engineering for a Low-Dose Drug
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A Robust Process for an mGluR5 Negative Allosteric Modulator: Difluoromethylation and Sonogashira Coupling on Large Scale
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Development of a Large Scale Asymmetric Synthesis of the Glucocorticoid Agonist BI 653048 BS H 3 PO 4
Reeves, Jonathan T., Fandrick, Daniel R., Tan, Zhulin, Song, Jinhua J., Rodriguez, Sonia, Qu, Bo, Kim, Soojin, Niemeier, Oliver, Li, Zhibin, Byrne, Denis, Campbell, Scot, Chitroda, Ashish, DeCroos, Phil, Fachinger, Thomas, Fuchs, Victor, Gonnella, Nina C., Grinberg, Nelu, Haddad, Nizar, Jäger, Burkhard, Lee, Heewon, Lorenz, Jon C., Ma, Shengli, Narayanan, Bikshandarkoil A., Nummy, Larry J., Premasiri, Ajith, Roschangar, Frank, Sarvestani, Max, Shen, Sherry, Spinelli, Earl, Sun, Xiufeng, Varsolona, Richard J., Yee, Nathan, Brenner, Michael, Senanayake, Chris H.
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Published in Journal of organic chemistry (19.04.2013)
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