The selective 5-HT1A receptor agonist, NLX-112, exerts anti-dyskinetic and anti-parkinsonian-like effects in MPTP-treated marmosets
Fisher, Ria, Hikima, Atsuko, Morris, Rebecca, Jackson, Michael J., Rose, Sarah, Varney, Mark A., Depoortere, Ronan, Newman-Tancredi, Adrian
Published in Neuropharmacology (01.05.2020)
Published in Neuropharmacology (01.05.2020)
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Journal Article
The novel 5-HT1A receptor agonist, NLX-112 reduces l-DOPA-induced abnormal involuntary movements in rat: A chronic administration study with microdialysis measurements
McCreary, Andrew C., Varney, Mark A., Newman-Tancredi, Adrian
Published in Neuropharmacology (01.06.2016)
Published in Neuropharmacology (01.06.2016)
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Journal Article
Pharmacodynamic, pharmacokinetic and rat brain receptor occupancy profile of NLX-112, a highly selective 5-HT1A receptor biased agonist
Depoortère, Ronan Y., McCreary, Andrew C., Vidal, Benjamin, Varney, Mark A., Zimmer, Luc, Newman-Tancredi, Adrian
Published in Naunyn-Schmiedeberg's archives of pharmacology (03.08.2024)
Published in Naunyn-Schmiedeberg's archives of pharmacology (03.08.2024)
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Effects of the Serotonin 5-HT1A Receptor Biased Agonists, F13714 and F15599, on Striatal Neurotransmitter Levels Following l-DOPA Administration in Hemi-Parkinsonian Rats
Newman-Tancredi, Adrian, Varney, Mark A., McCreary, Andrew C.
Published in Neurochemical research (01.05.2018)
Published in Neurochemical research (01.05.2018)
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Journal Article
Antinociceptive, antiallodynic and antihyperalgesic effects of the 5-HT1A receptor selective agonist, NLX-112 in mouse models of pain
Sałat, Kinga, Kołaczkowski, Marcin, Furgała, Anna, Rojek, Adriana, Śniecikowska, Joanna, Varney, Mark A., Newman-Tancredi, Adrian
Published in Neuropharmacology (01.10.2017)
Published in Neuropharmacology (01.10.2017)
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Journal Article
Identification of the 5-HT1A serotonin receptor as a novel therapeutic target in a C. elegans model of Machado-Joseph disease
Pereira-Sousa, Joana, Ferreira-Lomba, Bruna, Bellver-Sanchis, Aina, Vilasboas-Campos, Daniela, Fernandes, Jorge H., Costa, Marta D., Varney, Mark A., Newman-Tancredi, Adrian, Maciel, Patrícia, Teixeira-Castro, Andreia
Published in Neurobiology of disease (01.05.2021)
Published in Neurobiology of disease (01.05.2021)
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Journal Article
The selective 5-HT1A receptor agonist, NLX-112, overcomes tetrabenazine-induced catalepsy and depression-like behavior in the rat
Jastrzębska-Więsek, Magdalena, Wesołowska, Anna, Kołaczkowski, Marcin, Varney, Mark A, Newman-Tancredi, Adrian, Depoortere, RonanY
Published in Behavioural pharmacology (01.08.2022)
Published in Behavioural pharmacology (01.08.2022)
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Journal Article
Cortical 5-hydroxytryptamine 1A receptor biased agonist, NLX-101, displays rapid-acting antidepressant-like properties in the rat chronic mild stress model
Depoortère, Ronan, Papp, Mariusz, Gruca, Piotr, Lason-Tyburkiewicz, Magdalena, Niemczyk, Monika, Varney, Mark A, Newman-Tancredi, Adrian
Published in Journal of psychopharmacology (Oxford) (01.11.2019)
Published in Journal of psychopharmacology (Oxford) (01.11.2019)
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Journal Article
Activity of Serotonin 5‑HT1A Receptor Biased Agonists in Rat: Anxiolytic and Antidepressant-like properties
Jastrzębska-Więsek, Magdalena, Partyka, Anna, Rychtyk, Joanna, Śniecikowska, Joanna, Kołaczkowski, Marcin, Wesołowska, Anna, Varney, Mark A, Newman-Tancredi, Adrian
Published in ACS chemical neuroscience (16.05.2018)
Published in ACS chemical neuroscience (16.05.2018)
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Journal Article
Dissecting the contribution of 5-HT1A auto- and heteroreceptors in sucrose overconsumption in mice
Beecher, Kate, Wang, Joshua, Chehrehasa, Fatemeh, Depoortere, Ronan, Varney, Mark A., Newman-Tancredi, Adrian, Bartlett, Selena E., Belmer, Arnauld
Published in Biomedicine & pharmacotherapy (01.04.2022)
Published in Biomedicine & pharmacotherapy (01.04.2022)
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Journal Article
Novel Aryloxyethyl Derivatives of 1‑(1-Benzoylpiperidin-4-yl)methanamine as the Extracellular Regulated Kinases 1/2 (ERK1/2) Phosphorylation-Preferring Serotonin 5‑HT1A Receptor-Biased Agonists with Robust Antidepressant-like Activity
Sniecikowska, Joanna, Gluch-Lutwin, Monika, Bucki, Adam, Więckowska, Anna, Siwek, Agata, Jastrzebska-Wiesek, Magdalena, Partyka, Anna, Wilczyńska, Daria, Pytka, Karolina, Pociecha, Krzysztof, Cios, Agnieszka, Wyska, Elżbieta, Wesołowska, Anna, Pawłowski, Maciej, Varney, Mark A, Newman-Tancredi, Adrian, Kolaczkowski, Marcin
Published in Journal of medicinal chemistry (14.03.2019)
Published in Journal of medicinal chemistry (14.03.2019)
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Journal Article
Activity of Serotonin 5-HT 1A Receptor Biased Agonists in Rat: Anxiolytic and Antidepressant-like properties
Jastrzębska-Więsek, Magdalena, Partyka, Anna, Rychtyk, Joanna, Śniecikowska, Joanna, Kołaczkowski, Marcin, Wesołowska, Anna, Varney, Mark A, Newman-Tancredi, Adrian
Published in ACS chemical neuroscience (16.05.2018)
Published in ACS chemical neuroscience (16.05.2018)
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Journal Article
Enhanced aggressive phenotype of Tph2 knockout rats is associated with diminished 5-HT1A receptor sensitivity
Peeters, Deborah G.A., de Boer, Sietse F., Terneusen, Anneke, Newman-Tancredi, Adrian, Varney, Mark A., Verkes, Robbert-Jan, Homberg, Judith R.
Published in Neuropharmacology (15.07.2019)
Published in Neuropharmacology (15.07.2019)
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Differential distribution of voltage-gated calcium channel alpha-2 delta (α2δ) subunit mRNA-containing cells in the rat central nervous system and the dorsal root ganglia
Cole, Rebecca L., Lechner, Sandra M., Williams, Mark E., Prodanovich, Pat, Bleicher, Leo, Varney, Mark A., Gu, Guibao
Published in Journal of comparative neurology (1911) (24.10.2005)
Published in Journal of comparative neurology (1911) (24.10.2005)
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Journal Article
Novel Aryloxyethyl Derivatives of 1-(1-Benzoylpiperidin-4-yl)methanamine as the Extracellular Regulated Kinases 1/2 (ERK1/2) Phosphorylation-Preferring Serotonin 5-HT 1A Receptor-Biased Agonists with Robust Antidepressant-like Activity
Sniecikowska, Joanna, Gluch-Lutwin, Monika, Bucki, Adam, Więckowska, Anna, Siwek, Agata, Jastrzebska-Wiesek, Magdalena, Partyka, Anna, Wilczyńska, Daria, Pytka, Karolina, Pociecha, Krzysztof, Cios, Agnieszka, Wyska, Elżbieta, Wesołowska, Anna, Pawłowski, Maciej, Varney, Mark A, Newman-Tancredi, Adrian, Kolaczkowski, Marcin
Published in Journal of medicinal chemistry (14.03.2019)
Published in Journal of medicinal chemistry (14.03.2019)
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Journal Article
3-[(2-Methyl-1,3-thiazol-4-yl)ethynyl]- pyridine: A Potent and Highly Selective Metabotropic Glutamate Subtype 5 Receptor Antagonist with Anxiolytic Activity
Cosford, Nicholas D. P, Tehrani, Lida, Roppe, Jeffrey, Schweiger, Edwin, Smith, Nicholas D, Anderson, Jeffrey, Bristow, Linda, Brodkin, Jesse, Jiang, Xiaohui, McDonald, Ian, Rao, Sara, Washburn, Mark, Varney, Mark A
Published in Journal of medicinal chemistry (16.01.2003)
Published in Journal of medicinal chemistry (16.01.2003)
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Journal Article
Structural, Kinetic, and Pharmacodynamic Mechanisms of d‑Amino Acid Oxidase Inhibition by Small Molecules
Hopkins, Seth C, Heffernan, Michele L. R, Saraswat, Lakshmi D, Bowen, Carrie A, Melnick, Laurence, Hardy, Larry W, Orsini, Michael A, Allen, Michael S, Koch, Patrick, Spear, Kerry L, Foglesong, Robert J, Soukri, Mustapha, Chytil, Milan, Fang, Q. Kevin, Jones, Steven W, Varney, Mark A, Panatier, Aude, Oliet, Stephane H. R, Pollegioni, Loredano, Piubelli, Luciano, Molla, Gianluca, Nardini, Marco, Large, Thomas H
Published in Journal of medicinal chemistry (09.05.2013)
Published in Journal of medicinal chemistry (09.05.2013)
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Pharmacodynamic effects of a D-amino acid oxidase inhibitor indicate a spinal site of action in rat models of neuropathic pain
Hopkins, Seth C, Zhao, Fei-Yue, Bowen, Carrie A, Fang, Xin, Wei, Haifeng, Heffernan, Michele L R, Spear, Kerry L, Spanswick, David C, Varney, Mark A, Large, Thomas H
Published in The Journal of pharmacology and experimental therapeutics (01.06.2013)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2013)
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