The 5-HT1B receptor - a potential target for antidepressant treatment
Tiger, Mikael, Varnäs, Katarina, Okubo, Yoshiro, Lundberg, Johan
Published in Psychopharmacology (01.05.2018)
Published in Psychopharmacology (01.05.2018)
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Discovery and Evaluation of Clinical Candidate AZD3759, a Potent, Oral Active, Central Nervous System-Penetrant, Epidermal Growth Factor Receptor Tyrosine Kinase Inhibitor
Zeng, Qingbei, Wang, Jiabing, Cheng, Ziqiang, Chen, Kan, Johnström, Peter, Varnäs, Katarina, Li, David Yunzhi, Yang, Zhen Fan, Zhang, Xiaolin
Published in Journal of medicinal chemistry (22.10.2015)
Published in Journal of medicinal chemistry (22.10.2015)
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Effect of the myeloperoxidase inhibitor AZD3241 on microglia: a PET study in Parkinson's disease
Jucaite, Aurelija, Svenningsson, Per, Rinne, Juha O, Cselényi, Zsolt, Varnäs, Katarina, Johnström, Peter, Amini, Nahid, Kirjavainen, Anna, Helin, Semi, Minkwitz, Margaret, Kugler, Alan R, Posener, Joel A, Budd, Samantha, Halldin, Christer, Varrone, Andrea, Farde, Lars
Published in Brain (London, England : 1878) (01.09.2015)
Published in Brain (London, England : 1878) (01.09.2015)
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Preclinical Comparison of the Blood-brain barrier Permeability of Osimertinib with Other EGFR TKIs
Colclough, Nicola, Chen, Kan, Johnström, Peter, Strittmatter, Nicole, Yan, Yumei, Wrigley, Gail L, Schou, Magnus, Goodwin, Richard, Varnäs, Katarina, Adua, Sally J, Zhao, Minghui, Nguyen, Don X, Maglennon, Gareth, Barton, Peter, Atkinson, James, Zhang, Lin, Janefeldt, Annika, Wilson, Joanne, Smith, Aaron, Takano, Akihiro, Arakawa, Ryosuke, Kondrashov, Mikhail, Malmquist, Jonas, Revunov, Evgeny, Vazquez-Romero, Ana, Moein, Mohammad Mahdi, Windhorst, Albert D, Karp, Natasha A, Finlay, M Raymond V, Ward, Richard A, Yates, James W T, Smith, Paul D, Farde, Lars, Cheng, Zack, Cross, Darren A E
Published in Clinical cancer research (01.01.2021)
Published in Clinical cancer research (01.01.2021)
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A positron emission tomography study of the serotonin1B receptor effect of electroconvulsive therapy for severe major depressive episodes
Tiger, Mikael, Gärde, Martin, Tateno, Amane, Matheson, Granville J, Sakayori, Takeshi, Nogami, Tsuyoshi, Moriya, Hiroki, Varnäs, Katarina, Arakawa, Ryosuke, Okubo, Yoshiro
Published in Journal of affective disorders (01.11.2021)
Published in Journal of affective disorders (01.11.2021)
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Synthesis and preclinical evaluation of [18F]FSL25.1188, a reversible PET radioligand for monoamine oxidase-B
Dahl, Kenneth, Bernard-Gauthier, Vadim, Nag, Sangram, Varnäs, Katarina, Narayanaswami, Vidya, Mahdi Moein, Mohammad, Arakawa, Ryosuke, Vasdev, Neil, Halldin, Christer
Published in Bioorganic & medicinal chemistry letters (01.07.2019)
Published in Bioorganic & medicinal chemistry letters (01.07.2019)
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Synthesis and Autoradiography of Novel F‑18 Labeled Reversible Radioligands for Detection of Monoamine Oxidase B
Nag, Sangram, Jia, Zhisheng, Svedberg, Marie, Jackson, Alex, Ahmad, Rabia, Luthra, Sajinder, Varnäs, Katarina, Farde, Lars, Halldin, Christer
Published in ACS chemical neuroscience (16.12.2020)
Published in ACS chemical neuroscience (16.12.2020)
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Regional thinning of the cerebral cortex in schizophrenia: Effects of diagnosis, age and antipsychotic medication
Nesvåg, Ragnar, Lawyer, Glenn, Varnäs, Katarina, Fjell, Anders M, Walhovd, Kristine B, Frigessi, Arnoldo, Jönsson, Erik G, Agartz, Ingrid
Published in Schizophrenia research (01.01.2008)
Published in Schizophrenia research (01.01.2008)
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The metabotropic glutamate receptor 5 radioligand [11C]AZD9272 identifies unique binding sites in primate brain
Varnäs, Katarina, Juréus, Anders, Finnema, Sjoerd J., Johnström, Peter, Raboisson, Patrick, Amini, Nahid, Takano, Akihiro, Stepanov, Vladimir, Halldin, Christer, Farde, Lars
Published in Neuropharmacology (01.06.2018)
Published in Neuropharmacology (01.06.2018)
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The brain-penetrant clinical ATM inhibitor AZD1390 radiosensitizes and improves survival of preclinical brain tumor models
Durant, Stephen T, Zheng, Li, Wang, Yingchun, Chen, Kan, Zhang, Lingli, Zhang, Tianwei, Yang, Zhenfan, Riches, Lucy, Trinidad, Antonio G, Fok, Jacqueline H L, Hunt, Tom, Pike, Kurt G, Wilson, Joanne, Smith, Aaron, Colclough, Nicola, Reddy, Venkatesh Pilla, Sykes, Andrew, Janefeldt, Annika, Johnström, Peter, Varnäs, Katarina, Takano, Akihiro, Ling, Stephanie, Orme, Jonathan, Stott, Jonathan, Roberts, Caroline, Barrett, Ian, Jones, Gemma, Roudier, Martine, Pierce, Andrew, Allen, Jasmine, Kahn, Jenna, Sule, Amrita, Karlin, Jeremy, Cronin, Anna, Chapman, Melissa, Valerie, Kristoffer, Illingworth, Ruth, Pass, Martin
Published in Science advances (01.06.2018)
Published in Science advances (01.06.2018)
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Large Variation in Brain Exposure of Reference CNS Drugs: a PET Study in Nonhuman Primates
Schou, Magnus, Varnäs, Katarina, Lundquist, Stefan, Nakao, Ryuji, Amini, Nahid, Takano, Akihiro, Finnema, Sjoerd J., Halldin, Christer, Farde, Lars
Published in The international journal of neuropsychopharmacology (01.09.2015)
Published in The international journal of neuropsychopharmacology (01.09.2015)
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[C-11]CHDI-626, a PET Tracer Candidate for Imaging Mutant Huntingtin Aggregates with Reduced Binding to AD Pathological Proteins
Liu, Longbin, Johnson, Peter D., Prime, Michael E., Khetarpal, Vinod, Lee, Matthew R., Brown, Christopher J., Chen, Xuemei, Clark-Frew, Daniel, Coe, Samuel, Conlon, Mike, Davis, Randall, Ensor, Samantha, Esposito, Simone, Moren, Anton Forsberg, Gai, Xinjie, Green, Samantha, Greenaway, Catherine, Haber, James, Halldin, Christer, Hayes, Sarah, Herbst, Todd, Herrmann, Frank, He-mann, Manuela, Hsai, Ming Min, Kotey, Adrian, Mangette, John E., Mills, Matthew R., Monteagudo, Edith, Nag, Sangram, Nibbio, Martina, Orsatti, Laura, Schaertl, Sabine, Scheich, Christoph, Sproston, Joanne, Stepanov, Vladimir, Varnas, Katarina, Varrone, Andrea, Wityak, John, Mrzljak, Ladislav, Munoz-Sanjuan, Ignacio, Bard, Jonathan A., Dominguez, Celia
Published in Journal of medicinal chemistry (26.08.2021)
Published in Journal of medicinal chemistry (26.08.2021)
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Development of rapid multistep carbon-11 radiosynthesis of the myeloperoxidase inhibitor AZD3241 to assess brain exposure by PET microdosing
Johnström, Peter, Bergman, Linda, Varnäs, Katarina, Malmquist, Jonas, Halldin, Christer, Farde, Lars
Published in Nuclear medicine and biology (01.06.2015)
Published in Nuclear medicine and biology (01.06.2015)
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A positron emission tomography study in healthy volunteers to estimate mGluR5 receptor occupancy of AZD2066 — Estimating occupancy in the absence of a reference region
Kågedal, Matts, Cselényi, Zsolt, Nyberg, Svante, Raboisson, Patrick, Ståhle, Lars, Stenkrona, Per, Varnäs, Katarina, Halldin, Christer, Hooker, Andrew C., Karlsson, Mats O.
Published in NeuroImage (Orlando, Fla.) (15.11.2013)
Published in NeuroImage (Orlando, Fla.) (15.11.2013)
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Quantitative Analysis of [11C]AZ10419369 Binding to 5-HT1B Receptors in Human Brain
Varnäs, Katarina, Nyberg, Svante, Halldin, Christer, Varrone, Andrea, Takano, Akihiro, Karlsson, Per, Andersson, Jan, McCarthy, Dennis, Smith, Mark, Pierson, M Edward, Söderström, Johan, Farde, Lars
Published in Journal of cerebral blood flow and metabolism (01.01.2011)
Published in Journal of cerebral blood flow and metabolism (01.01.2011)
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Development of [Carbonyl-11C]AZ13198083, a Novel Histamine Type‑3 Receptor Radioligand with Favorable Kinetics
Dahl, Kenneth, Nakao, Ryuji, Amini, Nahid, Moein, Mohammad Mahdi, Finnema, Sjoerd, Malmquist, Jonas, Varnäs, Katarina, Schou, Magnus
Published in ACS chemical neuroscience (16.05.2018)
Published in ACS chemical neuroscience (16.05.2018)
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Altered striatal dopamine levels in Parkinson’s disease VPS35 D620N mutant transgenic aged mice
Vanan, Sarivin, Zeng, Xiaoxia, Chia, Sook Yoong, Varnäs, Katarina, Jiang, Mei, Zhang, Ke, Saw, Wuan Ting, Padmanabhan, Parasuraman, Yu, Wei-Ping, Zhou, Zhi-Dong, Halldin, Christer, Gulyás, Balázs, Tan, Eng-King, Zeng, Li
Published in Molecular brain (01.12.2020)
Published in Molecular brain (01.12.2020)
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