Safety, Tolerability, and Pharmacokinetics of JNJ-1802, a Pan-serotype Dengue Direct Antiviral Small Molecule, in a Phase 1, Double-Blind, Randomized, Dose-Escalation Study in Healthy Volunteers
Ackaert, Oliver, Vanhoutte, Frédéric, Verpoorten, Nathalie, Buelens, Annemie, Lachau-Durand, Sophie, Lammens, Lieve, Hoetelmans, Richard, Van Loock, Marnix, Herrera-Taracena, Guillermo
Published in Clinical infectious diseases (18.09.2023)
Published in Clinical infectious diseases (18.09.2023)
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Journal Article
Efficacy, Safety, Pharmacokinetics, and Pharmacodynamics of Filgotinib, a Selective JAK‐1 Inhibitor, After Short‐Term Treatment of Rheumatoid Arthritis: Results of Two Randomized Phase IIa Trials
Vanhoutte, Frédéric, Mazur, Minodora, Voloshyn, Oleksandr, Stanislavchuk, Mykola, Van der Aa, Annegret, Namour, Florence, Galien, René, Meuleners, Luc, van 't Klooster, Gerben
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.10.2017)
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.10.2017)
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Journal Article
Pharmacokinetics and Pharmacodynamics of Garetosmab (Anti‐Activin A): Results From a First‐in‐Human Phase 1 Study
Vanhoutte, Frédéric, Liang, Su, Ruddy, Marcella, Zhao, An, Drewery, Tiera, Wang, Yuhuan, DelGizzi, Richard, Forleo‐Neto, Eduardo, Rajadhyaksha, Manoj, Herman, Gary, Davis, John D.
Published in Journal of clinical pharmacology (01.11.2020)
Published in Journal of clinical pharmacology (01.11.2020)
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Journal Article
Evaluating the pharmacokinetics of beclometasone dipropionate/formoterol fumarate/glycopyrronium bromide delivered via pressurised metered-dose inhaler using a low global warming potential propellant
Rony, François, Cortellini, Mauro, Guasconi, Alessandro, Mathews, Kusum S., Piccinno, Annalisa, Poli, Gianluigi, Vanhoutte, Frédéric, Klein, Jelle
Published in Pulmonary pharmacology & therapeutics (01.06.2024)
Published in Pulmonary pharmacology & therapeutics (01.06.2024)
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Journal Article
Safety, pharmacokinetics and pharmacodynamics of GLPG0974, a potent and selective FFA2 antagonist, in healthy male subjects
Namour, Florence, Galien, René, Van Kaem, Tim, Van der Aa, Annegret, Vanhoutte, Frédéric, Beetens, Johan, Klooster, Gerben
Published in British journal of clinical pharmacology (01.07.2016)
Published in British journal of clinical pharmacology (01.07.2016)
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Journal Article
Randomized study of the effect of gadopiclenol, a new gadolinium‐based contrast agent, on the QTc interval in healthy subjects
Funck‐Brentano, Christian, Felices, Mathieu, Le Fur, Nathalie, Dubourdieu, Corinne, Desché, Pierre, Vanhoutte, Frédéric, Voiriot, Pascal
Published in British journal of clinical pharmacology (01.11.2020)
Published in British journal of clinical pharmacology (01.11.2020)
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Journal Article
Orally Bioavailable Macrocyclic Peptide That Inhibits Binding of PCSK9 to the Low Density Lipoprotein Receptor
Johns, Douglas G, Campeau, Louis-Charles, Banka, Puja, Bautmans, An, Bueters, Tjerk, Bianchi, Elisabetta, Branca, Danila, Bulger, Paul G, Crevecoeur, Inne, Ding, Fa-Xiang, Garbaccio, Robert M, Guetschow, Erik D, Guo, Yan, Ha, Sookhee N, Johnston, Jennifer M, Josien, Hubert, Kauh, Eunkyung A, Koeplinger, Kenneth A, Kuethe, Jeffrey T, Lai, Eseng, Lanning, Christine L, Lee, Anita Y H, Li, Li, Nair, Anilkumar G, O'Neill, Edward A, Stoch, S Aubrey, Thaisrivongs, David A, Tucker, Thomas J, Vachal, Petr, van Dyck, Kristien, Vanhoutte, Frederic P, Volckaert, Bram, Wolford, Dennis G, Xu, Andy, Zhao, Tian, Zhou, Dan, Zhou, Susan, Zhu, Xiaohong, Zokian, Hratch J, Walji, Abbas M, Wood, Harold B
Published in Circulation (New York, N.Y.) (11.07.2023)
Published in Circulation (New York, N.Y.) (11.07.2023)
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Journal Article
Safety, Pharmacokinetics, and Antiviral Activity of AT-527, a Novel Purine Nucleotide Prodrug, in Hepatitis C Virus-Infected Subjects with or without Cirrhosis
Berliba, Elina, Bogus, Maxim, Vanhoutte, Frédéric, Berghmans, Pieter-Jan, Good, Steven S, Moussa, Adel, Pietropaolo, Keith, Murphy, Robert L, Zhou, Xiao-Jian, Sommadossi, Jean-Pierre
Published in Antimicrobial agents and chemotherapy (01.12.2019)
Published in Antimicrobial agents and chemotherapy (01.12.2019)
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Journal Article
Pharmacokinetics and pharmacodynamics of mibavademab (a leptin receptor agonist): Results from a first‐in‐human phase I study
Gewitz, Andrew, Mendell, Jeanne, Wang, Yuhuan, Harris, Charles, Olenchock, Benjamin A., Podgrabinska, Simona, Zheng, Wenjun, Zhao, An, Pan, Hao, Vanhoutte, Frédéric, Davis, John D.
Published in Clinical and translational science (01.04.2024)
Published in Clinical and translational science (01.04.2024)
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Journal Article
Safety, Tolerability, and Pharmacokinetics of Single Ascending Doses of ELX‐02, a Potential Treatment for Genetic Disorders Caused by Nonsense Mutations, in Healthy Volunteers
Leubitz, Andi, Frydman‐Marom, Anat, Sharpe, Neal, Duzer, John, Campbell, Kathleen C.M., Vanhoutte, Frédéric
Published in Clinical pharmacology in drug development (01.11.2019)
Published in Clinical pharmacology in drug development (01.11.2019)
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Journal Article
Safety and immunogenicity of the measles vector-based SARS-CoV-2 vaccine candidate, V591, in adults: results from a phase 1/2 randomised, double-blind, placebo-controlled, dose-ranging trial
Vanhoutte, Frédéric, Liu, Wen, Wiedmann, Richard T., Haspeslagh, Liesbeth, Cao, Xin, Boundy, Keith, Aliprantis, Antonios, Davila, Michelle, Hartzel, Jonathan, Li, Jianing, McGuire, Mac, Ramsauer, Katrin, Tomberger, Yvonne, Tschismarov, Roland, Brown, Deborah D., Xu, Weifeng, Sachs, Jeffrey R., Russell, Kevin, Stoch, S. Aubrey, Lai, Eseng
Published in EBioMedicine (01.01.2022)
Published in EBioMedicine (01.01.2022)
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Journal Article
A dose escalating phase I study of GLPG0187, a broad spectrum integrin receptor antagonist, in adult patients with progressive high-grade glioma and other advanced solid malignancies
Cirkel, Geert A., Kerklaan, Bojana Milojkovic, Vanhoutte, Frédéric, der Aa, Annegret Van, Lorenzon, Giocondo, Namour, Florence, Pujuguet, Philippe, Darquenne, Sophie, de Vos, Filip Y. F., Snijders, Tom J., Voest, Emile E., Schellens, Jan H. M., Lolkema, Martijn P.
Published in Investigational new drugs (01.04.2016)
Published in Investigational new drugs (01.04.2016)
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Journal Article
Oral administration of GLPG0259, an inhibitor of MAPKAPK5, a new target for the treatment of rheumatoid arthritis: a phase II, randomised, double-blind, placebo-controlled, multicentre trial
Westhovens, René, Keyser, Filip De, Rekalov, Dmytro, Nasonov, Evgeny L, Beetens, Johan, Van der Aa, Annegret, Wigerinck, Piet, Namour, Florence, Vanhoutte, Frédéric, Durez, Patrick
Published in Annals of the rheumatic diseases (01.05.2013)
Published in Annals of the rheumatic diseases (01.05.2013)
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Journal Article
188 Exploration of GLPG0634, the First Selective JAK1 Inhibitor, in Inflammatory Bowel Disease Is Supported by Early Clinical Results and Mouse DSS-Colitis Data
Galien, Rene, Merciris, Didier, Vanhoutte, Frédéric P, Delachaume, Carole, Namour, Florence S, Vayssière, Béatrice, Van der Aa, Annegret, Brys, Reginald, van't Klooster, Gerben A
Published in Gastroenterology (New York, N.Y. 1943) (01.05.2014)
Published in Gastroenterology (New York, N.Y. 1943) (01.05.2014)
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Journal Article
Mo1234 The FFA2 Antagonist GLPG0974: A Promising Approach to Treat Neutrophil-Driven Inflammation
Vanhoutte, Frédéric P, Namour, Florence S, Dupont, Sonia, Pizzonero, Mathieu, De Vos, Steve, Sanière, Laurent, van der Aa, Annegret, Beetens, Johan, van 't Klooster, Gerben
Published in Gastroenterology (New York, N.Y. 1943) (01.05.2014)
Published in Gastroenterology (New York, N.Y. 1943) (01.05.2014)
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Journal Article
A Randomized, Double‐Blind, Placebo‐Controlled, Multiple Dose Escalation Study to Evaluate the Safety and Pharmacokinetics of ELX‐02 in Healthy Subjects
Leubitz, Andi, Vanhoutte, Frederic, Hu, Ming‐yi, Porter, Kaela, Gordon, Efrat, Tencer, Kathleen, Campbell, Kathleen, Banks, Kate, Haverty, Tom
Published in Clinical pharmacology in drug development (01.08.2021)
Published in Clinical pharmacology in drug development (01.08.2021)
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Journal Article
Pharmacokinetics, Safety, and Tolerability of GLPG0259, a Mitogen-Activated Protein Kinase-Activated Protein Kinase 5 (MAPKAPK5) Inhibitor, Given as Single and Multiple Doses to Healthy Male Subjects
Namour, Florence, Vanhoutte, Frédéric P., Beetens, Johan, Blockhuys, Stan, Weer, Marc De, Wigerinck, Piet
Published in Drugs in R&D (01.09.2012)
Published in Drugs in R&D (01.09.2012)
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Journal Article
Correlations between factors determining the pharmacokinetics and antiviral activity of HIV-1 non-nucleoside reverse transcriptase inhibitors of the diaryltriazine and diarylpyrimidine classes of compounds
Lewi, Paul, Arnold, Eddy, Andries, Koen, Bohets, Hilde, Borghys, Herman, Clark, Arthur, Daeyaert, Frits, Das, Kalyan, de Béthune, Marie-Pierre, de Jonge, Marc, Heeres, Jan, Koymans, Luc, Leempoels, Jos, Peeters, Jef, Timmerman, Philip, Van den Broeck, Walter, Vanhoutte, Frédéric, Van't Klooster, Gerben, Vinkers, Maarten, Volovik, Yulia, Janssen, Paul A J
Published in Drugs in R&D (2004)
Published in Drugs in R&D (2004)
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Journal Article
METHODS FOR THE TREATMENT OF INFLAMMATORY DISORDERS
WIGERINCK PIET TOM BERT PAUL, VANHOUTTE FREDERIC PAUL, VAN 'T KLOOSTER GERBEN ALBERT ELEUTHERIUS
Year of Publication 06.12.2017
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Year of Publication 06.12.2017
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