Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1
Hall, Adrian, Abendroth, Jan, Bolejack, Madison J., Ceska, Tom, Dell’Aiera, Sylvie, Ellis, Victoria, Fox, David, François, Cyril, Muruthi, Muigai M., Prével, Camille, Poullennec, Karine, Romanov, Sergei, Valade, Anne, Vanbellinghen, Alain, Yano, Jason, Geraerts, Martine
Published in ACS medicinal chemistry letters (14.07.2022)
Published in ACS medicinal chemistry letters (14.07.2022)
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Journal Article
Lead Optimization of Thiazolo[5,4‐ c ]piperidines: 3‐Cyclobutoxy Linker as a Key Spacer for H 3 R Inverse Agonists
Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie‐Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van houtvin, Nathalie
Published in ChemMedChem (01.12.2012)
Published in ChemMedChem (01.12.2012)
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Journal Article
Lead Optimization of Thiazolo[5,4-c]piperidines: 3-Cyclobutoxy Linker as a Key Spacer for H3R Inverse Agonists
Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van houtvin, Nathalie
Published in ChemMedChem (01.12.2012)
Published in ChemMedChem (01.12.2012)
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Journal Article
Phenyl-oxazoles, a New Family of Inverse Agonists at the H3 Histamine Receptor
Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie-Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Provins, Laurent
Published in ChemMedChem (01.02.2010)
Published in ChemMedChem (01.02.2010)
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Journal Article
Acetamide Scanning around Bicyclic Thiazoles: SAR at the H 3 Receptor
Denonne , Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie‐Laure, Detrait, Eric, Durieu, Véronique, Gillard, Michel, Lamberty, Yves, Lorent, Geneviève, Nicolas, Jean‐Marie, Vanbellinghen, Alain, Van Houtvin, Nathalie, Provins, Laurent
Published in ChemMedChem (05.09.2011)
Published in ChemMedChem (05.09.2011)
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Journal Article
Phenyl‐oxazoles, a New Family of Inverse Agonists at the H 3 Histamine Receptor
Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie‐Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Provins, Laurent
Published in ChemMedChem (01.02.2010)
Published in ChemMedChem (01.02.2010)
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Journal Article
Acetamide Scanning around Bicyclic Thiazoles: SAR at the H3 Receptor
Denonne , Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Detrait, Eric, Durieu, Véronique, Gillard, Michel, Lamberty, Yves, Lorent, Geneviève, Nicolas, Jean-Marie, Vanbellinghen, Alain, Van Houtvin, Nathalie, Provins, Laurent
Published in ChemMedChem (05.09.2011)
Published in ChemMedChem (05.09.2011)
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Journal Article
Discovery of a New Class of Non‐imidazole Oxazoline‐Based Histamine H 3 Receptor (H 3 R) Inverse Agonists
Célanire, Sylvain, Wijtmans, Maikel, Christophe, Bernard, Collart, Philippe, de Esch, Iwan, Dassesse, Donald, Delaunoy, Christel, Denonne, Frédéric, Durieu, Véronique, Gelens, Edith, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lebon, Florence, Nicolas, Jean‐Marie, Quéré, Luc, Snip, Erwin, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Timmerman, Henk, Talaga, Patrice, Leurs, Rob, Provins, Laurent
Published in ChemMedChem (06.07.2009)
Published in ChemMedChem (06.07.2009)
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Journal Article
Lead optimization of thiazolo[5,4-c]piperidines: 3-cyclobutoxy linker as a key spacer for H(3)R inverse agonists
Provins, Laurent, Denonne, Frédéric, Célanire, Sylvain, Christophe, Bernard, Defays, Sabine, Delaunoy, Christel, Delporte, Marie-Laure, Demaude, Thierry, Durieu, Véronique, Gillard, Michel, Hubert, Delphine, Lamberty, Yves, Lorent, Geneviève, Valade, Anne, Vanbellinghen, Alain, Van Houtvin, Nathalie
Published in ChemMedChem (01.12.2012)
Published in ChemMedChem (01.12.2012)
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Journal Article
Discovery of a New Class of Non-imidazole Oxazoline-Based Histamine H3 Receptor (H3R) Inverse Agonists
Célanire, Sylvain, Wijtmans, Maikel, Christophe, Bernard, Collart, Philippe, de Esch, Iwan, Dassesse, Donald, Delaunoy, Christel, Denonne, Frédéric, Durieu, Véronique, Gelens, Edith, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lebon, Florence, Nicolas, Jean-Marie, Quéré, Luc, Snip, Erwin, Vanbellinghen, Alain, Van houtvin, Nathalie, Verbois, Valérie, Timmerman, Henk, Talaga, Patrice, Leurs, Rob, Provins, Laurent
Published in ChemMedChem (06.07.2009)
Published in ChemMedChem (06.07.2009)
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Journal Article
Phenyl-oxazoles, a new family of inverse agonists at the H(3) histamine receptor
Denonne, Frédéric, Atienzar, Franck, Célanire, Sylvain, Christophe, Bernard, Delannois, Frédérique, Delaunoy, Christel, Delporte, Marie-Laure, Durieu, Véronique, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lorent, Geneviève, Vanbellinghen, Alain, Van Houtvin, Nathalie, Verbois, Valérie, Provins, Laurent
Published in ChemMedChem (01.02.2010)
Published in ChemMedChem (01.02.2010)
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Journal Article
Discovery of a new class of non-imidazole oxazoline-based histamine H(3) receptor (H(3)R) inverse agonists
Célanire, Sylvain, Wijtmans, Maikel, Christophe, Bernard, Collart, Philippe, de Esch, Iwan, Dassesse, Donald, Delaunoy, Christel, Denonne, Frédéric, Durieu, Véronique, Gelens, Edith, Gillard, Michel, Lallemand, Bénédicte, Lamberty, Yves, Lebon, Florence, Nicolas, Jean-Marie, Quéré, Luc, Snip, Erwin, Vanbellinghen, Alain, Van Houtvin, Nathalie, Verbois, Valérie, Timmerman, Henk, Talaga, Patrice, Leurs, Rob, Provins, Laurent
Published in ChemMedChem (01.07.2009)
Published in ChemMedChem (01.07.2009)
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Journal Article