Comparative sequence specificities of human 72- and 92-kDa gelatinases (type IV collagenases) and PUMP (matrilysin)
Netzel-Arnett, Sarah, Sang, Qing Xiang, Moore, William G. I, Navre, Marc, Birkedal-Hansen, Henning, Van Wart, Harold E
Published in Biochemistry (Easton) (29.06.1993)
Published in Biochemistry (Easton) (29.06.1993)
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Role of His-224 in the Anomalous pH Dependence of Human Stromelysin-1
Holman, Christopher M, Kan, Chen-Chen, Gehring, Michael R, Van Wart, Harold E
Published in Biochemistry (Easton) (12.01.1999)
Published in Biochemistry (Easton) (12.01.1999)
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Understanding the P1‘ Specificity of the Matrix Metalloproteinases: Effect of S1‘ Pocket Mutations in Matrilysin and Stromelysin-1
Welch, Anthony R, Holman, Christopher M, Huber, Martin, Brenner, Mitchell C, Browner, Michelle F, Van Wart, Harold E
Published in Biochemistry (Easton) (06.08.1996)
Published in Biochemistry (Easton) (06.08.1996)
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Proteolysis Involving Matrix Metalloproteinase 13 (Collagenase‐3) Is Required for Chondrocyte Differentiation That Is Associated with Matrix Mineralization
Wu, C. William, Tchetina, Elena V., Mwale, Fackson, Hasty, Karen, Pidoux, Isabelle, Reiner, Agnes, Chen, Jeffrey, Van Wart, Harold E., Poole, A. Robin
Published in Journal of bone and mineral research (01.04.2002)
Published in Journal of bone and mineral research (01.04.2002)
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Hydrolysis of a Broad Spectrum of Extracellular Matrix Proteins by Human Macrophage Elastase
Gronski, Jr, T J, Martin, R L, Kobayashi, D K, Walsh, B C, Holman, M C, Huber, M, Van Wart, H E, Shapiro, S D
Published in The Journal of biological chemistry (02.05.1997)
Published in The Journal of biological chemistry (02.05.1997)
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Comparison of the Peroxidase Reaction Kinetics of Prostaglandin H Synthase-1 and -2
Lu, G, Tsai, A L, Van Wart, H E, Kulmacz, R J
Published in The Journal of biological chemistry (04.06.1999)
Published in The Journal of biological chemistry (04.06.1999)
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Design and synthesis of orally active inhibitors of TNF synthesis as anti-rheumatoid arthritis drugs
Chen, Jian Jeffrey, Dewdney, Nolan, Lin, Xiaohong, Martin, Robert L, Walker, Keith A.M, Huang, Jane, Chu, Frances, Eugui, Elsie, Mirkovich, Anna, Kim, Yong, Sarma, Keshab, Arzeno, Humberto, Van Wart, Harold E
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
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Amino acid derived sulfonamide hydroxamates as inhibitors of procollagen C-Proteinase: solid-Phase synthesis of ornithine analogues
Dankwardt, Sharon M., Martin, Robert L., Chan, Christine S., Van Wart, Harold E., Walker, Keith A.M., Delaet, Nancy G., Robinson, Leslie A.
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
Published in Bioorganic & medicinal chemistry letters (20.08.2001)
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Amino acid derived sulfonamide hydroxamates as inhibitors of procollagen C-proteinase. Part 2: Solid-phase optimization of side chains
DANKWARDT, Sharon M, ABBOT, Sarah C, BROKA, Chris A, MARTIN, Robert L, CHAN, Christine S, SPRINGMAN, Eric B, VAN WART, Harold E, WALKER, Keith A. M
Published in Bioorganic & medicinal chemistry letters (22.04.2002)
Published in Bioorganic & medicinal chemistry letters (22.04.2002)
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Mode of hydrolysis of collagen-like peptides by class I and class II Clostridium histolyticum collagenases: evidence for both endopeptidase and tripeptidylcarboxypeptidase activities
Mookhtiar, Kasim, Steinbrink, D. Randall, Van Wart, Harold E
Published in Biochemistry (Easton) (01.11.1985)
Published in Biochemistry (Easton) (01.11.1985)
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Solid-phase synthesis of di- and tripeptidic hydroxamic acids as inhibitors of procollagen C-proteinase
Dankwardt, Sharon M, Billedeau, Roland J, Lawley, Linda K, Abbot, Sarah C, Martin, Robert L, Chan, Christine S, Van Wart, Harold E, Walker, Keith A.M
Published in Bioorganic & medicinal chemistry letters (20.11.2000)
Published in Bioorganic & medicinal chemistry letters (20.11.2000)
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