A lymphatic-absorbed multi-targeted kinase inhibitor for myelofibrosis therapy
Ross, Brian D., Jang, Youngsoon, Welton, Amanda, Bonham, Christopher A., Palagama, Dilrukshika S. W., Heist, Kevin, Boppisetti, Jagadish, Imaduwage, Kasun P., Robison, Tanner, King, Leah R., Zhang, Edward Z., Amirfazli, Cyrus, Luker, Kathryn E., Lee, Winston Y., Luker, Gary D., Chenevert, Thomas L., Van Dort, Marcian E.
Published in Nature communications (17.08.2022)
Published in Nature communications (17.08.2022)
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In Vivo Targeting and Positron Emission Tomography Imaging of Tumor with Intrinsically Radioactive Metal–Organic Frameworks Nanomaterials
Chen, Daiqin, Yang, Dongzhi, Dougherty, Casey A, Lu, Weifei, Wu, Hongwei, He, Xianran, Cai, Ting, Van Dort, Marcian E, Ross, Brian D, Hong, Hao
Published in ACS nano (25.04.2017)
Published in ACS nano (25.04.2017)
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Inhibition of Furin/Proprotein Convertase-catalyzed Surface and Intracellular Processing by Small Molecules
Komiyama, Tomoko, Coppola, Julia M., Larsen, Martha J., van Dort, Marcian E., Ross, Brian D., Day, Robert, Rehemtulla, Alnawaz, Fuller, Robert S.
Published in The Journal of biological chemistry (05.06.2009)
Published in The Journal of biological chemistry (05.06.2009)
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Positron Emission Tomography/Magnetic Resonance Imaging of Glioblastoma Using a Functionalized Gadofullerene Nanoparticle
Chen, Daiqin, Zhou, Yue, Yang, Dongzhi, Guan, Mirong, Zhen, Mingming, Lu, Weifei, Van Dort, Marcian E, Ross, Brian D, Wang, Chunru, Shu, Chunying, Hong, Hao
Published in ACS applied materials & interfaces (19.06.2019)
Published in ACS applied materials & interfaces (19.06.2019)
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Targeted Imaging and Therapy of Brain Cancer Using Theranostic Nanoparticles
Bhojani, Mahaveer Swaroop, Van Dort, Marcian, Rehemtulla, Alnawaz, Ross, Brian D
Published in Molecular pharmaceutics (06.12.2010)
Published in Molecular pharmaceutics (06.12.2010)
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Dual inhibition of allosteric mitogen-activated protein kinase (MEK) and phosphatidylinositol 3-kinase (PI3K) oncogenic targets with a bifunctional inhibitor
Van Dort, Marcian E., Galbán, Stefanie, Wang, Hanxiao, Sebolt-Leopold, Judith, Whitehead, Christopher, Hong, Hao, Rehemtulla, Alnawaz, Ross, Brian D.
Published in Bioorganic & medicinal chemistry (01.04.2015)
Published in Bioorganic & medicinal chemistry (01.04.2015)
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Structural effects of morpholine replacement in ZSTK474 on Class I PI3K isoform inhibition: Development of novel MEK/PI3K bifunctional inhibitors
Van Dort, Marcian E., Jang, Youngsoon, Bonham, Christopher A., Heist, Kevin, Palagama, Dilrukshika S.W., McDonald, Lucas, Zhang, Edward Z., Chenevert, Thomas L., Luker, Gary D., Ross, Brian D.
Published in European journal of medicinal chemistry (05.02.2022)
Published in European journal of medicinal chemistry (05.02.2022)
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The kinase activity of the Ser/Thr kinase BUB1 promotes TGF-β signaling
Nyati, Shyam, Schinske-Sebolt, Katrina, Pitchiaya, Sethuramasundaram, Chekhovskiy, Katerina, Chator, Areeb, Chaudhry, Nauman, Dosch, Joseph, Van Dort, Marcian E, Varambally, Sooryanarayana, Kumar-Sinha, Chandan, Nyati, Mukesh Kumar, Ray, Dipankar, Walter, Nils G, Yu, Hongtao, Ross, Brian Dale, Rehemtulla, Alnawaz
Published in Science signaling (06.01.2015)
Published in Science signaling (06.01.2015)
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Discovery of Bifunctional Oncogenic Target Inhibitors against Allosteric Mitogen-Activated Protein Kinase (MEK1) and Phosphatidylinositol 3‑Kinase (PI3K)
Van Dort, Marcian E, Hong, Hao, Wang, Hanxiao, Nino, Charles A, Lombardi, Rachel L, Blanks, Avery E, Galbán, Stefanie, Ross, Brian D
Published in Journal of medicinal chemistry (24.03.2016)
Published in Journal of medicinal chemistry (24.03.2016)
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Engineered Antibody Fragment against the Urokinase Plasminogen Activator for Fast Delineation of Triple-Negative Breast Cancer by Positron Emission Tomography
Lu, Weifei, Cong, Yiyang, Yang, Dongzhi, Chen, Daiqin, Yang, Guoyu, Wang, Yi, Van Dort, Marcian E, Ross, Brian D, Mazar, Andrew P, Chu, Bei-Bei, Hong, Hao
Published in Molecular pharmaceutics (05.04.2021)
Published in Molecular pharmaceutics (05.04.2021)
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A Bifunctional MAPK/PI3K Antagonist for Inhibition of Tumor Growth and Metastasis
Galbán, Stefanie, Apfelbaum, April A, Espinoza, Carlos, Heist, Kevin, Haley, Henry, Bedi, Karan, Ljungman, Mats, Galbán, Craig J, Luker, Gary D, Dort, Marcian Van, Ross, Brian D
Published in Molecular cancer therapeutics (01.11.2017)
Published in Molecular cancer therapeutics (01.11.2017)
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Applications of Molecular Imaging
Galbán, Craig J., Galbán, Stefanie, Van Dort, Marcian E., Luker, Gary D., Bhojani, Mahaveer S., Rehemtulla, Alnawaz, Ross, Brian D.
Published in Molecular Biology of Cancer: Translation to the Clinic (2010)
Published in Molecular Biology of Cancer: Translation to the Clinic (2010)
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Book Chapter
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Design and Investigation of a [18F]-Labeled Benzamide Derivative as a High Affinity Dual Sigma Receptor Subtype Radioligand for Prostate Tumor Imaging
Yang, Dongzhi, Comeau, Anthony, Bowen, Wayne D, Mach, Robert H, Ross, Brian D, Hong, Hao, Van Dort, Marcian E
Published in Molecular pharmaceutics (06.03.2017)
Published in Molecular pharmaceutics (06.03.2017)
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Antibody-based PET of uPA/uPAR signaling with broad applicability for cancer imaging
Yang, Dongzhi, Severin, Gregory W, Dougherty, Casey A, Lombardi, Rachel, Chen, Daiqin, Van Dort, Marcian E, Barnhart, Todd E, Ross, Brian D, Mazar, Andrew P, Hong, Hao
Published in Oncotarget (08.11.2016)
Published in Oncotarget (08.11.2016)
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Ocular Toxicity Profile of ST-162 and ST-168 as Novel Bifunctional MEK/PI3K Inhibitors
Smith, Andrew, Pawar, Mercy, Van Dort, Marcian E, Galbán, Stefanie, Welton, Amanda R, Thurber, Greg M, Ross, Brian D, Besirli, Cagri G
Published in Journal of ocular pharmacology and therapeutics (01.07.2018)
Published in Journal of ocular pharmacology and therapeutics (01.07.2018)
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Structure-Guided Design and Initial Studies of a Bifunctional MEK/PI3K Inhibitor (ST-168)
Van Dort, Marcian E, Galbán, Stefanie, Nino, Charles A, Hong, Hao, Apfelbaum, April A, Luker, Gary D, Thurber, Greg M, Atangcho, Lydia, Besirli, Cagri G, Ross, Brian D
Published in ACS medicinal chemistry letters (10.08.2017)
Published in ACS medicinal chemistry letters (10.08.2017)
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Evaluation of treatment-associated inflammatory response on diffusion-weighted magnetic resonance imaging and 2-[18F]-fluoro-2-deoxy-D-glucose-positron emission tomography imaging biomarkers
Galbán, Craig J, Bhojani, Mahaveer S, Lee, Kuei C, Meyer, Charles R, Van Dort, Marcian E, Kuszpit, Kyle K, Koeppe, Robert A, Ranga, Rajesh, Moffat, Bradford A, Johnson, Timothy D, Chenevert, Thomas L, Rehemtulla, Alnawaz, Ross, Brian D
Published in Clinical cancer research (01.03.2010)
Published in Clinical cancer research (01.03.2010)
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