Neoceptor Concept Based on Molecular Complementarity in GPCRs: A Mutant Adenosine A3 Receptor with Selectively Enhanced Affinity for Amine-Modified Nucleosides
Jacobson, Kenneth A, Gao, Zhan-Guo, Chen, Aishe, Barak, Dov, Kim, Soon-Ai, Lee, Kyeong, Link, Andreas, Rompaey, Philippe Van, van Calenbergh, Serge, Liang, Bruce T
Published in Journal of medicinal chemistry (22.11.2001)
Published in Journal of medicinal chemistry (22.11.2001)
Get full text
Journal Article
Modulation of adenosine receptor affinity and intrinsic efficacy in adenine nucleosides substituted at the 2-position
Ohno, Michihiro, Gao, Zhan-Guo, Van Rompaey, Philippe, Tchilibon, Susanna, Kim, Soo-Kyung, Harris, Brian A, Gross, Ariel S, Duong, Heng T, Van Calenbergh, Serge, Jacobson, Kenneth A
Published in Bioorganic & medicinal chemistry (01.06.2004)
Published in Bioorganic & medicinal chemistry (01.06.2004)
Get full text
Journal Article
Mycobacterium tuberculosis Thymidine Monophosphate Kinase Inhibitors: Biological Evaluation and Conformational Analysis of 2′- and 3′-Modified Thymidine Analogues
Van Rompaey, Philippe, Nauwelaerts, Koen, Vanheusden, Veerle, Rozenski, Jef, Munier-Lehmann, Hélène, Herdewijn, Piet, Van Calenbergh, Serge
Published in European journal of organic chemistry (01.08.2003)
Published in European journal of organic chemistry (01.08.2003)
Get full text
Journal Article
Llama-derived Single Variable Domains (Nanobodies) Directed against Chemokine Receptor CXCR7 Reduce Head and Neck Cancer Cell Growth in Vivo
Maussang, David, Mujić-Delić, Azra, Descamps, Francis J., Stortelers, Catelijne, Vanlandschoot, Peter, Stigter-van Walsum, Marijke, Vischer, Henry F., van Roy, Maarten, Vosjan, Maria, Gonzalez-Pajuelo, Maria, van Dongen, Guus A.M.S., Merchiers, Pascal, van Rompaey, Philippe, Smit, Martine J.
Published in The Journal of biological chemistry (11.10.2013)
Published in The Journal of biological chemistry (11.10.2013)
Get full text
Journal Article
Modeling the Adenosine Receptors: Comparison of the Binding Domains of A2A Agonists and Antagonists
Kim, Soo-Kyung, Gao, Zhan-Guo, Van Rompaey, Philippe, Gross, Ariel S, Chen, Aishe, Van Calenbergh, Serge, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (06.11.2003)
Published in Journal of medicinal chemistry (06.11.2003)
Get full text
Journal Article
Orthogonal Activation of the Reengineered A3 Adenosine Receptor (Neoceptor) Using Tailored Nucleoside Agonists
Gao, Zhan-Guo, Duong, Heng T, Sonina, Tatiana, Kim, Soo-Kyung, Van Rompaey, Philippe, Van Calenbergh, Serge, Mamedova, Liaman, Kim, Hea Ok, Kim, Myong Jung, Kim, Ae Yil, Liang, Bruce T, Jeong, Lak Shin, Jacobson, Kenneth A
Published in Journal of medicinal chemistry (04.05.2006)
Published in Journal of medicinal chemistry (04.05.2006)
Get full text
Journal Article
Thymidine and thymidine-5′- O-monophosphate analogues as inhibitors of Mycobacterium tuberculosis thymidylate kinase
Vanheusden, Veerle, Van Rompaey, Philippe, Munier-Lehmann, Hélène, Pochet, Sylvie, Herdewijn, Piet, Van Calenbergh, Serge
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
Published in Bioorganic & medicinal chemistry letters (15.09.2003)
Get full text
Journal Article
Exploring human adenosine A3 receptor complementarity and activity for adenosine analogues modified in the ribose and purine moiety
VAN ROMPAEY, Philippe, JACOBSON, Kenneth A, GROSS, Ariel S, GAO, Zhan-Guo, VAN CALENBERGH, Serge
Published in Bioorganic & medicinal chemistry (15.02.2005)
Published in Bioorganic & medicinal chemistry (15.02.2005)
Get full text
Journal Article
Exploring human adenosine A 3 receptor complementarity and activity for adenosine analogues modified in the ribose and purine moiety
Van Rompaey, Philippe, Jacobson, Kenneth A., Gross, Ariel S., Gao, Zhan-Guo, Van Calenbergh, Serge
Published in Bioorganic & medicinal chemistry (2005)
Published in Bioorganic & medicinal chemistry (2005)
Get full text
Journal Article
Orthogonal Activation of the Reengineered A 3 Adenosine Receptor (Neoceptor) Using Tailored Nucleoside Agonists
Gao, Zhan-Guo, Duong, Heng T., Sonina, Tatiana, Kim, Soo-Kyung, Van Rompaey, Philippe, Van Calenbergh, Serge, Mamedova, Liaman, Kim, Hea Ok, Kim, Myong Jung, Kim, Ae Yil, Liang, Bruce T., Jeong, Lak Shin, Jacobson, Kenneth A.
Published in Journal of medicinal chemistry (01.05.2006)
Published in Journal of medicinal chemistry (01.05.2006)
Get full text
Journal Article
Modeling the Adenosine Receptors: Comparison of the Binding Domains of A 2A Agonists and Antagonists
Kim, Soo-Kyung, Gao, Zhan-Guo, Van Rompaey, Philippe, Gross, Ariel S., Chen, Aishe, Van Calenbergh, Serge, Jacobson, Kenneth A.
Published in Journal of medicinal chemistry (01.11.2003)
Published in Journal of medicinal chemistry (01.11.2003)
Get full text
Journal Article
METHOD FOR GENERATION OF IMMUNOGLOBULIN SEQUENCES
VAN ROMPAEY, PHILIPPE, ASSUNCAO, JOANA, NOLTE, FRIEDRICH, GONZALEZ, MARIA, LAEREMANS, TOON, STORTELERS, CATELIJNE
Year of Publication 24.01.2023
Get full text
Year of Publication 24.01.2023
Patent
Thymidine and thymidine-5'-O-monophosphate analogues as inhibitors of Mycobacterium tuberculosis thymidylate kinase: Recent advances in the design of kinase inhibitors as novel therapeutic agents
VANHEUSDEN, Veerle, VAN ROMPAEY, Philippe, MUNIER-LEHMANN, Hélène, POCHET, Sylvie, HERDEWIJN, Piet, VAN CALENBERGH, Serge
Published in Bioorganic & medicinal chemistry letters (2003)
Get full text
Published in Bioorganic & medicinal chemistry letters (2003)
Journal Article
Bispecific CXCR4-CD4 polypeptides with potent anti-HIV activity
Stortelers, Catelijne, Vanlandschoot, Peter, Schols, Dominique, Van Rompaey, Philippe, Soares, Hugo
Year of Publication 29.06.2021
Get full text
Year of Publication 29.06.2021
Patent
Bispecific CXCR4-CD-4 polypeptides with potent anti-HIV activity
Stortelers, Catelijne, Vanlandschoot, Peter, Schols, Dominique, Van Rompaey, Philippe, Soares, Hugo
Year of Publication 13.05.2021
Get full text
Year of Publication 13.05.2021
Patent
Neoceptor Concept Based on Molecular Complementarity in GPCRs: A Mutant Adenosine A 3 Receptor with Selectively Enhanced Affinity for Amine-Modified Nucleosides
Jacobson, Kenneth A., Gao, Zhan-Guo, Chen, Aishe, Barak, Dov, Kim, Soon-Ai, Lee, Kyeong, Link, Andreas, Rompaey, Philippe Van, van Calenbergh, Serge, Liang, Bruce T.
Published in Journal of medicinal chemistry (01.11.2001)
Published in Journal of medicinal chemistry (01.11.2001)
Get full text
Journal Article
BISPECIFIC CXCR4-CD4 POLYPEPTIDES WITH POTENT ANTI-HIV ACTIVITY
Stortelers, Catelijne, Vanlandschoot, Peter, Schols, Dominique, Van Rompaey, Philippe, Soares, Hugo
Year of Publication 26.09.2019
Get full text
Year of Publication 26.09.2019
Patent