Synthesis, Identification, and Structure–Activity Relationship Analysis of GATA4 and NKX2‑5 Protein–Protein Interaction Modulators
Jumppanen, Mikael, Kinnunen, Sini M, Välimäki, Mika J, Talman, Virpi, Auno, Samuli, Bruun, Tanja, Boije af Gennäs, Gustav, Xhaard, Henri, Aumüller, Ingo B, Ruskoaho, Heikki, Yli-Kauhaluoma, Jari
Published in Journal of medicinal chemistry (12.09.2019)
Published in Journal of medicinal chemistry (12.09.2019)
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Switching of hypertrophic signalling towards enhanced cardiomyocyte identity and maturity by a GATA4-targeted compound
Pohjolainen, Lotta, Kinnunen, Sini M, Auno, Samuli, Kiriazis, Alexandros, Pohjavaara, Saana, Kari-Koskinen, Julia, Zore, Matej, Jumppanen, Mikael, Yli-Kauhaluoma, Jari, Talman, Virpi, Ruskoaho, Heikki, Välimäki, Mika J
Published in Stem cell research & therapy (02.01.2024)
Published in Stem cell research & therapy (02.01.2024)
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Cardiac Actions of a Small Molecule Inhibitor Targeting GATA4–NKX2-5 Interaction
Kinnunen, Sini M., Tölli, Marja, Välimäki, Mika J., Gao, Erhe, Szabo, Zoltan, Rysä, Jaana, Ferreira, Mónica P. A., Ohukainen, Pauli, Serpi, Raisa, Correia, Alexandra, Mäkilä, Ermei, Salonen, Jarno, Hirvonen, Jouni, Santos, Hélder A., Ruskoaho, Heikki
Published in Scientific reports (15.03.2018)
Published in Scientific reports (15.03.2018)
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In vivo biocompatibility of porous silicon biomaterials for drug delivery to the heart
Tölli, Marja A, Ferreira, Mónica P.A, Kinnunen, Sini M, Rysä, Jaana, Mäkilä, Ermei M, Szabó, Zoltán, Serpi, Raisa E, Ohukainen, Pauli J, Välimäki, Mika J, Correia, Alexandra M.R, Salonen, Jarno J, Hirvonen, Jouni T, Ruskoaho, Heikki J, Santos, Hélder A
Published in Biomaterials (01.09.2014)
Published in Biomaterials (01.09.2014)
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GATA-targeted compounds modulate cardiac subtype cell differentiation in dual reporter stem cell line
Välimäki, Mika J, Leigh, Robert S, Kinnunen, Sini M, March, Alexander R, de Sande, Ana Hernández, Kinnunen, Matias, Varjosalo, Markku, Heinäniemi, Merja, Kaynak, Bogac L, Ruskoaho, Heikki
Published in Stem cell research & therapy (18.03.2021)
Published in Stem cell research & therapy (18.03.2021)
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Discovery of Small Molecules Targeting the Synergy of Cardiac Transcription Factors GATA4 and NKX2‑5
Välimäki, Mika J, Tölli, Marja A, Kinnunen, Sini M, Aro, Jani, Serpi, Raisa, Pohjolainen, Lotta, Talman, Virpi, Poso, Antti, Ruskoaho, Heikki J
Published in Journal of medicinal chemistry (28.09.2017)
Published in Journal of medicinal chemistry (28.09.2017)
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Domain-Independent Inhibition of CBP/p300 Attenuates α‑Synuclein Aggregation
Hlushchuk, Irena, Ruskoaho, Heikki, Domanskyi, Andrii, Airavaara, Mikko, Välimäki, Mika J
Published in ACS chemical neuroscience (07.07.2021)
Published in ACS chemical neuroscience (07.07.2021)
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Affinity chromatography reveals direct binding of the GATA4–NKX2-5 interaction inhibitor (3i-1000) with GATA4
Jumppanen, Mikael, Kinnunen, Sini M., Zore, Matej, Välimäki, Mika J., Talman, Virpi, Gennäs, Gustav Boije af, Ruskoaho, Heikki J., Yli-Kauhaluoma, Jari
Published in Scientific reports (18.04.2024)
Published in Scientific reports (18.04.2024)
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GATA4-targeted compound exhibits cardioprotective actions against doxorubicin-induced toxicity in vitro and in vivo: establishment of a chronic cardiotoxicity model using human iPSC-derived cardiomyocytes
Karhu, S. Tuuli, Kinnunen, Sini M., Tölli, Marja, Välimäki, Mika J., Szabó, Zoltán, Talman, Virpi, Ruskoaho, Heikki
Published in Archives of toxicology (01.06.2020)
Published in Archives of toxicology (01.06.2020)
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Stem cells are the most sensitive screening tool to identify toxicity of GATA4-targeted novel small-molecule compounds
Karhu, S. Tuuli, Välimäki, Mika J., Jumppanen, Mikael, Kinnunen, Sini M., Pohjolainen, Lotta, Leigh, Robert S., Auno, Samuli, Földes, Gábor, Boije af Gennäs, Gustav, Yli-Kauhaluoma, Jari, Ruskoaho, Heikki, Talman, Virpi
Published in Archives of toxicology (01.09.2018)
Published in Archives of toxicology (01.09.2018)
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Journal Article
Stem cells are the most sensitive screening tool to identify toxicity of GATA4- targeted small-molecule compounds
Karhu, Tuuli, Valimaki, Mika, Jumppanen, Mikael, Pohjolainen, Lotta, Leigh, Robert, Foldes, Gabor, Gennas, Gustav Boije Af, Yli-Kauhaluoma, Jari, Ruskoaho, Heikki, Talman, Virpi
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
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Journal Article
Discovery of Small Molecules Targeting the Synergy of Cardiac Transcription Factors GATA4 and NKX2-5
Ruskoaho, Heikki J, Aro, Jani, Serpi, Raisa, Pohjolainen, Lotta, Talman, Virpi, Poso, Antti, Rysa, Jaana, Kinnunen, Sini, Tolli, Marja, Valimaki, Mika
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
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The Acceptor and Site Specificity of α3-Fucosyltransferase V
Pykäri, Maria, Toivonen, Suvi, Natunen, Jari, Niemelä, Ritva, Salminen, Heidi, Aitio, Olli, Ekström, Minna, Parmanne, Pinja, Välimäki, Mika, Alais, Jocelyne, Augé, Claudine, Lowe, John B., Renkonen, Ossi, Renkonen, Risto
Published in The Journal of biological chemistry (01.12.2000)
Published in The Journal of biological chemistry (01.12.2000)
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Journal Article
ISOXAZOLE-AMIDES FOR TREATING CARDIAC DISEASES
BOIJE AF GENNÄS, Gustav, YLI-KAUHALUOMA, Jari, JUMPPANEN, Mikael, RUSKOAHO, Heikki, VÄLIMÄKI, Mika, KINNUNEN, Sini, TÖLLI, Marja
Year of Publication 29.03.2018
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Year of Publication 29.03.2018
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