Synthesis, Crystallization, and Biological Evaluation of an Orally Active Prodrug of Gemcitabine
Bender, David M, Bao, Jingqi, Dantzig, Anne H, Diseroad, William D, Law, Kevin L, Magnus, Nicholas A, Peterson, Jeffrey A, Perkins, Everett J, Pu, Yangwei J, Reutzel-Edens, Susan M, Remick, David M, Starling, James J, Stephenson, Gregory A, Vaid, Radhe K, Zhang, Deyi, McCarthy, James R
Published in Journal of medicinal chemistry (26.11.2009)
Published in Journal of medicinal chemistry (26.11.2009)
Get full text
Journal Article
Rapid Development and Scale-Up of a 1H-4-Substituted Imidazole Intermediate Enabled by Chemistry in Continuous Plug Flow Reactors
May, Scott A, Johnson, Martin D, Braden, Timothy M, Calvin, Joel R, Haeberle, Brian D, Jines, Amy R, Miller, Richard D, Plocharczyk, Edward F, Rener, Gregory A, Richey, Rachel N, Schmid, Christopher R, Vaid, Radhe K, Yu, Hannah
Published in Organic process research & development (18.05.2012)
Published in Organic process research & development (18.05.2012)
Get full text
Journal Article
A Practical Method for Functionalized Peptide or Amide Bond Formation in Aqueous−Ethanol Media with EDC as Activator
Pu, Yangwei John, Vaid, Radhe K, Boini, Sathish K, Towsley, Robert W, Doecke, Christopher W, Mitchell, David
Published in Organic process research & development (20.03.2009)
Published in Organic process research & development (20.03.2009)
Get full text
Journal Article
A Practical Synthesis of 2-{4-[4-Fluoro-3-(trifluoromethyl)phenyl]-2-(piperidin-4-yl)-1H-imidazol-1-yl}-N,N-dimethylethanamine
Vaid, Radhe K., Spitler, Jeremy, Boini, Sathish, Henry, Kenneth, Jiansheng, Xu, Gao, Baitao, Lu, Xiaoquan
Published in Synthesis (Stuttgart) (01.07.2012)
Published in Synthesis (Stuttgart) (01.07.2012)
Get more information
Journal Article
An Asymmetric Synthesis of a Chiral Sulfone Acid with Concomitant Hydrolysis and Oxidation to Enable the Preparation of a Glucokinase Activator
DeBaillie, Amy C, Magnus, Nicholas A, Laurila, Michael E, Wepsiec, James P, Ruble, J. Craig, Petkus, Jeffrey J, Vaid, Radhe K, Niemeier, Jeffry K, Mick, Joseph F, Gunter, Thomas Z
Published in Organic process research & development (21.09.2012)
Published in Organic process research & development (21.09.2012)
Get full text
Journal Article
Development of a Manufacturing Process for 1-(1-Pyridin-2-yl methyl-piperidin-4-yl)-1H-indole: A Key Intermediate for Protein Kinase C Inhibitor LY317615
Boini, Sathish, Moder, Kenneth P, Vaid, Radhe K, Kopach, Micheal, Kobierski, M
Published in Organic process research & development (17.11.2006)
Published in Organic process research & development (17.11.2006)
Get full text
Journal Article
Hypervalent iodine oxidation of silyl enol ethers under Lewis-acid conditions in methanol. A general route to .alpha.-methoxy ketones
Moriarty, Robert M, Prakash, Om, Duncan, Michael P, Vaid, Radhe K, Musallam, Hikmat A
Published in Journal of organic chemistry (01.01.1987)
Published in Journal of organic chemistry (01.01.1987)
Get full text
Journal Article
A novel intramolecular cyclopropanation using iodonium ylides
Moriarty, Robert M, Prakash, Om, Vaid, Radhe K, Zhao, Lei
Published in Journal of the American Chemical Society (01.08.1989)
Published in Journal of the American Chemical Society (01.08.1989)
Get full text
Journal Article
Process Development of (1S,2S,5R,6S)- Spiro[bicyclo[3.1.0]hexane-2‘,5‘-dioxo-2,4‘-imidazolidine]-6-carboxylic Acid, (R)-α-Methylbenzenemethanamine Salt (LSN344309)
Rasmy, Ossama M, Vaid, Radhe K, Semo, Michael J, Chelius, Erik C, Robey, Roger L, Alt, Charles A, Rhodes, Gary A, Vicenzi, Jeffery T
Published in Organic process research & development (01.01.2006)
Published in Organic process research & development (01.01.2006)
Get full text
Journal Article
Development and Production of an Enantioselective Tetrahydroisoquinoline Synthesis Enabled by Continuous Cryogenic Lithium–Halogen Exchange
Cole, Kevin P., Argentine, Mark D., Conder, Edward W., Vaid, Radhe K., Feng, Pengyao, Jia, Mo, Huang, Ping, Liu, Peng, Sun, Baoquan, Tadayon, Sam, Zhu, Cheng, Zhu, Ruiheng
Published in Organic process research & development (16.10.2020)
Published in Organic process research & development (16.10.2020)
Get full text
Journal Article
Rapid Development and Scale-Up of a 1 H -4-Substituted Imidazole Intermediate Enabled by Chemistry in Continuous Plug Flow Reactors
May, Scott A., Johnson, Martin D., Braden, Timothy M., Calvin, Joel R., Haeberle, Brian D., Jines, Amy R., Miller, Richard D., Plocharczyk, Edward F., Rener, Gregory A., Richey, Rachel N., Schmid, Christopher R., Vaid, Radhe K., Yu, Hannah
Published in Organic process research & development (18.05.2012)
Published in Organic process research & development (18.05.2012)
Get full text
Journal Article
HYPERVALENT IODINE OXIDATION OF AMINES USING IODOSOBENZENE - SYNTHESIS OF NITRILES, KETONES AND LACTAMS
MORIARTY, RM, VAID, RK, DUNCAN, MP, OCHIAI, M, INENAGA, M, NAGAO, Y
Published in Tetrahedron letters (01.01.1988)
Published in Tetrahedron letters (01.01.1988)
Get more information
Journal Article
Counterion effects in the preparation of aldehyde–bisulfite adducts
Kissane, Marie G., Frank, Scott A., Rener, Gregory A., Ley, Christopher P., Alt, Charles A., Stroud, Paul A., Vaid, Radhe K., Boini, Sathish K., McKee, Laura A., Vicenzi, Jeffrey T., Stephenson, Gregory A.
Published in Tetrahedron letters (27.11.2013)
Published in Tetrahedron letters (27.11.2013)
Get full text
Journal Article
ChemInform Abstract: Synthesis of Methyl 7,9-Dimethyl-5-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carboxylate and Its Analogues
Vaid, Radhe K., Boini, Sathish K., Alt, Charles A., Spitler, Jeremy T., Hadden, Chad E., Frank, Scott A., Moher, Eric D.
Published in ChemInform (01.03.2015)
Published in ChemInform (01.03.2015)
Get full text
Journal Article
Synthesis of Methyl 7,9-Dimethyl-5-oxo-2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carboxylate and Its Analogues
Vaid, Radhe K., Boini, Sathish K., Alt, Charles A., Spitler, Jeremy T., Hadden, Chad E., Frank, Scott A., Moher, Eric D.
Published in Synthesis (Stuttgart) (15.09.2014)
Published in Synthesis (Stuttgart) (15.09.2014)
Get more information
Journal Article
OXIDATIVE DECARBOXYLATION OF CYCLIC AMINO-ACIDS AND DEHYDROGENATION OF CYCLIC SECONDARY-AMINES WITH IODOSOBENZENE
OCHIAI, M, INENAGA, M, NAGAO, Y, MORIARTY, RM, VAID, RK, DUNCAN, MP
Published in Tetrahedron letters (01.01.1988)
Published in Tetrahedron letters (01.01.1988)
Get more information
Journal Article
Synthesis of (2-{4-[4-Fluoro-3-(trifluoromethyl)phenyl]-2-piperidin-4-yl-1H-imidazol-1-yl}ethyl)dimethylamine
Vaid, Radhe K., Boini, Sathish, Spitler, Jeremy T., Pu, Yangwei John, May, Scott A., Yu, Hannah, Wu Sizhong, Fu, Jie, Zhang, Guoliang
Published in Synthesis (Stuttgart) (03.06.2013)
Published in Synthesis (Stuttgart) (03.06.2013)
Get more information
Journal Article