O-GlcNAcylation Regulates Cancer Metabolism and Survival Stress Signaling via Regulation of the HIF-1 Pathway
Ferrer, Christina M., Lynch, Thomas P., Sodi, Valerie L., Falcone, John N., Schwab, Luciana P., Peacock, Danielle L., Vocadlo, David J., Seagroves, Tiffany N., Reginato, Mauricio J.
Published in Molecular cell (05.06.2014)
Published in Molecular cell (05.06.2014)
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Monitoring and modulating O-GlcNAcylation: assays and inhibitors of O-GlcNAc processing enzymes
Alteen, Matthew G, Tan, Hong Yee, Vocadlo, David J
Published in Current opinion in structural biology (01.06.2021)
Published in Current opinion in structural biology (01.06.2021)
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The primary familial brain calcification-associated protein MYORG is an α-galactosidase with restricted substrate specificity
Meek, Richard W., Brockerman, Jacob, Fordwour, Osei B., Zandberg, Wesley F., Davies, Gideon J., Vocadlo, David J.
Published in PLoS biology (01.09.2022)
Published in PLoS biology (01.09.2022)
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O-GlcNAc occurs cotranslationally to stabilize nascent polypeptide chains
Zhu, Yanping, Liu, Ta-Wei, Cecioni, Samy, Eskandari, Razieh, Zandberg, Wesley F, Vocadlo, David J
Published in Nature chemical biology (01.05.2015)
Published in Nature chemical biology (01.05.2015)
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Discovery of MK-8719, a Potent O‑GlcNAcase Inhibitor as a Potential Treatment for Tauopathies
Selnick, Harold G, Hess, J. Fred, Tang, Cuyue, Liu, Kun, Schachter, Joel B, Ballard, Jeanine E, Marcus, Jacob, Klein, Daniel J, Wang, Xiaohai, Pearson, Michelle, Savage, Mary J, Kaul, Ramesh, Li, Tong-Shuang, Vocadlo, David J, Zhou, Yuanxi, Zhu, Yongbao, Mu, Changwei, Wang, Yaode, Wei, Zhongyong, Bai, Chang, Duffy, Joseph L, McEachern, Ernest J
Published in Journal of medicinal chemistry (27.11.2019)
Published in Journal of medicinal chemistry (27.11.2019)
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Hijacking a biosynthetic pathway yields a glycosyltransferase inhibitor within cells
Vocadlo, David J, Gloster, Tracey M, Zandberg, Wesley F, Heinonen, Julia E, Shen, David L, Deng, Lehua
Published in Nature chemical biology (01.03.2011)
Published in Nature chemical biology (01.03.2011)
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HCF-1 is cleaved in the active site of O-GlcNAc transferase
Lazarus, Michael B, Jiang, Jiaoyang, Kapuria, Vaibhav, Bhuiyan, Tanja, Janetzko, John, Zandberg, Wesley F, Vocadlo, David J, Herr, Winship, Walker, Suzanne
Published in Science (American Association for the Advancement of Science) (06.12.2013)
Published in Science (American Association for the Advancement of Science) (06.12.2013)
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Targeting neuronal lysosomal dysfunction caused by β-glucocerebrosidase deficiency with an enzyme-based brain shuttle construct
Gehrlein, Alexandra, Udayar, Vinod, Anastasi, Nadia, Morella, Martino L, Ruf, Iris, Brugger, Doris, von der Mark, Sophia, Thoma, Ralf, Rufer, Arne, Heer, Dominik, Pfahler, Nina, Jochner, Anton, Niewoehner, Jens, Wolf, Luise, Fueth, Matthias, Ebeling, Martin, Villaseñor, Roberto, Zhu, Yanping, Deen, Matthew C, Shan, Xiaoyang, Ehsaei, Zahra, Taylor, Verdon, Sidransky, Ellen, Vocadlo, David J, Freskgård, Per-Ola, Jagasia, Ravi
Published in Nature communications (12.04.2023)
Published in Nature communications (12.04.2023)
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Bicyclic Picomolar OGA Inhibitors Enable Chemoproteomic Mapping of Its Endogenous Post-translational Modifications
González-Cuesta, Manuel, Sidhu, Peter, Ashmus, Roger A, Males, Alexandra, Proceviat, Cameron, Madden, Zarina, Rogalski, Jason C, Busmann, Jil A, Foster, Leonard J, García Fernández, José M, Davies, Gideon J, Ortiz Mellet, Carmen, Vocadlo, David J
Published in Journal of the American Chemical Society (19.01.2022)
Published in Journal of the American Chemical Society (19.01.2022)
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Differential effects of an O-GlcNAcase inhibitor on tau phosphorylation
Yu, Yang, Zhang, Lan, Li, Xiaojing, Run, Xiaoqin, Liang, Zhihou, Li, Yi, Liu, Ying, Lee, Moon H, Grundke-Iqbal, Inge, Iqbal, Khalid, Vocadlo, David J, Liu, Fei, Gong, Cheng-Xin
Published in PloS one (19.04.2012)
Published in PloS one (19.04.2012)
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Drosophila O-GlcNAc transferase (OGT) is encoded by the Polycomb group (PcG) gene, super sex combs (sxc)
Sinclair, Donald A.R, Syrzycka, Monika, Macauley, Matthew S, Rastgardani, Tara, Komljenovic, Ivana, Vocadlo, David J, Brock, Hugh W, Honda, Barry M
Published in Proceedings of the National Academy of Sciences - PNAS (11.08.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (11.08.2009)
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A Direct Fluorescent Activity Assay for Glycosyltransferases Enables Convenient High‐Throughput Screening: Application to O‐GlcNAc Transferase
Alteen, Matthew G., Gros, Christina, Meek, Richard W., Cardoso, David A., Busmann, Jil A., Sangouard, Gontran, Deen, Matthew C., Tan, Hong‐Yee, Shen, David L., Russell, Cecilia C., Davies, Gideon J., Robinson, Phillip J., McCluskey, Adam, Vocadlo, David J.
Published in Angewandte Chemie International Edition (08.06.2020)
Published in Angewandte Chemie International Edition (08.06.2020)
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Substrate-Guided Front-Face Reaction Revealed by Combined Structural Snapshots and Metadynamics for the Polypeptide N-Acetylgalactosaminyltransferase 2
Lira-Navarrete, Erandi, Iglesias-Fernández, Javier, Zandberg, Wesley F., Compañón, Ismael, Kong, Yun, Corzana, Francisco, Pinto, B. Mario, Clausen, Henrik, Peregrina, Jesús M., Vocadlo, David J., Rovira, Carme, Hurtado-Guerrero, Ramon
Published in Angewandte Chemie (International ed.) (28.07.2014)
Published in Angewandte Chemie (International ed.) (28.07.2014)
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