Exploiting a water network to achieve enthalpy-driven, bromodomain-selective BET inhibitors
Shadrick, William R., Slavish, Peter J., Chai, Sergio C., Waddell, Brett, Connelly, Michele, Low, Jonathan A., Tallant, Cynthia, Young, Brandon M., Bharatham, Nagakumar, Knapp, Stefan, Boyd, Vincent A., Morfouace, Marie, Roussel, Martine F., Chen, Taosheng, Lee, Richard E., Kiplin Guy, R., Shelat, Anang A., Potter, Philip M.
Published in Bioorganic & medicinal chemistry (01.01.2018)
Published in Bioorganic & medicinal chemistry (01.01.2018)
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Journal Article
A High-Throughput Screen Reveals New Small-Molecule Activators and Inhibitors of Pantothenate Kinases
Sharma, Lalit Kumar, Leonardi, Roberta, Lin, Wenwei, Boyd, Vincent A, Goktug, Asli, Shelat, Anang A, Chen, Taosheng, Jackowski, Suzanne, Rock, Charles O
Published in Journal of medicinal chemistry (12.02.2015)
Published in Journal of medicinal chemistry (12.02.2015)
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Journal Article
Bromodomain-Selective BET Inhibitors Are Potent Antitumor Agents against MYC-Driven Pediatric Cancer
Slavish, P Jake, Chi, Liying, Yun, Mi-Kyung, Tsurkan, Lyudmila, Martinez, Nancy E, Jonchere, Barbara, Chai, Sergio C, Connelly, Michele, Waddell, M Brett, Das, Sourav, Neale, Geoffrey, Li, Zhenmei, Shadrick, William R, Olsen, Rachelle R, Freeman, Kevin W, Low, Jonathan A, Price, Jeanine E, Young, Brandon M, Bharatham, Nagakumar, Boyd, Vincent A, Yang, Jun, Lee, Richard E, Morfouace, Marie, Roussel, Martine F, Chen, Taosheng, Savic, Daniel, Guy, R Kiplin, White, Stephen W, Shelat, Anang A, Potter, Philip M
Published in Cancer research (Chicago, Ill.) (01.09.2020)
Published in Cancer research (Chicago, Ill.) (01.09.2020)
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Journal Article
Targeting Histone Demethylases in MYC-Driven Neuroblastomas with Ciclopirox
Yang, Jun, Milasta, Sandra, Hu, Dongli, AlTahan, Alaa M, Interiano, Rodrigo B, Zhou, Junfang, Davidson, Jesse, Low, Jonathan, Lin, Wenwei, Bao, Ju, Goh, Pollyanna, Nathwani, Amit C, Wang, Ruoning, Wang, Yingdi, Ong, Su Sien, Boyd, Vincent A, Young, Brandon, Das, Sourav, Shelat, Anang, Wu, Yinan, Li, Zhenmei, Zheng, Jie J, Mishra, Ashutosh, Cheng, Yong, Qu, Chunxu, Peng, Junmin, Green, Douglas R, White, Stephen, Guy, R Kiplin, Chen, Taosheng, Davidoff, Andrew M
Published in Cancer research (Chicago, Ill.) (01.09.2017)
Published in Cancer research (Chicago, Ill.) (01.09.2017)
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Journal Article
Tissue Penetration of a Novel Spectinamide Antibiotic for the Treatment of Tuberculosis
Madhura, Dora Babu, Trivedi, Ashit, Liu, Jiuyu, Boyd, Vincent A., Jeffries, Cynthia, Loveless, Vivian, Lee, Richard E., Meibohm, Bernd
Published in The AAPS journal (01.05.2016)
Published in The AAPS journal (01.05.2016)
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Journal Article
Identification and Characterization of an Allosteric Inhibitory Site on Dihydropteroate Synthase
Hammoudeh, Dalia I, Daté, Mihir, Yun, Mi-Kyung, Zhang, Weixing, Boyd, Vincent A, Viacava Follis, Ariele, Griffith, Elizabeth, Lee, Richard E, Bashford, Donald, White, Stephen W
Published in ACS chemical biology (20.06.2014)
Published in ACS chemical biology (20.06.2014)
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Journal Article
Structure−Activity Relationships of Substituted 1-Pyridyl-2-phenyl-1,2-ethanediones: Potent, Selective Carboxylesterase Inhibitors
Young, Brandon M, Hyatt, Janice L, Bouck, David C, Chen, Taosheng, Hanumesh, Parimala, Price, Jeanine, Boyd, Vincent A, Potter, Philip M, Webb, Thomas R
Published in Journal of medicinal chemistry (23.12.2010)
Published in Journal of medicinal chemistry (23.12.2010)
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Journal Article
Evaluation of Diarylureas for Activity Against Plasmodium falciparum
Zhang, Yiqun, Anderson, Marc, Weisman, Jennifer L, Lu, Min, Choy, Cindy J, Boyd, Vincent A, Price, Jeanine, Sigal, Martina, Clark, Julie, Connelly, Michele, Zhu, Fangyi, Guiguemde, W. Armand, Jeffries, Cynthia, Yang, Lei, Lemoff, Andrew, Liou, Ally P, Webb, Thomas R, DeRisi, Joseph L, Guy, R. Kiplin
Published in ACS medicinal chemistry letters (09.12.2010)
Published in ACS medicinal chemistry letters (09.12.2010)
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Journal Article
Radiosynthesis of antitumor spliceosome modulators
Goronga, Tinopiwa, Boyd, Vincent A., Lagisetti, Chandraiah, Jeffries, Cynthia, Webb, Thomas R.
Published in Applied radiation and isotopes (01.09.2011)
Published in Applied radiation and isotopes (01.09.2011)
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Journal Article
Preparation of 2-deoxy-.beta.-C-arylglycosides and C-arylglycals from carbohydrate lactones
Boyd, Vincent A, Drake, Brian E, Sulikowski, Gary A
Published in Journal of organic chemistry (01.05.1993)
Published in Journal of organic chemistry (01.05.1993)
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Journal Article
Pyrimidinone conjugates for the assignment of the absolute configuration of α-chiral carboxylic acids by 1H-NMR
Murray, Robert S., Boyd, Vincent A., Lynch, Vincent M., Negrete, George R.
Published in ARKIVOC (22.03.2002)
Published in ARKIVOC (22.03.2002)
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PROPIONIC ACID DERIVATIVES AND METHODS OF USE THEREOF
THRASH, Thomas, P, BIEDIGER, Ronald, J, BOYD, Vincent, A, YOUNG, Brandon, M, BENISH, Michele, A, HARDY, Lindsay, Bonner, MARKET, Robert, V
Year of Publication 25.09.2024
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Year of Publication 25.09.2024
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PROPIONSYRE-DERIVATER OG DERES ANVENDELSESFORMÅL
THRASH, Thomas, P, BIEDIGER, Ronald, J, BOYD, Vincent, A, YOUNG, Brandon, M, BENISH, Michele, A, HARDY, Lindsay, Bonner, MARKET, Robert, V
Year of Publication 19.02.2024
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Year of Publication 19.02.2024
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PROPIONIC ACID DERIVATIVES AND METHODS OF USE THEREOF
THRASH, Thomas, P, BIEDIGER, Ronald, J, BOYD, Vincent, A, YOUNG, Brandon, M, BENISH, Michele, A, HARDY, Lindsay, Bonner, MARKET, Robert, V
Year of Publication 22.11.2023
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Year of Publication 22.11.2023
Patent
Tetrahydroquinoline-based bromodomain inhibitors
Boyd, Vincent A, Shelat, Anang, Shadrick, William Robert, Slavish, P Jake, Guy, R. Kip, Bharatham, Nagakumar, Young, Brandon M, Price, Jeanine E
Year of Publication 17.10.2023
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Year of Publication 17.10.2023
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