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Published in Journal of medicinal chemistry (24.12.2009)
Published in Journal of medicinal chemistry (24.12.2009)
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Discovery of a Bromodomain and Extraterminal Inhibitor with a Low Predicted Human Dose through Synergistic Use of Encoded Library Technology and Fragment Screening
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Published in Journal of medicinal chemistry (23.01.2020)
Published in Journal of medicinal chemistry (23.01.2020)
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NAV1.8 억제제로서의 2,3-디히드로퀴나졸린 화합물
VIMAL MYTHILY, GUANG JIE, HO MING HSUN, HOANG TRAM H, YING MABEN, MILLER WILLIAM H, ELBAN MARK, WASHBURN DAVID G, DAVIS RODERICK S, ROMANO JOSEPH J
Year of Publication 10.03.2022
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Year of Publication 10.03.2022
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Exploring the SAR of the β‑Ketoacyl-ACP Synthase Inhibitor GSK3011724A and Optimization around a Genotoxic Metabolite
Cunningham, Fraser, Esquivias, Jorge, Fernández-Menéndez, Raquel, Pérez, Arancha, Guardia, Ana, Escribano, Jaime, Rivero, Cristina, Vimal, Mythily, Cacho, Mónica, de Dios-Antón, Paco, Martínez-Martínez, María Santos, Jiménez, Elena, Huertas Valentín, Leticia, Rebollo-López, María José, López-Román, Eva María, Sousa-Morcuende, Verónica, Rullas, Joaquín, Neu, Margaret, Chung, Chun-wa, Bates, Robert H
Published in ACS infectious diseases (08.05.2020)
Published in ACS infectious diseases (08.05.2020)
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Synthesis and structure-activity relationships of a series of (1H-pyrazol-4-yl)acetamide antagonists of the P2X7 receptor
CHAMBERS, Laura J, STEVENS, Alexander J, THEOBALD, Pam J, BESWICK, Paul J, GLEAVE, Robert J, ROMAN, Shilina A, SENGER, Stefan, MOSES, Andrew P, MICHEL, Anton D, WALTER, Daryl S, DAVIES, David J, LIVERMORE, David G, FONFRIA, Elena, DEMONT, Emmanuel H, VIMAL, Mythily
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
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The identification a novel, selective, non-steroidal, functional glucocorticoid receptor antagonist
Rimland, Joseph, Dunne, Angela, Hunjan, Suchete S., Sasse, Rosemary, Uings, Iain, Montanari, Dino, Caivano, Matilde, Shah, Poonam, Standing, David, Gray, David, Brown, David, Cairns, William, Trump, Ryan, Smith, Paul W., Bertheleme, Nicolas, D’Alessandro, Pier, Gul, Sheraz, Vimal, Mythily, Smith, David N., Watson, Stephen P.
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
Published in Bioorganic & medicinal chemistry letters (01.04.2010)
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Synthesis and structure-activity relationships of a series of (1H-pyrazol-4-yl)acetamide antagonists of the P2X sub(7) receptor
Chambers, Laura J, Stevens, Alexander J, Moses, Andrew P, Michel, Anton D, Walter, Daryl S, Davies, David J, Livermore, David G, Fonfria, Elena, Demont, Emmanuel H, Vimal, Mythily, Theobald, Pam J, Beswick, Paul J, Gleave, Robert J, Roman, Shilina A, Senger, Stefan
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
Published in Bioorganic & medicinal chemistry letters (15.05.2010)
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Journal Article
Synthesis and structure–activity relationships of a series of (1 H-pyrazol-4-yl)acetamide antagonists of the P2X 7 receptor
Chambers, Laura J., Stevens, Alexander J., Moses, Andrew P., Michel, Anton D., Walter, Daryl S., Davies, David J., Livermore, David G., Fonfria, Elena, Demont, Emmanuel H., Vimal, Mythily, Theobald, Pam J., Beswick, Paul J., Gleave, Robert J., Roman, Shilina A., Senger, Stefan
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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2,3-dihydroquinazolin compounds as NAV1.8 inhibitors
Jie GUANG, Mark ELBAN, Maben YING, William H. MILLER, Joseph J. ROMANO, David G. WASHBURN, Tram H. HOANG, Ming-Hsun HO, Roderick S. DAVIS, Mythily VIMAL
Year of Publication 14.12.2023
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Year of Publication 14.12.2023
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Compuestos 2,3-dihidroquinazolin como inhibidores nav1 .8
HOANG, Tram H, MILLER, William H, ELBAN, Mark, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 21.04.2023
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Year of Publication 21.04.2023
Patent
2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS
ELBAN, Mark, HOANG, Tram H, MILLER, William H, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 06.04.2023
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Year of Publication 06.04.2023
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2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS
HOANG, Tram H, MILLER, William H, ELBAN, Mark, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 04.05.2022
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Year of Publication 04.05.2022
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COMPOSÉS 2,3-DIHYDROQUINAZOLINE EN TANT QU'INHIBITEURS DE NAV1.8
ELBAN, Mark, HOANG, Tram H, MILLER, William H, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 04.05.2022
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Year of Publication 04.05.2022
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2,3-dihydroquinazolin compounds as NAV1.8 inhibitors
HOANG, Tram H, MILLER, William H, ELBAN, Mark, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 27.01.2022
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Year of Publication 27.01.2022
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Split-split. A multiple synthesiser approach to efficient automated parallel synthesis
Brooking, Paul, Doran, Andrew, Grimsey, Paul, Hird, Nicholas W., MacLachlan, William S., Vimal, Mythily
Published in Tetrahedron letters (12.02.1999)
Published in Tetrahedron letters (12.02.1999)
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2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS
ROMANO, JOSEPH J, GUANG, JIE, ELBAN, MARK, YING, MABEN, HOANG, TRAM H, HO, MING-HSUN, VIMAL, MYTHILY, MILLER, WILLIAM H, DAVIS, RODERICK S, WASHBURN, DAVID G
Year of Publication 30.12.2020
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Year of Publication 30.12.2020
Patent
2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS
HOANG, Tram H, MILLER, William H, ELBAN, Mark, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 30.12.2020
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Year of Publication 30.12.2020
Patent
Blockade of human and porcine myocardial 5-HT4 receptors by SB 203186
Parker, S G, Taylor, E M, Hamburger, S A, Vimal, M, Kaumann, A J
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.12.1995)
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.12.1995)
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Journal Article
2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS
ELBAN Mark, GUANG Jie, ROMANO Joseph J, WASHBURN David G, HO Ming - Hsun, VIMAL Mythily, YING Maben, DAVIS Roderick S, HOANG Tram H, MILLER William H
Year of Publication 16.02.2022
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Year of Publication 16.02.2022
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2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS
HO MING-HSUN, VIMAL MYTHILY, HWANG TAE H, GUANG JIE, YING MABEN, MILLER WILLIAM H, ELBAN MARK, WASHBURN DAVID G, DAVIS RODERICK S, ROMANO JOSEPH J
Year of Publication 11.02.2022
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Year of Publication 11.02.2022
Patent