Structural insights into probe-dependent positive allosterism of the GLP-1 receptor
Bueno, Ana B., Sun, Bingfa, Willard, Francis S., Feng, Dan, Ho, Joseph D., Wainscott, David B., Showalter, Aaron D., Vieth, Michal, Chen, Qi, Stutsman, Cynthia, Chau, Betty, Ficorilli, James, Agejas, Francisco J., Cumming, Graham R., Jiménez, Alma, Rojo, Isabel, Kobilka, Tong Sun, Kobilka, Brian K., Sloop, Kyle W.
Published in Nature chemical biology (01.10.2020)
Published in Nature chemical biology (01.10.2020)
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Journal Article
Identification of tyrosine kinase inhibitors that halt Plasmodium falciparum parasitemia
Kesely, Kristina, Noomuna, Panae, Vieth, Michal, Hipskind, Philip, Haldar, Kasturi, Pantaleo, Antonella, Turrini, Francesco, Low, Philip S
Published in PloS one (12.11.2020)
Published in PloS one (12.11.2020)
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Journal Article
Molecular Basis for Necitumumab Inhibition of EGFR Variants Associated with Acquired Cetuximab Resistance
Bagchi, Atrish, Haidar, Jaafar N, Eastman, Scott W, Vieth, Michal, Topper, Michael, Iacolina, Michelle D, Walker, Jason M, Forest, Amelie, Shen, Yang, Novosiadly, Ruslan D, Ferguson, Kathryn M
Published in Molecular cancer therapeutics (01.02.2018)
Published in Molecular cancer therapeutics (01.02.2018)
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Journal Article
Crystal structure of human RIOK2 bound to a specific inhibitor
Wang, Jing, Varin, Thibault, Vieth, Michal, Elkins, Jonathan M
Published in Open biology (01.04.2019)
Published in Open biology (01.04.2019)
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Journal Article
A high-throughput screen against pantothenate synthetase (PanC) identifies 3-biphenyl-4-cyanopyrrole-2-carboxylic acids as a new class of inhibitor with activity against Mycobacterium tuberculosis
Kumar, Anuradha, Casey, Allen, Odingo, Joshua, Kesicki, Edward A, Abrahams, Garth, Vieth, Michal, Masquelin, Thierry, Mizrahi, Valerie, Hipskind, Philip A, Sherman, David R, Parish, Tanya
Published in PloS one (07.11.2013)
Published in PloS one (07.11.2013)
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Journal Article
What general conclusions can we draw from kinase profiling data sets?
Sutherland, Jeffrey J., Gao, Cen, Cahya, Suntara, Vieth, Michal
Published in Biochimica et biophysica acta (01.07.2013)
Published in Biochimica et biophysica acta (01.07.2013)
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Journal Article
Reconstruction of 3D structures of MET antibodies from electron microscopy 2D class averages
Chen, Qi, Vieth, Michal, Timm, David E, Humblet, Christine, Schneidman-Duhovny, Dina, Chemmama, Ilan E, Sali, Andrej, Zeng, Wei, Lu, Jirong, Liu, Ling
Published in PloS one (13.04.2017)
Published in PloS one (13.04.2017)
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Journal Article
Characteristic Physical Properties and Structural Fragments of Marketed Oral Drugs
Vieth, Michal, Siegel, Miles G, Higgs, Richard E, Watson, Ian A, Robertson, Daniel H, Savin, Kenneth A, Durst, Gregory L, Hipskind, Philip A
Published in Journal of medicinal chemistry (01.01.2004)
Published in Journal of medicinal chemistry (01.01.2004)
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Journal Article
Kinomics: characterizing the therapeutically validated kinase space
Vieth, Michal, Sutherland, Jeffrey J., Robertson, Daniel H., Campbell, Robert M.
Published in Drug discovery today (15.06.2005)
Published in Drug discovery today (15.06.2005)
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Journal Article
Kinomics—structural biology and chemogenomics of kinase inhibitors and targets
Vieth, Michal, Higgs, Richard E., Robertson, Daniel H., Shapiro, Michael, Gragg, Ellen A., Hemmerle, Horst
Published in BBA - Proteins and Proteomics (11.03.2004)
Published in BBA - Proteins and Proteomics (11.03.2004)
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Book Review
Journal Article
Novel route to the synthesis of 4-quinolyl isothiocyanates
Zhong, Boyu, Al-Awar, Rima S., Shih, Chuan, Grimes, John H., Vieth, Michal, Hamdouchi, Chafiq
Published in Tetrahedron letters (27.03.2006)
Published in Tetrahedron letters (27.03.2006)
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Journal Article
Assessing search strategies for flexible docking
Vieth, Michal, Hirst, Jonathan D., Dominy, Brian N., Daigler, Heidi, Brooks III, Charles L.
Published in Journal of computational chemistry (15.11.1998)
Published in Journal of computational chemistry (15.11.1998)
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Journal Article
Predicting the Conformational Variability of Abl Tyrosine Kinase using Molecular Dynamics Simulations and Markov State Models
Meng, Yilin, Gao, Cen, Clawson, David K, Atwell, Shane, Russell, Marijane, Vieth, Michal, Roux, Benoît
Published in Journal of chemical theory and computation (08.05.2018)
Published in Journal of chemical theory and computation (08.05.2018)
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Journal Article
Structural determinants of dual incretin receptor agonism by tirzepatide
Sun, Bingfa, Willard, Francis S, Feng, Dan, Alsina-Fernandez, Jorge, Chen, Qi, Vieth, Michal, Ho, Joseph D, Showalter, Aaron D, Stutsman, Cynthia, Ding, Liyun, Suter, Todd M, Dunbar, James D, Carpenter, John W, Mohammed, Faiz Ahmad, Aihara, Eitaro, Brown, Robert A, Bueno, Ana B, Emmerson, Paul J, Moyers, Julie S, Kobilka, Tong Sun, Coghlan, Matthew P, Kobilka, Brian K, Sloop, Kyle W
Published in Proceedings of the National Academy of Sciences - PNAS (29.03.2022)
Published in Proceedings of the National Academy of Sciences - PNAS (29.03.2022)
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Journal Article